Impact of Target Warhead and Linkage Vector on Inducing Protein Degradation: Comparison of Bromodomain and Extra-Terminal (BET) Degraders Derived from Triazolodiazepine (JQ1) and Tetrahydroquinoline (I-BET726) BET Inhibitor Scaffolds

Title
Impact of Target Warhead and Linkage Vector on Inducing Protein Degradation: Comparison of Bromodomain and Extra-Terminal (BET) Degraders Derived from Triazolodiazepine (JQ1) and Tetrahydroquinoline (I-BET726) BET Inhibitor Scaffolds
Authors
Keywords
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Journal
JOURNAL OF MEDICINAL CHEMISTRY
Volume 61, Issue 2, Pages 504-513
Publisher
American Chemical Society (ACS)
Online
2017-06-09
DOI
10.1021/acs.jmedchem.6b01912

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