Metal-free iodine-catalyzed direct cross-dehydrogenative coupling (CDC) between pyrazoles and thiols

Chemoselective cross-coupling reaction of sodium sulfinates with phenols under aqueous conditions

(2016) Fuhong Xiao et al.   GREEN CHEMISTRY

Iodine-catalyzed thiolation of electron-rich aromatics using sulfonyl hydrazides as sulfenylation reagents

(2016) Xia Zhao et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

KIO3-Catalyzed Aerobic Cross-Coupling Reactions of Enaminones and Thiophenols: Synthesis of Polyfunctionalized Alkenes by Metal-Free C–H Sulfenylation

(2016) Jie-Ping Wan et al.   ORGANIC LETTERS

Palladium N-heterocyclic carbene catalyzed regioselective thiolation of 1-aryl-3-methyl-1H-pyrazol-5(4H)-ones using aryl thiols

(2016) Vishal B. Purohit et al.   TETRAHEDRON

A copper-catalyzed cascade reaction of o-bromoarylisothiocyanates with isocyanides leading to benzo[d]imidazo[5,1-b]thiazoles under ligand-free conditions

(2016) Kelu Yan et al.   Organic Chemistry Frontiers

Copper-catalyzed domino synthesis of benzo[b]thiophene/imidazo[1,2-a]pyridines by sequential Ullmann-type coupling and intramolecular C(sp2)–H thiolation

(2016) Kelu Yan et al.   Organic Chemistry Frontiers

Discovery of 4-(phenyl)thio-1H-pyrazole derivatives as agonists of GPR109A, a high affinity niacin receptor

(2015) Hyeon Young Kim et al.   ARCHIVES OF PHARMACAL RESEARCH

Synthesis and biological evaluation of pyrazolylthiazole carboxylic acids as potent anti-inflammatory–antimicrobial agents

(2015) Poonam Khloya et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Recent advances in bioactive pyrazoles

(2015) Ş.Güniz Küçükgüzel et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Iodine catalyzed cross-dehydrogenative C–S coupling by C(sp2)–H bond activation: direct access to aryl sulfides from aryl thiols

(2015) Santosh Kumar Reddy Parumala et al.   GREEN CHEMISTRY

Palladium-Catalyzed Chelation-Assisted Regioselective Oxidative Dehydrogenative Homocoupling/Ortho-Hydroxylation in N-Phenylpyrazoles

(2015) Harikrishna Batchu et al.   JOURNAL OF ORGANIC CHEMISTRY

Catalyst-Free Regioselective C-3 Thiocyanation of Imidazopyridines

(2015) Daoshan Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal-Free Iodine-Catalyzed Direct Arylthiation of Substituted Anilines with Thiols

(2015) Daoshan Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 2-Aryl and 3-Aryl Benzo[b]furan Thioethers Using Aryl Sulfonyl Hydrazides as Sulfenylation Reagents

(2015) Xia Zhao et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal-Free Iodine-Catalyzed Synthesis of Fully Substituted Pyrazoles and Its Sulphenylation

(2015) Jun Sun et al.   JOURNAL OF ORGANIC CHEMISTRY

Catalyst-free direct decarboxylative coupling of α-keto acids with thiols: a facile access to thioesters

(2015) Kelu Yan et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Iodine-catalyzed regioselective thiolation of imidazo[1,2-a]pyridines using sulfonyl hydrazides as a thiol surrogate

(2015) Avik Kumar Bagdi et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Byproduct promoted regioselective sulfenylation of indoles with sulfinic acids

(2015) Cong-Rong Liu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Direct thiolation of methoxybenzenes with thiols under metal-free conditions by iodine catalysis

(2015) Kelu Yan et al.   TETRAHEDRON LETTERS

Iodine-mediated thiolation of phenol/phenylamine derivatives and sodium arylsulfinates in neat water

(2015) Dingyi Wang et al.   RSC Advances

Iodine-Catalyzed Regioselective Sulfenylation of Indoles with Sodium Sulfinates

(2014) Fuhong Xiao et al.   ADVANCED SYNTHESIS & CATALYSIS

Iron or boron-catalyzed C–H arylthiation of substituted phenols at room temperature

(2014) Hua Tian et al.   CHEMICAL COMMUNICATIONS

p-Toluenesulphonic acid-promoted, I2-catalysed sulphenylation of pyrazolones with aryl sulphonyl hydrazides

(2014) Xia Zhao et al.   CHEMICAL COMMUNICATIONS

Transition-Metal-Free Coupling Reactions

(2014) Chang-Liang Sun et al.   CHEMICAL REVIEWS

Iodine-Mediated Thiolation of Substituted Naphthols/Naphthylamines and Arylsulfonyl Hydrazides via C(sp2)–H Bond Functionalization

(2014) Xing Kang et al.   JOURNAL OF ORGANIC CHEMISTRY

A Solvent- and Metal-Free Synthesis of 3-Chacogenyl-indoles Employing DMSO/I2 as an Eco-friendly Catalytic Oxidation System

(2014) Juliano B. Azeredo et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium Catalyzed Aryl(alkyl)thiolation of Unactivated Arenes

(2014) Perumal Saravanan et al.   ORGANIC LETTERS

K2S2O8/arenesulfinate: an unprecedented thiolating system enabling selective sulfenylation of indoles under metal-free conditions

