Synthesis of [(1,2,3-Triazol-1-yl)methyl]boronic Acids Through Click Chemistry: Easy Access to a Potential Scaffold for Protease Inhibitors

1,2,3-Triazole in Heterocyclic Compounds, Endowed with Biological Activity, through 1,3-Dipolar Cycloadditions

(2014) Antonino Lauria et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Click Chemistry for Drug Development and Diverse Chemical–Biology Applications

(2013) Prakasam Thirumurugan et al.   CHEMICAL REVIEWS

Focusing on boron in medicinal chemistry

(2013) P Veeraraghavan Ramachandran   Future Medicinal Chemistry

Click Chemistry in Peptide-Based Drug Design

(2013) Huiyuan Li et al.   MOLECULES

Boron Containing Compounds as Protease Inhibitors

(2012) Reem Smoum et al.   CHEMICAL REVIEWS

The impact of click chemistry in medicinal chemistry

(2012) Jingli Hou et al.   Expert Opinion on Drug Discovery

Fragment-guided design of subnanomolar  -lactamase inhibitors active in vivo

(2012) O. Eidam et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Aminoboronic acids and esters: from synthetic challenges to the discovery of unique classes of enzyme inhibitors

(2011) Sabrina Touchet et al.   CHEMICAL SOCIETY REVIEWS

Boron-containing inhibitors of synthetases

(2011) Stephen J. Baker et al.   CHEMICAL SOCIETY REVIEWS

Regioselective Synthesis and Slow-Release Suzuki–Miyaura Cross-Coupling of MIDA Boronate-Functionalized Isoxazoles and Triazoles

(2011) Jonathan E. Grob et al.   JOURNAL OF ORGANIC CHEMISTRY

Design, Synthesis, Crystal Structures, and Antimicrobial Activity of Sulfonamide Boronic Acids as β-Lactamase Inhibitors

(2010) Oliv Eidam et al.   JOURNAL OF MEDICINAL CHEMISTRY

Click Reactions and Boronic Acids: Applications, Issues, and Potential Solutions

(2010) Chaofeng Dai et al.   MOLECULES

Identification of the first fluorescent α-amidoboronic acids that change fluorescent properties upon sugar binding

(2009) Shan Jin et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Fluoride protects boronic acids in the copper(i)-mediated click reaction

(2009) Shan Jin et al.   CHEMICAL COMMUNICATIONS

When in Rome, reform. Radical reform of the Italian research and education systems is needed to address the lack of autonomy and lack of funding

(2009) Marta Paterlini   EMBO REPORTS

A direct route to triazole boronic esters and their application in the synthesis of small molecule arrays

(2009) Jianhui Huang et al.   TETRAHEDRON LETTERS

Cu-Catalyzed Azide−Alkyne Cycloaddition

(2008) Morten Meldal et al.   CHEMICAL REVIEWS

Dipeptide Boronic Acid Inhibitors of Dipeptidyl Peptidase IV: Determinants of Potency and in Vivo Efficacy and Safety

(2008) Beth A. Connolly et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of a (β-acetamido-α-acetoxyethyl)boronic ester via azido boronic esters

(2008) Donald S. Matteson et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

Copper-Facilitated Suzuki Reactions: Application to 2-Heterocyclic Boronates

(2008) James Z. Deng et al.   ORGANIC LETTERS

Structure-based optimization of cephalothin-analogue boronic acids as β-lactamase inhibitors

(2007) Stefania Morandi et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Click chemistry reactions in medicinal chemistry: Applications of the 1,3-dipolar cycloaddition between azides and alkynes

(2007) Gian Cesare Tron et al.   MEDICINAL RESEARCH REVIEWS

α-Amido boronic acids: A synthetic challenge and their properties as serine protease inhibitors

(2007) Donald S. Matteson   MEDICINAL RESEARCH REVIEWS