Iridium(iii)-catalyzed regioselective C7-sulfonamidation of indoles

Palladium-Catalyzed C–H Arylation of Indoles at the C7 Position

(2016) Youqing Yang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Direct Access to 7-Aminoindoles via Iridium-Catalyzed Mild C–H Amidation of N-Pivaloylindoles with Organic Azides

(2016) Youyoung Kim et al.   ORGANIC LETTERS

Transition-Metal-Catalyzed C–N Bond Forming Reactions Using Organic Azides as the Nitrogen Source: A Journey for the Mild and Versatile C–H Amination

(2015) Kwangmin Shin et al.   ACCOUNTS OF CHEMICAL RESEARCH

Transition Metal-Catalyzed CH Activation of Indoles

(2015) Alexander H. Sandtorv   ADVANCED SYNTHESIS & CATALYSIS

Rhodium(III)-Catalyzed Selective CH Cyanation of Indolines and Indoles with an Easily Accessible Cyano Source

(2015) Neeraj Kumar Mishra et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-Catalyzed (2+1) Annulation of Acetophenones with Maleimides: Direct Synthesis of Cyclopropanes

(2015) Srimanta Manna et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rhodium-Catalyzed Regioselective C7-Functionalization of N -Pivaloylindoles

(2015) Lanting Xu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Oxidative regioselective amination of chromones exposes potent inhibitors of the hedgehog signaling pathway

(2015) Rajarshi Samanta et al.   CHEMICAL COMMUNICATIONS

Rhodium(iii)-catalyzed C7-position C–H alkenylation and alkynylation of indolines

(2015) Xiao-Fei Yang et al.   CHEMICAL COMMUNICATIONS

A review on recent developments of indole-containing antiviral agents

(2015) Ming-Zhi Zhang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Rh(III)-Catalyzed C7-Thiolation and Selenation of Indolines

(2015) Wucheng Xie et al.   JOURNAL OF ORGANIC CHEMISTRY

Iridium(III)-Catalyzed C-7 Selective C–H Alkynylation of Indolines at Room Temperature

(2015) Yunxiang Wu et al.   JOURNAL OF ORGANIC CHEMISTRY

Mild Rh(III)-Catalyzed C7-Allylation of Indolines with Allylic Carbonates

(2015) Jihye Park et al.   JOURNAL OF ORGANIC CHEMISTRY

Access to Six- and Seven-Membered 1,7-Fused Indolines via Rh(III)-Catalyzed Redox-Neutral C7-Selective C–H Functionalization of Indolines with Alkynes and Alkenes

(2015) Xuan Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Total Synthesis of Verruculogen and Fumitremorgin A Enabled by Ligand-Controlled C–H Borylation

(2015) Yu Feng et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Iridium(III)-Catalyzed Direct Arylation of C–H Bonds with Diaryliodonium Salts

(2015) Pan Gao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Atom-Economical Transformation of Diaryliodonium Salts: Tandem C–H and N–H Arylation of Indoles

(2015) Sachin G. Modha et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Expedient Synthesis of Pyrroloquinolinones by Rh-Catalyzed Annulation of N-Carbamoyl Indolines with Alkynes through a Directed C–H Functionalization/C–N Cleavage Sequence

(2015) Xiao-Fei Yang et al.   ORGANIC LETTERS

Copper(I)-Catalyzed Radical Addition of Acetophenones to Alkynes in Furan Synthesis

(2015) Srimanta Manna et al.   ORGANIC LETTERS

Iridium- and Rhodium-Catalyzed C–H Activation and Formyl Alkynylation of Benzaldehydes under Chelation-Assistance

(2015) He Wang et al.   ORGANIC LETTERS

Palladium-Catalyzed Regioselective Decarboxylative Alkylation of Arenes and Heteroarenes with Aliphatic Carboxylic Acids

(2015) Chanchal Premi et al.   ORGANIC LETTERS

Hypervalent Iodine(III) in Direct Oxidative Amination of Arenes with Heteroaromatic Amines

(2015) Srimanta Manna et al.   ORGANIC LETTERS

Catalytic Methods for Aromatic C–H Amination: An Ideal Strategy for Nitrogen-Based Functional Molecules

(2015) Jiao Jiao et al.   ACS Catalysis

Iridium(I)-Catalyzed Direct CH Bond Alkylation of the C-7 Position of Indolines with Alkenes

(2014) Shiguang Pan et al.   ADVANCED SYNTHESIS & CATALYSIS

Air-Stable Carbonyl(pentamethylcyclopentadienyl)cobalt Diiodide Complex as a Precursor for Cationic (Pentamethylcyclopentadienyl)cobalt(III) Catalysis: Application for Directed C-2 Selective CH Amidation of Indoles

(2014) Bo Sun et al.   ADVANCED SYNTHESIS & CATALYSIS

Iridium-Catalyzed Direct CH Amidation with Weakly Coordinating Carbonyl Directing Groups under Mild Conditions

(2014) Jinwoo Kim et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Cascade Multicomponent Synthesis of Indoles, Pyrazoles, and Pyridazinones by Functionalization of Alkenes

(2014) Kiran Matcha et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Methylation of CH Bonds Using CO2and H2

(2014) Yuehui Li et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalytic Oxidative Annulation of Benzamide Derivatives with Alkynes

(2014) Srimanta Manna et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Metal-Free Annulation of Arenes with 2-Aminopyridine Derivatives: The Methyl Group as a Traceless Non-Chelating Directing Group

(2014) Srimanta Manna et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Decarboxylative acylation of indolines with α-keto acids under palladium catalysis: a facile strategy for the synthesis of 7-substituted indoles

(2014) Minyoung Kim et al.   CHEMICAL COMMUNICATIONS

Ruthenium-Catalyzed C7 Amidation of Indoline CH Bonds with Sulfonyl Azides

(2014) Changduo Pan et al.   CHEMISTRY-A EUROPEAN JOURNAL

Rhodium(III)- and Iridium(III)-Catalyzed C7 Alkylation of Indolines with Diazo Compounds

(2014) Wen Ai  et al.   CHEMISTRY-A EUROPEAN JOURNAL

Hypervalent Iodine-Mediated Selective Oxidative Functionalization of (Thio)chromones with Alkanes

(2014) Rishikesh Narayan et al.   CHEMISTRY-A EUROPEAN JOURNAL

Ir(III)-Catalyzed C7-Position-Selective Oxidative CH Alkenylation of Indolines with Alkenes in Air

(2014) Shiguang Pan et al.   Chemistry-An Asian Journal

IrIII-Catalyzed Direct C-7 Amidation of Indolines with Sulfonyl, Acyl, and Aryl Azides at Room Temperature

(2014) Wei Hou et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Iridium(III)-Catalyzed Direct C-7 Amination of Indolines with Organic Azides

(2014) Kwangmin Shin et al.   JOURNAL OF ORGANIC CHEMISTRY

C7-Derivatization of C3-Alkylindoles Including Tryptophans and Tryptamines

(2014) Richard P. Loach et al.   JOURNAL OF ORGANIC CHEMISTRY

Mild Aminoacylation of Indoles and Pyrroles through a Three-Component Reaction with Ynol Ethers and Sulfonyl Azides

(2014) Joshua S. Alford et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cu(II)-Mediated C–H Amidation and Amination of Arenes: Exceptional Compatibility with Heterocycles

(2014) Ming Shang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rh(III)- and Ir(III)-Catalyzed C–H Alkynylation of Arenes under Chelation Assistance

(2014) Fang Xie et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Oxygen Atom Transfer to a Half-Sandwich Iridium Complex: Clean Oxidation Yielding a Molecular Product

(2014) Christopher R. Turlington et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rhodium(iii)-catalyzed regioselective C2-amidation of indoles with N-(2,4,6-trichlorobenzoyloxy)amides and its synthetic application to the development of a novel potential PPARγ modulator

(2014) Jingjing Shi et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Exceptionally Mild Palladium(II)-Catalyzed Dehydrogenative C–H/C–H Arylation of Indolines at the C-7 Position under Air

(2014) Lin-Yu Jiao et al.   ORGANIC LETTERS

Comparative Investigations of Cp*-Based Group 9 Metal-Catalyzed Direct C–H Amination of Benzamides

(2014) Travis M. Figg et al.   ORGANOMETALLICS

Oxidative C–H amination reactions

(2013) Marie-Laure Louillat et al.   CHEMICAL SOCIETY REVIEWS

Oxidative Palladium(II)-Catalyzed Dehydrogenative CH/CH Cross-Coupling of 2,3-Substituted Indolines with Arenes at the C7 Position

(2013) Lin-Yu Jiao et al.   CHEMISTRY-A EUROPEAN JOURNAL

Regioselective C2 Oxidative Olefination of Indoles and Pyrroles through Cationic Rhodium(III)-Catalyzed CH Bond Activation