(2014) Honghua Rao et al.   RSC Advances

Metal-free n-Et4NBr-catalyzed radical cyclization of disulfides and alkynes leading to benzothiophenes under mild conditions

(2014) Daoshan Yang et al.   RSC Advances

Synthesis of 3-sulfenylated indoles by a simple NaOH promoted sulfenylation reaction

(2014) Yunyun Liu et al.   RSC Advances

Iodine-Catalyzed Regioselective Sulfenylation of Indoles with Sulfonyl Hydrazides

(2013) Fu-Lai Yang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and properties of a Cu(ii) complexing pyrazole ligandoside in DNA

(2013) M. Su et al.   CHEMICAL COMMUNICATIONS

New pyrazole derivatives containing 1,2,4-triazoles and benzoxazoles as potent antimicrobial and analgesic agents

(2013) A.M. Vijesh et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

K2CO3 promoted direct sulfenylation of indoles: a facile approach towards 3-sulfenylindoles

(2013) Peng Sang et al.   GREEN CHEMISTRY

Iodine-catalyzed efficient 2-arylsulfanylphenol formation from thiols and cyclohexanones

(2013) Yunfeng Liao et al.   GREEN CHEMISTRY

Transition-Metal-Free Synthesis of Unsymmetrical Diaryl Chalcogenides from Arenes and Diaryl Dichalcogenides

(2013) Ch Durga Prasad et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal-Free Oxidative C(sp3)–H Bond Thiolation of Ethers with Disulfides

(2013) Sheng-rong Guo et al.   ORGANIC LETTERS

Transition metal-free direct C–H bond thiolation of 1,3,4-oxadiazoles and related heteroarenes

(2012) Liang-Hua Zou et al.   CHEMICAL COMMUNICATIONS

Visible light-induced 3-sulfenylation of N-methylindoles with arylsulfonyl chlorides

(2012) Min Chen et al.   CHEMICAL COMMUNICATIONS

Iodine-catalyzed oxidative system for 3-sulfenylation of indoles with disulfides using DMSO as oxidant under ambient conditions in dimethyl carbonate

(2012) Wenlei Ge et al.   GREEN CHEMISTRY

Pyrazoles as Promising Scaffold for the Synthesis of Anti-Inflammatory and/or Antimicrobial Agent: A Review

(2012) Adnan A. Bekhit et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Novel C–H functionalization of arenes: palladium-catalyzed synthesis of diaryl sulfides

(2011) Pazhamalai Anbarasan et al.   CHEMICAL COMMUNICATIONS

TBHP-mediated oxidative thiolation of an sp3 C–H bond adjacent to a nitrogen atom in an amide

(2011) Ri-Yuan Tang et al.   CHEMICAL COMMUNICATIONS

Synthesis of di(hetero)aryl sulfides by directly using arylsulfonyl chlorides as a sulfur source

(2011) Qian Wu et al.   CHEMICAL COMMUNICATIONS

Transition-Metal-Catalyzed C−S, C−Se, and C−Te Bond Formation via Cross-Coupling and Atom-Economic Addition Reactions

(2011) Irina P. Beletskaya et al.   CHEMICAL REVIEWS

Intermolecular Dehydrogenative Heck Reactions

(2011) Jean Le Bras et al.   CHEMICAL REVIEWS

Catalytic Dehydrogenative Cross-Coupling: Forming Carbon−Carbon Bonds by Oxidizing Two Carbon−Hydrogen Bonds

(2011) Charles S. Yeung et al.   CHEMICAL REVIEWS

Structure Based Drug Design of Crizotinib (PF-02341066), a Potent and Selective Dual Inhibitor of Mesenchymal–Epithelial Transition Factor (c-MET) Kinase and Anaplastic Lymphoma Kinase (ALK)

(2011) J. Jean Cui et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of Pyrazoles via Electrophilic Cyclization

(2011) Metin Zora et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Mediated C–H Activation/C–S Cross-Coupling of Heterocycles with Thiols

(2011) Sadananda Ranjit et al.   JOURNAL OF ORGANIC CHEMISTRY

Ruthenium-Catalyzed Meta Sulfonation of 2-Phenylpyridines

(2011) Ourida Saidi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis and biological evaluation of some thiazolylpyrazole derivatives as dual anti-inflammatory antimicrobial agents

(2010) Adnan A. Bekhit et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Cu(II)-Mediated Methylthiolation of Aryl C−H Bonds with DMSO

(2010) Lingling Chu et al.   ORGANIC LETTERS

A reusable FeCl3·6H2O/cationic 2,2′-bipyridyl catalytic system for the coupling of aryl iodides with thiols in water under aerobic conditions

(2009) Wei-Yi Wu et al.   GREEN CHEMISTRY

Copper/Amino Acid Catalyzed Cross-Couplings of Aryl and Vinyl Halides with Nucleophiles†

(2008) Dawei Ma et al.   ACCOUNTS OF CHEMICAL RESEARCH

Iron-Catalyzed S-Arylation of Thiols with Aryl Iodides

(2008) Arkaitz Correa et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rhodium-Catalyzed Substitution Reaction of Aryl Fluorides with Disulfides:p-Orientation in the Polyarylthiolation of Polyfluorobenzenes

(2008) Mieko Arisawa et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY