Tricyclic coumarin sulphonate derivatives with alkaline phosphatase inhibitory effects: in vitro and docking studies

Coumarin sulfonates: New alkaline phosphatase inhibitors; in vitro and in silico studies

(2017) Uzma Salar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Gastrointestinal and hepatic mechanisms limiting entry and dissemination of lipopolysaccharide into the systemic circulation

(2016) Mathilde Guerville et al.   AMERICAN JOURNAL OF PHYSIOLOGY-GASTROINTESTINAL AND LIVER PHYSIOLOGY

Synthesis of New Tricyclic and Tetracyclic Fused Coumarin Sulfonate Derivatives and Their Inhibitory Effects on LPS-Induced Nitric Oxide and PGE2Productions in RAW 264.7 Macrophages: Part 2

(2016) Mohammed I. El-Gamal et al.   ARCHIV DER PHARMAZIE

A New Series of Cycloalkane-fused Coumarin Sulfonates: Synthesis andIn VitroAntiproliferative Screening

(2016) Mohammed I. El-Gamal et al.   BULLETIN OF THE KOREAN CHEMICAL SOCIETY

Inhibition of Alkaline Phosphatase: An Emerging New Drug Target

(2015) Mariya Rashida et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Investigation of quinoline-4-carboxylic acid as a highly potent scaffold for the development of alkaline phosphatase inhibitors: synthesis, SAR analysis and molecular modelling studies

(2015) Imtiaz Khan et al.   RSC Advances

Synthesis, in vitro antiproliferative activity, and in silico studies of fused tricyclic coumarin sulfonate derivatives

(2014) Mohammed I. El-Gamal et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Catalytic Signature of a Heat-Stable, Chimeric Human Alkaline Phosphatase with Therapeutic Potential

(2014) Tina Kiffer-Moreira et al.   PLoS One

Synthesis of tricyclic fused coumarin sulfonates and their inhibitory effects on LPS-induced nitric oxide and PGE2 productions in RAW 264.7 macrophages

(2013) Hyeon-Lok Jang et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Identification of novel chromone based sulfonamides as highly potent and selective inhibitors of alkaline phosphatases

(2013) Mariya al-Rashida et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

The Role of Phosphatases in the Initiation of Skeletal Mineralization

(2012) José Luis Millán   CALCIFIED TISSUE INTERNATIONAL

Cellular function and molecular structure of ecto-nucleotidases

(2012) Herbert Zimmermann et al.   Purinergic Signalling

Loss of skeletal mineralization by the simultaneous ablation of PHOSPHO1 and alkaline phosphatase function: A unified model of the mechanisms of initiation of skeletal calcification

(2010) Manisha C Yadav et al.   JOURNAL OF BONE AND MINERAL RESEARCH

Assay Format as a Critical Success Factor for Identification of Novel Inhibitor Chemotypes of Tissue-Nonspecific Alkaline Phosphatase from High-Throughput Screening

(2010) Thomas D.Y. Chung et al.   MOLECULES

High-throughput screening of tissue-nonspecific alkaline phosphatase for identification of effectors with diverse modes of action

(2010) Eduard A Sergienko et al.   Nature Protocols

Discovery and Validation of a Series of Aryl Sulfonamides as Selective Inhibitors of Tissue-Nonspecific Alkaline Phosphatase (TNAP)

(2009) Russell Dahl et al.   JOURNAL OF MEDICINAL CHEMISTRY