(2013) Bin Li et al.   CHEMISTRY-A EUROPEAN JOURNAL

Iridium-Catalyzed Direct Arene C–H Bond Amidation with Sulfonyl- and Aryl Azides

(2013) Donggun Lee et al.   JOURNAL OF ORGANIC CHEMISTRY

Ir(III)-Catalyzed Mild C–H Amidation of Arenes and Alkenes: An Efficient Usage of Acyl Azides as the Nitrogen Source

(2013) Jaeyune Ryu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Biomedical Importance of Indoles

(2013) Nagendra Kaushik et al.   MOLECULES

Oxidative Palladium(II)-Catalyzed C-7 Alkenylation of Indolines

(2013) Lin-Yu Jiao et al.   ORGANIC LETTERS

Direct Olefination at the C-4 Position of Tryptophan via C–H Activation: Application to Biomimetic Synthesis of Clavicipitic Acid

(2013) Qiang Liu et al.   ORGANIC LETTERS

Rhodium(III)-Catalyzed Direct Regioselective Synthesis of 7-Substituted Indoles

(2013) Zengqiang Song et al.   ORGANIC LETTERS

Mild and Efficient C2-Alkenylation of Indoles with Alkynes Catalyzed by a Cobalt Complex

(2012) Zhenhua Ding et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Inhibitors of HIV-1 attachment. Part 7: Indole-7-carboxamides as potent and orally bioavailable antiviral agents

(2012) Kap-Sun Yeung et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Therapeutic potential and molecular mechanism of a novel sulfonamide anticancer drug, indisulam (E7070) in combination with CPT-11 for cancer treatment

(2012) Yoichi Ozawa et al.   CANCER CHEMOTHERAPY AND PHARMACOLOGY

Ir(I)-Catalyzed C–H Bond Alkylation of C2-Position of Indole with Alkenes: Selective Synthesis of Linear or Branched 2-Alkylindoles

(2012) Shiguang Pan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Pd(II)-Catalyzed Regioselective 2-Alkylation of Indoles via a Norbornene-Mediated C–H Activation: Mechanism and Applications

(2012) Lei Jiao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rhodium-catalyzed regioselective amidation of indoles with sulfonyl azides via C–H bond activation

(2012) Jingjing Shi et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Theoretical Study of Mechanism and Selectivity of Copper-Catalyzed C–H Bond Amidation of Indoles

(2011) Stefano Santoro et al.   JOURNAL OF ORGANIC CHEMISTRY

Mild and Selective Ru-Catalyzed Formylation and Fe-Catalyzed Acylation of Free (N–H) Indoles Using Anilines as the Carbonyl Source

(2011) Wenliang Wu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-/Copper-Catalyzed Regioselective Amination and Chloroamination of Indoles

(2011) Xue-Yuan Liu et al.   ORGANIC LETTERS

Copper-Catalyzed Highly Regioselective Oxidative CH Bond Amidation of 2-Arylpyridine Derivatives and 1-Methylindoles

(2010) Qi Shuai et al.   ADVANCED SYNTHESIS & CATALYSIS

Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety

(2010) Anna J. Kochanowska-Karamyan et al.   CHEMICAL REVIEWS

Insertion of nitrene and chalcogenolate groups into the Ir–C σ bond in a cyclometalated iridium(III) complex

(2010) Yiu-Keung Sau et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

Iridium-Catalyzed, Silyl-Directed Borylation of Nitrogen-Containing Heterocycles

(2010) Daniel W. Robbins et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rh Catalyzed Olefination and Vinylation of Unactivated Acetanilides

(2010) Frederic W. Patureau et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rhodium(III)-Catalyzed Intermolecular Hydroarylation of Alkynes

(2010) Derek J. Schipper et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium(II)-Catalyzed Regioselective Direct C2 Alkenylation of Indoles and Pyrroles Assisted by theN-(2-Pyridyl)sulfonyl Protecting Group

(2009) Alfonso García-Rubia et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Functionalization of Indoles in a New Dimension

(2009) Marco Bandini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Direct Arylation of (Hetero)Arenes with Aryl Boronic Acids

(2008) Shang-Dong Yang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Cu(II)-Catalyzed Direct and Site-Selective Arylation of Indoles Under Mild Conditions

(2008) Robert J. Phipps et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY