11-Azaartemisinin cocrystals with preserved lactam : acid heterosynthons
Published 2018 View Full Article
- Home
- Publications
- Publication Search
- Publication Details
Title
11-Azaartemisinin cocrystals with preserved lactam : acid heterosynthons
Authors
Keywords
-
Journal
CRYSTENGCOMM
Volume 20, Issue 9, Pages 1205-1219
Publisher
Royal Society of Chemistry (RSC)
Online
2018-01-10
DOI
10.1039/c7ce01875d
References
Ask authors/readers for more resources
Related references
Note: Only part of the references are listed.- Controlled release of artemisone for the treatment of experimental cerebral malaria
- (2017) Jacob Golenser et al. Parasites & Vectors
- Methylene Homologues of Artemisone: An Unexpected Structure-Activity Relationship and a Possible Implication for the Design of C10-Substituted Artemisinins
- (2016) Yuet Wu et al. ChemMedChem
- Supply and Demand in the Ball Mill: Competitive Cocrystal Reactions
- (2016) Franziska Fischer et al. CRYSTAL GROWTH & DESIGN
- Design of Cocrystals for Molecules with Limited Hydrogen Bonding Functionalities: Propyphenazone as a Model System
- (2016) Lucy K. Mapp et al. CRYSTAL GROWTH & DESIGN
- On the predictability of supramolecular interactions in molecular cocrystals – the view from the bench
- (2016) Mérina K. Corpinot et al. CRYSTENGCOMM
- In vitro activity of artemisone and artemisinin derivatives against extracellular and intracellular Helicobacter pylori
- (2016) Francesca Sisto et al. INTERNATIONAL JOURNAL OF ANTIMICROBIAL AGENTS
- Antimalarial Chemotherapy: Natural Product Inspired Development of Preclinical and Clinical Candidates with Diverse Mechanisms of Action
- (2016) Elena Fernández-Álvaro et al. JOURNAL OF MEDICINAL CHEMISTRY
- Influence of Coformer Stoichiometric Ratio on Pharmaceutical Cocrystal Dissolution: Three Cocrystals of Carbamazepine/4-Aminobenzoic Acid
- (2016) Zi Li et al. MOLECULAR PHARMACEUTICS
- The Case for Development of 11-Aza-artemisinins for Malaria
- (2015) Rozanne Harmse et al. CURRENT MEDICINAL CHEMISTRY
- Are the Crystal Structures of Enantiopure and Racemic Mandelic Acids Determined by Kinetics or Thermodynamics?
- (2015) Rebecca K. Hylton et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- In vitro anti-cancer effects of artemisone nano-vesicular formulations on melanoma cells
- (2015) Anupma Dwivedi et al. Nanomedicine-Nanotechnology Biology and Medicine
- A molecular mechanism of artemisinin resistance in Plasmodium falciparum malaria
- (2015) Alassane Mbengue et al. NATURE
- Malaria medicines: a glass half full?
- (2015) Timothy N. C. Wells et al. NATURE REVIEWS DRUG DISCOVERY
- The anatomy of a comprehensive constrained, restrained refinement program for the modern computing environment –Olex2dissected
- (2015) Luc J. Bourhis et al. Acta Crystallographica A-Foundation and Advances
- Crystal structure refinement withSHELXL
- (2015) George M. Sheldrick Acta Crystallographica Section C-Structural Chemistry
- Stimulation of Suicidal Erythrocyte Death by Artesunate
- (2014) Kousi Alzoubi et al. CELLULAR PHYSIOLOGY AND BIOCHEMISTRY
- Continuous synthesis of artemisinin-derived medicines
- (2014) Kerry Gilmore et al. CHEMICAL COMMUNICATIONS
- Cocrystal Formation between Chiral Compounds: How Cocrystals Differ from Salts
- (2014) Géraldine Springuel et al. CRYSTAL GROWTH & DESIGN
- Pharmaceutical co-crystals – are we there yet?
