Palladium-catalyzed tandem addition/cyclization in aqueous medium: synthesis of 2-arylindoles

Efficient synthesis of isoquinolines in water by a Pd-catalyzed tandem reaction of functionalized alkylnitriles with arylboronic acids

(2017) Kun Hu et al.   GREEN CHEMISTRY

The Development of a Palladium-Catalyzed Tandem Addition/Cyclization for the Construction of Indole Skeletons

(2017) Shuling Yu et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-catalyzed C–O bond cleavage and cyclization: synthesis of indazolo[3,2-b]quinazolinones

(2017) Rui Qiao et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Mild and selective base-free C–H arylation of heteroarenes: experiment and computation

(2017) Hannes P. L. Gemoets et al.   Chemical Science

Commercial Supported Gold Nanoparticles Catalyzed Alkyne Hydroamination and Indole Synthesis

(2016) Shengzong Liang et al.   ADVANCED SYNTHESIS & CATALYSIS

Design, Synthesis, and Structure–Activity Relationship Study of Novel Indole-2-carboxamide Derivatives as Anti-inflammatory Agents for the Treatment of Sepsis

(2016) Zhiguo Liu et al.   JOURNAL OF MEDICINAL CHEMISTRY

Indole-2-carboxamide-based MmpL3 Inhibitors Show Exceptional Antitubercular Activity in an Animal Model of Tuberculosis Infection

(2016) Jozef Stec et al.   JOURNAL OF MEDICINAL CHEMISTRY

Improved Potency of Indole-Based NorA Efflux Pump Inhibitors: From Serendipity toward Rational Design and Development

(2016) Federica Buonerba et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Hexacyclic, Iboga-Derived Monoterpenoid Indole with a Contracted Tetrahydroazepine C-Ring and Incorporation of an Isoxazolidine Moiety, a Seco-Corynanthean, an Aspidosperma-Aspidosperma Bisindole with Anticancer Properties, and the Absolute Configuration of the Pyridopyrimidine Indole Alkaloid, Vernavosine

(2016) Choy-Eng Nge et al.   JOURNAL OF NATURAL PRODUCTS

Monoterpene Indole Alkaloids from the Fruit of Tabernaemontana litoralis and Differential Alkaloid Composition in Various Fruit Components

(2016) Yang Qu et al.   JOURNAL OF NATURAL PRODUCTS

One-Pot Synthesis of Substituted Benzo[b]furans and Indoles from Dichlorophenols/Dichloroanilines Using a Palladium–Dihydroxyterphenylphosphine Catalyst

(2016) Miyuki Yamaguchi et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-catalyzed direct arylation of indoles with arylsulfonyl hydrazides

(2016) Congrong Liu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Diborane-Mediated Deoxygenation of o-Nitrostyrenes To Form Indoles

(2016) Kai Yang et al.   ORGANIC LETTERS

Active and Recyclable Catalytic Synthesis of Indoles by Reductive Cyclization of 2-(2-Nitroaryl)acetonitriles in the Presence of Co–Rh Heterobimetallic Nanoparticles with Atmospheric Hydrogen under Mild Conditions

(2016) Isaac Choi et al.   ORGANIC LETTERS

Tandem Addition/Cyclization for Access to Isoquinolines and Isoquinolones via Catalytic Carbopalladation of Nitriles

(2016) Linjun Qi et al.   ORGANIC LETTERS

Catalytic Synthesis of Substituted Indoles and Quinolines from the Dehydrative C–H Coupling of Arylamines with 1,2- and 1,3-Diols

(2016) Hanbin Lee et al.   ORGANOMETALLICS

An Efficient Reusable Mesoporous Solid-Based Pd Catalyst for Selective C2 Arylation of Indoles in Water

(2016) Linlin Duan et al.   ACS Catalysis

Catalytic α-Arylation of Imines Leading to N-Unprotected Indoles and Azaindoles

(2016) Enrico Marelli et al.   ACS Catalysis

Intramolecular Cooperative CC Bond Cleavage Reaction of 1,3-Dicarbonyl Compounds with 2-Iodoanilines to Giveo-(N-Acylamino)aryl Ketones and Multisubstituted Indoles

(2015) Qi Xing  et al.   CHEMISTRY-A EUROPEAN JOURNAL

Indole Alkaloids from Chaetomium globosum

(2015) Guo-Bo Xu et al.   JOURNAL OF NATURAL PRODUCTS

Regioselective Synthesis of Indolo[1,2-c]quinazolines and 11H-Indolo[3,2-c]quinolines via Copper-Catalyzed Cascade Reactions of 2-(2-Bromoaryl)-1H-indoles with Aldehydes and Aqueous Ammonia

