Intramolecular functional group differentiation as a strategy for the synthesis of bridged bicyclic β-amino acids

Synthesis of a 2,5-Diazabicyclo[2.2.1]heptane-Derived α,β-Diamino Acid

(2015) Oleksandr Grygorenko et al.   SYNTHESIS-STUTTGART

Bicyclic β-amino acids

(2015) Oleksandr O. Grygorenko   TETRAHEDRON

N-[6-(4-Butanoyl-5-methyl-1H-pyrazol-1-yl)pyridazin-3-yl]-5-chloro-1-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-1H-indole-3-carboxamide (SAR216471), a Novel Intravenous and Oral, Reversible, and Directly Acting P2Y12 Antagonist

(2014) Christophe Boldron et al.   JOURNAL OF MEDICINAL CHEMISTRY

Oxabicyclooctane-Linked Novel Bacterial Topoisomerase Inhibitors as Broad Spectrum Antibacterial Agents

(2014) Sheo B. Singh et al.   ACS Medicinal Chemistry Letters

Diversity-Oriented Approaches to Unusual α-Amino Acids and Peptides: Step Economy, Atom Economy, Redox Economy, and Beyond

(2013) Sambasivarao Kotha et al.   JOURNAL OF ORGANIC CHEMISTRY

Quantifying the chemical beauty of drugs

(2012) G. Richard Bickerton et al.   Nature Chemistry

A chiral pool based approach to antipodes of α-cuparenone

(2012) Subhash P. Chavan et al.   TETRAHEDRON-ASYMMETRY

Bicyclic Conformationally Restricted Diamines

(2011) Oleksandr O. Grygorenko et al.   CHEMICAL REVIEWS

Integral Stereocontrolled Synthesis of a Spiro-norlignan, Sequosempervirin A: Revision of Absolute Configuration

(2011) Yuji Ito et al.   ORGANIC LETTERS

A Practical Asymmetric Synthesis of Isopropyl (1R,2S)-Dehydrocoronamate

(2011) Wenjun Tang et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Route to three-dimensional fragments using diversity-oriented synthesis

(2011) A. W. Hung et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Synthesis of 3-azabicyclo[4.1.0]heptane-1-carboxylic acid

(2010) Carmela Napolitano et al.   TETRAHEDRON

Synthesis of enantiopure (R,R)- and (S,S)-cis-2,3-propanoprolines

(2010) Natalia A. Kopylova et al.   TETRAHEDRON-ASYMMETRY

Diversity-oriented synthesis of bicyclic and tricyclic alkaloids

(2009) Mónica Díaz-Gavilán et al.   CHEMICAL COMMUNICATIONS

Diversity-Oriented Synthesis of Morpholine-Containing Molecular Scaffolds

(2009) Claudia Lalli et al.   CHEMISTRY-A EUROPEAN JOURNAL

Conformationally Restricted Nonchiral Pipecolic Acid Analogues

(2009) Dmytro S. Radchenko et al.   JOURNAL OF ORGANIC CHEMISTRY

Recent progress on the stereoselective synthesis of cyclic quaternary α-amino acids

(2009) Carlos Cativiela et al.   TETRAHEDRON-ASYMMETRY

Peptidomimetics, a synthetic tool of drug discovery

(2008) Josef Vagner et al.   CURRENT OPINION IN CHEMICAL BIOLOGY