- (2014) N. Blagden et al. CRYSTENGCOMM
- New Orally Active Amino- and Hydroxy-Functionalized 11-Azaartemisinins and Their Derivatives with High Order of Antimalarial Activity against Multidrug-Resistant Plasmodium yoelii in Swiss Mice1
- (2014) Chandan Singh et al. JOURNAL OF MEDICINAL CHEMISTRY
- New Uses for Old Drugs: The Tale of Artemisinin Derivatives in the Elimination of Schistosomiasis Japonica in China
- (2014) Yi-Xin Liu et al. MOLECULES
- Mechanism for Polymorphic Transformation of Artemisinin during High Temperature Extrusion
- (2013) Chaitrali Kulkarni et al. CRYSTAL GROWTH & DESIGN
- Cocrystals of Nicotinamide and (R)-Mandelic Acid in Many Ratios with Anomalous Formation Properties
- (2013) Si-Wei Zhang et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Halogen Bonding and Pharmaceutical Cocrystals: The Case of a Widely Used Preservative
- (2013) Michele Baldrighi et al. MOLECULAR PHARMACEUTICS
- High-level semi-synthetic production of the potent antimalarial artemisinin
- (2013) C. J. Paddon et al. NATURE
- Antimalarial drug discovery — approaches and progress towards new medicines
- (2013) Erika L. Flannery et al. NATURE REVIEWS MICROBIOLOGY
- Artemisinins: Pharmacological actions beyond anti-malarial
- (2013) Wanxing Eugene Ho et al. PHARMACOLOGY & THERAPEUTICS
- Continuous-Flow Synthesis of the Anti-Malaria Drug Artemisinin
- (2012) François Lévesque et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Quantifying Homo- and Heteromolecular Hydrogen Bonds as a Guide for Adduct Formation
- (2012) Amit Delori et al. CHEMISTRY-A EUROPEAN JOURNAL
- Crystal Engineering of Stable Temozolomide Cocrystals
- (2012) N. Jagadeesh Babu et al. Chemistry-An Asian Journal
- Innovative Chiral Resolution Using Enantiospecific Co-Crystallization in Solution
- (2012) Géraldine Springuel et al. CRYSTAL GROWTH & DESIGN
- Polymorphs, Salts, and Cocrystals: What’s in a Name?
- (2012) Srinivasulu Aitipamula et al. CRYSTAL GROWTH & DESIGN
- Surprisingly complex supramolecular behaviour in the crystal structures of a family of mono-substituted salicylic acids
- (2012) Riccardo Montis et al. CRYSTENGCOMM
- EDMA: a computer program for topological analysis of discrete electron densities
- (2012) Lukáš Palatinus et al. JOURNAL OF APPLIED CRYSTALLOGRAPHY
- A Concise Synthesis of (+)-Artemisinin
- (2012) Chunyin Zhu et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Simultaneously Improving the Mechanical Properties, Dissolution Performance, and Hygroscopicity of Ibuprofen and Flurbiprofen by Cocrystallization with Nicotinamide
- (2012) Shing Fung Chow et al. PHARMACEUTICAL RESEARCH
- Solubility Advantage of Amorphous Drugs and Pharmaceutical Cocrystals
- (2011) N. Jagadeesh Babu et al. CRYSTAL GROWTH & DESIGN
- Some thoughts about the single crystal growth of small molecules
- (2011) Bernhard Spingler et al. CRYSTENGCOMM
- Pharmaceutical cocrystals: An overview
- (2011) Ning Qiao et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- The discovery of artemisinin (qinghaosu) and gifts from Chinese medicine
- (2011) Youyou Tu NATURE MEDICINE
- Facile Oxidation of Leucomethylene Blue and Dihydroflavins by Artemisinins: Relationship with Flavoenzyme Function and Antimalarial Mechanism of Action
- (2010) Richard K. Haynes et al. ChemMedChem
- 1:1 and 2:1 Urea−Succinic Acid Cocrystals: Structural Diversity, Solution Chemistry, and Thermodynamic Stability
- (2010) Amjad Alhalaweh et al. CRYSTAL GROWTH & DESIGN
- New solid forms of artemisinin obtained through cocrystallisation
- (2010) Shyam Karki et al. CRYSTENGCOMM
- What made sesquiterpene lactones reach cancer clinical trials?
