The binding selectivity of vonoprazan (TAK-438) to the gastric H+,K+-ATPase
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Title
The binding selectivity of vonoprazan (TAK-438) to the gastric H+,K+-ATPase
Authors
Keywords
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Journal
ALIMENTARY PHARMACOLOGY & THERAPEUTICS
Volume 42, Issue 11-12, Pages 1315-1326
Publisher
Wiley
Online
2015-10-01
DOI
10.1111/apt.13414
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Note: Only part of the references are listed.- Randomised clinical trial: safety, tolerability, pharmacokinetics and pharmacodynamics of repeated doses of TAK-438 (vonoprazan), a novel potassium-competitive acid blocker, in healthy male subjects
- (2015) H. Jenkins et al. ALIMENTARY PHARMACOLOGY & THERAPEUTICS
- Randomised clinical trial: a dose-ranging study of vonoprazan, a novel potassium-competitive acid blocker, vs. lansoprazole for the treatment of erosive oesophagitis
- (2015) K. Ashida et al. ALIMENTARY PHARMACOLOGY & THERAPEUTICS
- Acid-inhibitory effects of vonoprazan 20 mg compared with esomeprazole 20 mg or rabeprazole 10 mg in healthy adult male subjects - a randomised open-label cross-over study
- (2015) Y. Sakurai et al. ALIMENTARY PHARMACOLOGY & THERAPEUTICS
- Vonoprazan: First Global Approval
- (2015) Karly P. Garnock-Jones DRUGS
- Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Single Rising TAK-438 (Vonoprazan) Doses in Healthy Male Japanese/non-Japanese Subjects
- (2015) Yuuichi Sakurai et al. Clinical and Translational Gastroenterology
- Systematic Comparison of Molecular Conformations of H+,K+-ATPase Reveals an Important Contribution of the A-M2 Linker for the Luminal Gating
- (2014) Kazuhiro Abe et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- Protonated Form: The Potent Form of Potassium-Competitive Acid Blockers
- (2014) Hua-Jun Luo et al. PLoS One
- A Randomized, Comparative Trial of a Potassium-Competitive Acid Blocker (AZD0865) and Esomeprazole for the Treatment of Patients With Nonerosive Reflux Disease
- (2013) John Dent et al. AMERICAN JOURNAL OF GASTROENTEROLOGY
- Discovery, synthesis, and biological evaluation of novel pyrrole derivatives as highly selective potassium-competitive acid blockers
- (2012) Haruyuki Nishida et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Discovery of a Novel Pyrrole Derivative 1-[5-(2-Fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine Fumarate (TAK-438) as a Potassium-Competitive Acid Blocker (P-CAB)
- (2012) Yasuyoshi Arikawa et al. JOURNAL OF MEDICINAL CHEMISTRY
- Clinical trial: Inhibitory effect of revaprazan on gastric acid secretion in healthy male subjects
- (2010) Hyung-Keun Kim et al. JOURNAL OF GASTROENTEROLOGY AND HEPATOLOGY
- 1-[5-(2-Fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine Monofumarate (TAK-438), a Novel and Potent Potassium-Competitive Acid Blocker for the Treatment of Acid-Related Diseases
- (2010) Y. Hori et al. JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
- Acid peptic diseases: pharmacological approach to treatment
- (2009) Alex Mejia et al. Expert Review of Clinical Pharmacology
- The gastric HK-ATPase: structure, function, and inhibition
- (2008) Jai Moo Shin et al. PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY
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