Second generation of thiazolylmannosides, FimH antagonists for E. coli-induced Crohn's disease
Published 2016 View Full Article
- Home
- Publications
- Publication Search
- Publication Details
Title
Second generation of thiazolylmannosides, FimH antagonists for E. coli-induced Crohn's disease
Authors
Keywords
-
Journal
ORGANIC & BIOMOLECULAR CHEMISTRY
Volume 14, Issue 16, Pages 3913-3925
Publisher
Royal Society of Chemistry (RSC)
Online
2016-03-23
DOI
10.1039/c6ob00424e
References
Ask authors/readers for more resources
Related references
Note: Only part of the references are listed.- Glycopolymers as Antiadhesives of E. coli Strains Inducing Inflammatory Bowel Diseases
- (2015) Xibo Yan et al. BIOMACROMOLECULES
- Thiourea-Bridged Nanodiamond Glycoconjugates as Inhibitors of Bacterial Adhesion
- (2015) Claudia Fessele et al. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
- Selective S-deacetylation inspired by native chemical ligation: practical syntheses of glycosyl thiols and drug mercapto-analogues
- (2015) Penghua Shu et al. GREEN CHEMISTRY
- FimH Antagonists: Bioisosteres To Improve the in Vitro and in Vivo PK/PD Profile
- (2015) Simon Kleeb et al. JOURNAL OF MEDICINAL CHEMISTRY
- Inhibition of type 1 fimbriae-mediated Escherichia coli adhesion and biofilm formation by trimeric cluster thiomannosides conjugated to diamond nanoparticles
- (2015) Manakamana Khanal et al. Nanoscale
- Inhibition profiles of mono- and polyvalent FimH antagonists against 10 different Escherichia coli strains
- (2015) T. Chalopin et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- 3-(Dimethylamino)-1-propylamine: A Cheap and Versatile Reagent for Removal of Byproducts in Carbohydrate Chemistry
- (2015) Sofie Meng Andersen et al. ORGANIC LETTERS
- Selective Antimicrobial and Antibiofilm Disrupting Properties of Functionalized Diamond Nanoparticles AgainstEscherichia coliandStaphylococcus aureus
- (2015) Manakamana Khanal et al. PARTICLE & PARTICLE SYSTEMS CHARACTERIZATION
- Development of Heptylmannoside-Based Glycoconjugate Antiadhesive Compounds against Adherent-Invasive Escherichia coli Bacteria Associated with Crohn's Disease
- (2015) A. Sivignon et al. mBio
- Glycomimetics versus Multivalent Glycoconjugates for the Design of High Affinity Lectin Ligands
- (2014) Samy Cecioni et al. CHEMICAL REVIEWS
- Towards bacterial adhesion-based therapeutics and detection methods
- (2014) Núria Parera Pera et al. MedChemComm
- Heptyl α-D-Mannosides Grafted on a β-Cyclodextrin Core To Interfere withEscherichia coliAdhesion: An In Vivo Multivalent Effect
- (2013) Julie Bouckaert et al. CHEMISTRY-A EUROPEAN JOURNAL
- Thiazolylaminomannosides As Potent Antiadhesives of Type 1 Piliated Escherichia coli Isolated from Crohn’s Disease Patients
- (2013) Sami Brument et al. JOURNAL OF MEDICINAL CHEMISTRY
- The Tyrosine Gate as a Potential Entropic Lever in the Receptor-Binding Site of the Bacterial Adhesin FimH
- (2012) Adinda Wellens et al. BIOCHEMISTRY
- Multivalent glycoconjugates as anti-pathogenic agents
- (2012) Anna Bernardi et al. CHEMICAL SOCIETY REVIEWS
- Antiadhesion Therapy for Urinary Tract Infections—A Balanced PK/PD Profile Proved To Be Key for Success
- (2012) Xiaohua Jiang et al. JOURNAL OF MEDICINAL CHEMISTRY
- Lead Optimization Studies on FimH Antagonists: Discovery of Potent and Orally Bioavailable Ortho-Substituted Biphenyl Mannosides
- (2012) Zhenfu Han et al. JOURNAL OF MEDICINAL CHEMISTRY
- Squaric Acid Monoamide Mannosides as Ligands for the Bacterial Lectin FimH: Covalent Inhibition or Not?
- (2011) Carsten Grabosch et al. CHEMBIOCHEM
- Clustering of Escherichia coli Type-1 Fimbrial Adhesins by Using Multimeric Heptyl α-D-Mannoside Probes with a Carbohydrate Core
- (2011) Mehdi Almant et al. CHEMISTRY-A EUROPEAN JOURNAL
- The Bacterial Lectin FimH, a Target for Drug Discovery - Carbohydrate Inhibitors of Type 1 Fimbriae-Mediated Bacterial Adhesion
- (2011) Mirja Hartmann et al. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
- Treatment and Prevention of Urinary Tract Infection with Orally Active FimH Inhibitors
- (2011) C. K. Cusumano et al. Science Translational Medicine
- The functional valency of dodecamannosylated fullerenes with Escherichia coli FimH—towards novel bacterial antiadhesives
- (2010) Maxime Durka et al. CHEMICAL COMMUNICATIONS
- FimH Antagonists for the Oral Treatment of Urinary Tract Infections: From Design and Synthesis to in Vitro and in Vivo Evaluation
- (2010) Tobias Klein et al. JOURNAL OF MEDICINAL CHEMISTRY
- Ultrasound-assisted synthesis of C-glycosides
- (2010) Dilip V. Jarikote et al. TETRAHEDRON LETTERS
- Synthetic Multimeric Heptyl Mannosides as Potent Antiadhesives of UropathogenicEscherichia coli
- (2009) Sébastien G. Gouin et al. ChemMedChem
- Intervening with Urinary Tract Infections Using Anti-Adhesives Based on the Crystal Structure of the FimH–Oligomannose-3 Complex
- (2008) Adinda Wellens et al. PLoS One
Find Funding. Review Successful Grants.
Explore over 25,000 new funding opportunities and over 6,000,000 successful grants.
ExploreAdd your recorded webinar
Do you already have a recorded webinar? Grow your audience and get more views by easily listing your recording on Peeref.
Upload Now