- (2010) Akram Ghantous et al. DRUG DISCOVERY TODAY
- Benefits of cocrystallisation in pharmaceutical materials science: an update
- (2010) Tomislav Friščić et al. JOURNAL OF PHARMACY AND PHARMACOLOGY
- The Molecular Mechanism of Action of Artemisinin—The Debate Continues
- (2010) Paul M. O’Neill et al. MOLECULES
- Improving Mechanical Properties of Crystalline Solids by Cocrystal Formation: New Compressible Forms of Paracetamol
- (2009) Shyam Karki et al. ADVANCED MATERIALS
- Predicting Multicomponent Crystal Formation: The Interplay between Homomeric and Heteromeric Interactions
- (2009) Guangwen He et al. CRYSTAL GROWTH & DESIGN
- The Reemergence of Cocrystals: The Crystal Clear Writing Is on the WallIntroduction to Virtual Special Issue on Pharmaceutical Cocrystals
- (2009) CRYSTAL GROWTH & DESIGN
- Solubility Advantage of Pharmaceutical Cocrystals
- (2009) David J. Good et al. CRYSTAL GROWTH & DESIGN
- Synthesis and Structural Characterization of Cocrystals and Pharmaceutical Cocrystals: Mechanochemistry vs Slow Evaporation from Solution
- (2009) David R. Weyna et al. CRYSTAL GROWTH & DESIGN
- Pharmaceutical Cocrystals and Their Physicochemical Properties
- (2009) Nate Schultheiss et al. CRYSTAL GROWTH & DESIGN
- OLEX2: a complete structure solution, refinement and analysis program
- (2009) Oleg V. Dolomanov et al. JOURNAL OF APPLIED CRYSTALLOGRAPHY
- Artemisinin Resistance inPlasmodium falciparumMalaria
- (2009) Arjen M. Dondorp et al. NEW ENGLAND JOURNAL OF MEDICINE
- Towards Prediction of Stoichiometry in Crystalline Multicomponent Complexes
- (2008) Aurora J. Cruz-Cabeza et al. CHEMISTRY-A EUROPEAN JOURNAL
- The Antiviral Activities of Artemisinin and Artesunate
- (2008) Thomas Efferth et al. CLINICAL INFECTIOUS DISEASES
- Improving Mechanical Properties of Caffeine and Methyl Gallate Crystals by Cocrystallization
- (2008) Changquan Calvin Sun et al. CRYSTAL GROWTH & DESIGN
- Applying Hot-Stage Microscopy to Co-Crystal Screening: A Study of Nicotinamide with Seven Active Pharmaceutical Ingredients
- (2008) David J. Berry et al. CRYSTAL GROWTH & DESIGN
- Can the Formation of Pharmaceutical Cocrystals Be Computationally Predicted? I. Comparison of Lattice Energies
- (2008) Nizar Issa et al. CRYSTAL GROWTH & DESIGN
- Screening strategies based on solubility and solution composition generate pharmaceutically acceptable cocrystals of carbamazepine
- (2008) Scott L. Childs et al. CRYSTENGCOMM
- On the thermodynamics of cocrystal formation
- (2008) R SCHARTMAN INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Mercury CSD 2.0– new features for the visualization and investigation of crystal structures
- (2008) Clare F. Macrae et al. JOURNAL OF APPLIED CRYSTALLOGRAPHY
- Amino- and Hydroxy-Functionalized 11-Azaartemisinins and Their Derivatives
- (2008) Ajit Shankar Singh et al. ORGANIC LETTERS
- Artemisinins: their growing importance in medicine
- (2008) Sanjeev Krishna et al. TRENDS IN PHARMACOLOGICAL SCIENCES
Publish scientific posters with Peeref
Peeref publishes scientific posters from all research disciplines. Our Diamond Open Access policy means free access to content and no publication fees for authors.
Learn MoreCreate your own webinar
Interested in hosting your own webinar? Check the schedule and propose your idea to the Peeref Content Team.
Create Now