Indazole: a medicinally important heterocyclic moiety

Synthesis and SAR of 4-aryl-1-(indazol-5-yl)pyridin-2(1H)ones as MCH-1 antagonists for the treatment of obesity

(2010) Mark Hadden et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

5-Piperazinyl-3-sulfonylindazoles as Potent and Selective 5-Hydroxytryptamine-6 Antagonists

(2010) Kevin G. Liu et al.   JOURNAL OF MEDICINAL CHEMISTRY

Discovery of (3S,3aR)-2-(3-Chloro-4-cyanophenyl)-3-cyclopentyl-3,3a,4,5-tetrahydro-2H-benzo[g]indazole-7-carboxylic Acid (PF-3882845), an Orally Efficacious Mineralocorticoid Receptor (MR) Antagonist for Hypertension and Nephropathy

(2010) Marvin J. Meyers et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of 3-[(N-carboalkoxy)ethylamino]-indazole-dione derivatives and their biological activities on human liver carbonyl reductase

(2009) Solomon Berhe et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, antimicrobial activity and QSAR studies of new 2,3-disubstituted-3,3a,4,5,6,7-hexahydro-2H-indazoles

(2009) Maninder Minu et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and biological evaluation of substituted 2-phenyl-2H-indazole-7-carboxamides as potent poly(ADP-ribose) polymerase (PARP) inhibitors

(2009) Rita Scarpelli et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Discovery of 2-{4-[(3S)-Piperidin-3-yl]phenyl}-2H-indazole-7-carboxamide (MK-4827): A Novel Oral Poly(ADP-ribose)polymerase (PARP) Inhibitor Efficacious in BRCA-1 and -2 Mutant Tumors

(2009) Philip Jones et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and biological evaluation of 3,5-diaminoindazoles as cyclin-dependent kinase inhibitors

(2008) Jinho Lee et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and antiproliferative activity of 3-amino-N-phenyl-1H-indazole-1-carboxamides

(2008) Demetrio Raffa et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Identification of (R)-1-(5-tert-Butyl-2,3-dihydro-1H-inden-1-yl)-3-(1H-indazol-4-yl)urea (ABT-102) as a Potent TRPV1 Antagonist for Pain Management

(2008) Arthur Gomtsyan et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and structure–activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists

(2007) Itsuro Shimada et al.   BIOORGANIC & MEDICINAL CHEMISTRY

GdCl3 catalysed Grieco condensation: A facile approach for the synthesis of novel pyrimidine and annulated pyrimidine fused indazole derivatives in single pot under mild conditions and their anti-microbial activity

(2007) T. Yakaiah et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY