Investigation of quinoline-4-carboxylic acid as a highly potent scaffold for the development of alkaline phosphatase inhibitors: synthesis, SAR analysis and molecular modelling studies
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Title
Investigation of quinoline-4-carboxylic acid as a highly potent scaffold for the development of alkaline phosphatase inhibitors: synthesis, SAR analysis and molecular modelling studies
Authors
Keywords
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Journal
RSC Advances
Volume 5, Issue 79, Pages 64404-64413
Publisher
Royal Society of Chemistry (RSC)
Online
2015-07-24
DOI
10.1039/c5ra12455g
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Note: Only part of the references are listed.- Diarylsulfonamides and their bioisosteres as dual inhibitors of alkaline phosphatase and carbonic anhydrase: Structure activity relationship and molecular modelling studies
- (2015) Mariya al-Rashida et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Pathophysiological Role of Vascular Smooth Muscle Alkaline Phosphatase in Medial Artery Calcification
- (2015) Campbell R Sheen et al. JOURNAL OF BONE AND MINERAL RESEARCH
- Catalytic Signature of a Heat-Stable, Chimeric Human Alkaline Phosphatase with Therapeutic Potential
- (2014) Tina Kiffer-Moreira et al. PLoS One
- Identification of a selective inhibitor of murine intestinal alkaline phosphatase (ML260) by concurrent ultra-high throughput screening against human and mouse isozymes
- (2013) Robert J. Ardecky et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Identification of novel chromone based sulfonamides as highly potent and selective inhibitors of alkaline phosphatases
- (2013) Mariya al-Rashida et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- SAR-Based Optimization of a 4-Quinoline Carboxylic Acid Analogue with Potent Antiviral Activity
- (2013) Priyabrata Das et al. ACS Medicinal Chemistry Letters
- Palladium-Catalyzed Sequential Formation of CC Bonds: Efficient Assembly of 2-Substituted and 2,3-Disubstituted Quinolines
- (2012) Xiaochen Ji et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Synthesis of 6-substituted 9-methoxy-11H-indeno[1,2-c]quinoline-11-one derivatives as potential anticancer agents
- (2012) Chih-Hua Tseng et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Synthesis and antiproliferative evaluation of 3-phenylquinolinylchalcone derivatives against non-small cell lung cancers and breast cancers
- (2012) Chih-Hua Tseng et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- A consistent description of HYdrogen bond and DEhydration energies in protein–ligand complexes: methods behind the HYDE scoring function
- (2012) Nadine Schneider et al. JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN
- Synthesis and anti-HCV activity evaluation of anilinoquinoline derivatives
- (2011) Huang-Kai Peng et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis and anti-HIV activity of alkylated quinoline 2,4-diols
- (2010) Nafees Ahmed et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Quinolines and structurally related heterocycles as antimalarials
- (2010) Kirandeep Kaur et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Novel quinoline and naphthalene derivatives as potent antimycobacterial agents
- (2010) Ram Shankar Upadhayaya et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis and Antiproliferative Evaluation of Certain Indeno[1,2-c]quinoline Derivatives. Part 2
- (2010) Chih-Hua Tseng et al. JOURNAL OF MEDICINAL CHEMISTRY
- Reversal Agent and Linker Variants of Reversed Chloroquines: Activities againstPlasmodium falciparum
- (2010) Simeon Andrews et al. JOURNAL OF MEDICINAL CHEMISTRY
- High-throughput screening of tissue-nonspecific alkaline phosphatase for identification of effectors with diverse modes of action
- (2010) Eduard A Sergienko et al. Nature Protocols
- Synthesis and evaluation of benzo[b]thiophene derivatives as inhibitors of alkaline phosphatases
- (2009) Lina Li et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Design and synthesis of selective inhibitors of Placental Alkaline Phosphatase
- (2009) Marion Lanier et al. BIOORGANIC & MEDICINAL CHEMISTRY
- New 1,3-oxazolo[4,5-c]quinoline derivatives: Synthesis and evaluation of antibacterial and antituberculosis properties
- (2009) Sumesh Eswaran et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Identification of benzofuro[2,3- b ]quinoline derivatives as a new class of antituberculosis agents
- (2009) Chiao-Li Yang et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Discovery and Validation of a Series of Aryl Sulfonamides as Selective Inhibitors of Tissue-Nonspecific Alkaline Phosphatase (TNAP)
- (2009) Russell Dahl et al. JOURNAL OF MEDICINAL CHEMISTRY
- Design and synthesis of pyrazole derivatives as potent and selective inhibitors of tissue-nonspecific alkaline phosphatase (TNAP)
- (2008) Shyama Sidique et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
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