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Improving the Binding Affinity of in-Vitro-Evolved Cyclic Peptides by Inserting Atoms into the Macrocycle Backbone

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Half-Life Extension of Biopharmaceuticals using Chemical Methods: Alternatives to PEGylation

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(2016) Roland E. Kontermann   EXPERT OPINION ON BIOLOGICAL THERAPY

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A Synthetic Factor XIIa Inhibitor Blocks Selectively Intrinsic Coagulation Initiation

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Identification of Structure-Activity Relationships from Screening a Structurally Compact DNA-Encoded Chemical Library

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The role of albumin receptors in regulation of albumin homeostasis: Implications for drug delivery

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A biomimetic approach for enhancing the in vivo half-life of peptides

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Factor XII: a drug target for safe interference with thrombosis and inflammation

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mRNA display: from basic principles to macrocycle drug discovery

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Bicyclic Peptide Inhibitor Reveals Large Contact Interface with a Protease Target

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Bicyclic Peptides with Optimized Ring Size Inhibit Human Plasma Kallikrein and its Orthologues While Sparing Paralogous Proteases

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Bicyclization and Tethering to Albumin Yields Long-Acting Peptide Antagonists

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Design of the Novel Protraction Mechanism of Insulin Degludec, an Ultra-long-Acting Basal Insulin

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Phage-encoded combinatorial chemical libraries based on bicyclic peptides

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A Portable Albumin Binder from a DNA-Encoded Chemical Library

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