Journal
SYNLETT
Volume 27, Issue 6, Pages 941-945Publisher
GEORG THIEME VERLAG KG
DOI: 10.1055/s-0035-1560548
Keywords
asymmetric synthesis; chirality; sulfoxides; indoles; total synthesis
Categories
Funding
- JSPS KAKENHI [25860014]
- Grants-in-Aid for Scientific Research [25860014] Funding Source: KAKEN
Ask authors/readers for more resources
The first example of an enantioselective intermolecular interrupted Pummerer reaction has been developed by the utilization of a C-2-symmetric chiral sulfoxide. The reaction was used for the enantioselective synthesis of C3a-substituted pyrroloindolines in a one-pot procedure starting from tryptamine. The synthetic utility of the reaction was further demonstrated by its application to the highly concise total synthesis of (+)-psychotriasine.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available