Converting disulfide bridges in native peptides to stable methylene thioacetals

Acetone-Linked Peptides: A Convergent Approach for Peptide Macrocyclization and Labeling

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Peptide stapling techniques based on different macrocyclisation chemistries

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Discovery, Synthesis, and Structure–Activity Relationships of Conotoxins

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Selenoether oxytocin analogues have analgesic properties in a mouse model of chronic abdominal pain

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1,2,3-Triazoles as Amide Bond Mimics: Triazole Scan Yields Protease-Resistant Peptidomimetics for Tumor Targeting

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Multifaceted Roles of Disulfide Bonds. Peptides as Therapeutics

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A Perfluoroaryl-Cysteine SNAr Chemistry Approach to Unprotected Peptide Stapling

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Structurally Diverse Cyclisation Linkers Impose Different Backbone Conformations in Bicyclic Peptides

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Peptides As Therapeutics with Enhanced Bioactivity

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Peptoids: Bio-Inspired Polymers as Potential Pharmaceuticals

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Development of α-Helical Calpain Probes by Mimicking a Natural Protein–Protein Interaction

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Azapeptides and their therapeutic potential

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α-Conotoxin ImI Incorporating Stable Cystathionine Bridges Maintains Full Potency and Identical Three-Dimensional Structure

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Contemporary strategies for peptide macrocyclization

(2011) Christopher J. White et al.   Nature Chemistry

Modulating Oxytocin Activity and Plasma Stability by Disulfide Bond Engineering

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Cyclodepsipeptides - Potential Drugs and Lead Compounds in the Drug Development Process

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Synthetic therapeutic peptides: science and market

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Phage-encoded combinatorial chemical libraries based on bicyclic peptides

(2009) Christian Heinis et al.   Nature Chemical Biology

Towards Heat-stable Oxytocin Formulations: Analysis of Degradation Kinetics and Identification of Degradation Products

(2009) Andrea Hawe et al.   PHARMACEUTICAL RESEARCH

Peptidomimetics, a synthetic tool of drug discovery

(2008) Josef Vagner et al.   CURRENT OPINION IN CHEMICAL BIOLOGY

Oxytocin, Vasopressin, and the Neurogenetics of Sociality

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