(2015) Shenghai Guo et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Naphtho[1′,2′:4,5]imidazo[1,2-a]pyridines and Imidazo[5,1,2-cd]indolizines Through Pd-Catalyzed Cycloaromatization of 2-Phenylimidazo[1,2-a]pyridines with Alkynes

(2015) Peiyuan Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Synthesis of 2-Arylquinazolinones from 2-Arylindoles with Amines or Ammoniums

(2015) Yadong Feng et al.   JOURNAL OF ORGANIC CHEMISTRY

Organotrifluoroborates: Another Branch of the Mighty Oak

(2015) Gary A. Molander   JOURNAL OF ORGANIC CHEMISTRY

Palladium catalyzed decarboxylative acylation of arylboronic acid with ethyl cyanoacetate as a new acylating agent: synthesis of alkyl aryl ketones

(2015) Md Yousuf et al.   NEW JOURNAL OF CHEMISTRY

An efficient and practical synthesis of [2-11C]indole via superfast nucleophilic [11C]cyanation and RANEY® Nickel catalyzed reductive cyclization

(2015) So Jeong Lee et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Ruthenium-Catalyzed Heteroatom-Directed Regioselective C–H Arylation of Indoles Using a Removable Tether

(2015) Virendra Kumar Tiwari et al.   ORGANIC LETTERS

Merging C–H Activation and Alkene Difunctionalization at Room Temperature: A Palladium-Catalyzed Divergent Synthesis of Indoles and Indolines

(2015) Manash Kumar Manna et al.   ORGANIC LETTERS

Synthesis of 2-Substituted Indoles through Visible Light-Induced Photocatalytic Cyclizations of Styryl Azides

(2014) Xu-Dong Xia et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-catalyzed direct C–H arylation of pyridine N-oxides with arylboronic esters: one-pot synthesis of 2-arylpyridines

(2014) Yan Shen et al.   CHEMICAL COMMUNICATIONS

Palladium-Catalyzed Cascade Reaction of 2-Amino-N′-arylbenzohydrazides with Triethyl Orthobenzoates To Construct Indazolo[3,2-b]quinazolinones

(2014) Weiguang Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium(II)-Catalyzed Desulfitative Synthesis of Aryl Ketones from Sodium Arylsulfinates and Nitriles: Scope, Limitations, and Mechanistic Studies

(2014) Bobo Skillinghaug et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-catalyzed direct addition of arylboronic acids to 2-aminobenzonitrile derivatives: synthesis, biological evaluation and in silico analysis of 2-aminobenzophenones, 7-benzoyl-2-oxoindolines, and 7-benzoylindoles

(2014) Jiuxi Chen et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Palladium-catalyzed tandem reaction of 2-hydroxyarylacetonitriles with sodium sulfinates: one-pot synthesis of 2-arylbenzofurans

(2014) Jiuxi Chen et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Pd-Catalyzed Intramolecular Aerobic Oxidative C–H Amination of 2-Aryl-3-(arylamino)quinazolinones: Synthesis of Fluorescent Indazolo[3,2-b]quinazolinones

(2014) Weiguang Yang et al.   ORGANIC LETTERS

A highly efficient and recyclable Fe3O4 magnetic nanoparticle immobilized palladium catalyst for the direct C-2 arylation of indoles with arylboronic acids

(2014) Lei Zhang et al.   Catalysis Science & Technology

Oxidation of 2-arylindoles for synthesis of 2-arylbenzoxazinones with oxone as the sole oxidant

(2013) Xiao-Li Lian et al.   CHEMICAL COMMUNICATIONS

Palladium-Catalyzed Addition of Potassium Aryltrifluoroborates to Aliphatic Nitriles: Synthesis of Alkyl Aryl Ketones, Diketone Compounds, and 2-Arylbenzo[b]furans

(2013) Xingyong Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Unexpected Copper-Catalyzed Cascade Synthesis of Quinazoline Derivatives

(2013) Zhongyan Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium(II)-Catalyzed Cyclization Reaction of 2-(Alk-2′-ynyl- oxy)benzonitriles or 2-(Alk-2′-ynylamino)benzonitriles: A Facile Way to 2H-Chromene and 1,2-Dihydroquinoline Derivatives

(2012) Guoqin Xia et al.   ADVANCED SYNTHESIS & CATALYSIS

Palladium-Catalyzed Aerobic Oxidative Coupling of Acyl Chlorides with Arylboronic Acids

(2012) Jiuxi Chen et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-Catalyzed Activation of Dioxygen: Oxidative Cyclization of 2-Arylindoles

(2012) Peng Sang et al.   ADVANCED SYNTHESIS & CATALYSIS

A Metal-Free Sulfenylation and Bromosulfenylation of Indoles: Controllable Synthesis of 3-Arylthioindoles and 2-Bromo-3-arylthioindoles

(2012) Dayun Huang et al.   ADVANCED SYNTHESIS & CATALYSIS

Ligand-free copper-catalyzed coupling of nitroarenes with arylboronic acids

(2012) Jilei Zhang et al.   GREEN CHEMISTRY

Nickel-Catalyzed Intermolecular Insertion of Aryl Iodides to Nitriles: A Novel Method to Synthesize Arylketones

(2012) Jen-Chieh Hsieh et al.   ORGANIC LETTERS

Synthesis of ketones by palladium-catalysed desulfitative reaction of arylsulfinic acids with nitriles

(2011) Tao Miao et al.   CHEMICAL COMMUNICATIONS

Direct Synthesis of Aryl Ketones by Palladium-Catalyzed Desulfinative Addition of Sodium Sulfinates to Nitriles

(2011) Jing Liu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Palladium-Catalyzed Direct 2-Alkylation of Indoles by Norbornene-Mediated Regioselective Cascade C–H Activation

(2011) Lei Jiao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Decarboxylative Coupling of Isatoic Anhydrides with Arylboronic Acids

(2011) Wei Lu et al.   ORGANIC LETTERS

The Coupling of Arylboronic Acids with Nitroarenes Catalyzed by Rhodium

(2011) Xingwang Zheng et al.   ORGANIC LETTERS

The Development of Catalytic Nucleophilic Additions of Terminal Alkynes in Water†

(2010) Chao-Jun Li   ACCOUNTS OF CHEMICAL RESEARCH

“On Water” Direct and Site-Selective Pd-Catalysed CH Arylation of (NH)-Indoles

(2010) Lionel Joucla et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of Aryl Ketones by Palladium(II)-Catalyzed Decarboxylative Addition of Benzoic Acids to Nitriles

(2010) Jonas Lindh et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Water: Nature’s Reaction Enforcer—Comparative Effects for Organic Synthesis “In-Water” and “On-Water”

(2010) Richard N. Butler et al.   CHEMICAL REVIEWS

Reduction of polycyclic aromatic hydrocarbons promoted by cobalt or manganese nanoparticles

(2010) Fabiana Nador et al.   TETRAHEDRON

Copper-CatalyzedN-Arylation/Hydroamin(d)ation Domino Synthesis of Indoles and its Application to the Preparation of a Chek1/KDR Kinase Inhibitor Pharmacophore

(2009) Lutz Ackermann et al.   ADVANCED SYNTHESIS & CATALYSIS

Nitrile Ligated Transition Metal Complexes with Weakly Coordinating Counteranions and Their Catalytic Applications

(2009) Silvana F. Rach et al.   CHEMICAL REVIEWS

Synthesis and potent antifungal activity againstCandidaspecies of some novel 1H-benzimidazoles

(2009) Hakan Göker et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Synthesis of indoles via alkylidenation of acyl hydrazides

(2009) Kevin Hisler et al.   TETRAHEDRON LETTERS

Palladium-Catalyzed Direct Arylation of (Hetero)Arenes with Aryl Boronic Acids

(2008) Shang-Dong Yang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Dirhodium(II)-Catalyzed Intramolecular CH Amination of Aryl Azides

(2008) Meihua Shen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Room Temperature and Phosphine Free Palladium Catalyzed Direct C-2 Arylation of Indoles

(2008) Nathalie Lebrasseur et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Regiochemistry of the microwave-assisted reaction between aromatic amines and α-bromoketones to yield substituted 1H-indoles

(2008) Yosu Vara et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

One-Pot Synthesis of 2-Substituted Indoles from 2-Aminobenzyl Phosphonium Salts. A Formal Total Synthesis of Arcyriacyanin A

(2008) George A. Kraus et al.   ORGANIC LETTERS

The chemistry of homophthalic acid: a new synthetic strategy for construction of substituted isocoumarin and indole skeletons

(2008) Sevil Özcan et al.   TETRAHEDRON

Potassium Organotrifluoroborates:  New Perspectives in Organic Synthesis

(2007) Sylvain Darses et al.   CHEMICAL REVIEWS