Identification, Characterization, and Optimization of 2,8-Disubstituted-1,5-naphthyridines as Novel Plasmodium falciparum Phosphatidylinositol-4-kinase Inhibitors with in Vivo Efficacy in a Humanized Mouse Model of Malaria

Title
Identification, Characterization, and Optimization of 2,8-Disubstituted-1,5-naphthyridines as Novel Plasmodium falciparum Phosphatidylinositol-4-kinase Inhibitors with in Vivo Efficacy in a Humanized Mouse Model of Malaria
Authors
Keywords
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Journal
JOURNAL OF MEDICINAL CHEMISTRY
Volume 61, Issue 13, Pages 5692-5703
Publisher
American Chemical Society (ACS)
Online
2018-06-12
DOI
10.1021/acs.jmedchem.8b00648

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