N-Bromosuccinimide promoted and base switchable one pot synthesis of α-imido and α-amino ketones from styrenes

Stereoselective Actions of Methylenedioxypyrovalerone (MDPV) To Inhibit Dopamine and Norepinephrine Transporters and Facilitate Intracranial Self-Stimulation in Rats

(2015) R. Kolanos et al.   ACS Chemical Neuroscience

Chiral Resolution and Absolute Configuration of the Enantiomers of the Psychoactive “Designer Drug” 3,4-Methylenedioxypyrovalerone

(2015) Masaki Suzuki et al.   CHIRALITY

Multi-step synthesis strategies towards 1,2-amino alcohols with special emphasis on phenylpropanolamines

(2015) Torsten Sehl et al.   JOURNAL OF MOLECULAR CATALYSIS B-ENZYMATIC

Catalyst-Free and Metal-Free Electrophilic Bromoamidation of Unactivated Olefins Using the N-Bromosuccinimide/Sulfonamide Protocol

(2015) Wesley Zongrong Yu et al.   JOURNAL OF ORGANIC CHEMISTRY

A Versatile and One-Pot Strategy to Synthesize α-Amino Ketones from Benzylic Secondary Alcohols Using N-Bromosuccinimide

(2015) Somraj Guha et al.   ORGANIC LETTERS

Metal-free protocol for the synthesis of α-bromo ketones from olefins using TsNBr2

(2015) Kamal Krishna Rajbongshi et al.   TETRAHEDRON LETTERS

Transition-Metal-Free Oxidative α-C–H Amination of Ketones via a Radical Mechanism: Mild Synthesis of α-Amino Ketones

(2014) Qing Jiang et al.   JOURNAL OF ORGANIC CHEMISTRY

Diastereoselective synthesis of functionalized pyrrolidines through N-bromosuccinimide-induced aziridine ring expansion cascade of cinnamylaziridine

(2014) Jing Zhou et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Hybrid Dopamine Uptake Blocker–Serotonin Releaser Ligands: A New Twist on Transporter-Focused Therapeutics

(2014) Bruce E. Blough et al.   ACS Medicinal Chemistry Letters

“Deconstruction” of the Abused Synthetic Cathinone Methylenedioxypyrovalerone (MDPV) and an Examination of Effects at the Human Dopamine Transporter

(2013) Renata Kolanos et al.   ACS Chemical Neuroscience

Substituted methcathinones differ in transporter and receptor interactions

(2013) Amy J. Eshleman et al.   BIOCHEMICAL PHARMACOLOGY

Simple Catalytic Mechanism for the Direct Coupling of α-Carbonyls with Functionalized Amines: A One-Step Synthesis of Plavix

(2013) Ryan W. Evans et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The novel recreational drug 3,4-methylenedioxypyrovalerone (MDPV) is a potent psychomotor stimulant: Self-administration and locomotor activity in rats

(2013) S.M. Aarde et al.   NEUROPHARMACOLOGY

Ag- and Au-Catalyzed Addition of Alcohols to Ynimides: β-Regioselective Carbonylation and Production of Oxazoles

(2013) Takuya Sueda et al.   ORGANIC LETTERS

Catalytic Intermolecular Haloamidation of Simple Alkenes with N-Halophthalimide as Both Nitrogen and Halogen Source

(2013) Lu Song et al.   ORGANIC LETTERS

N-Bromosuccinimide/1,8-Diazabicyclo[5.4.1]undec-7-ene Combination: β-Amination of Chalcones via a Tandem Bromoamination/Debromination Sequence

(2013) Ying Wei et al.   ORGANIC LETTERS

N-Bromoimide/DBU Combination as a New Strategy for Intermolecular Allylic Amination

(2013) Ying Wei et al.   ORGANIC LETTERS

Mephedrone and methylenedioxypyrovalerone (MDPV), major constituents of “bath salts,” produce opposite effects at the human dopamine transporter

(2013) Krasnodara Cameron et al.   PSYCHOPHARMACOLOGY

NIS-Catalyzed Reactions: Amidation of Acetophenones and Oxidative Amination of Propiophenones

(2012) Manjunath Lamani et al.   CHEMISTRY-A EUROPEAN JOURNAL

Highly Enantioselective Electrophilic α-Bromination of Enecarbamates: Chiral Phosphoric Acid and Calcium Phosphate Salt Catalysts

(2012) Aurélien Alix et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Powerful Cocaine-Like Actions of 3,4-Methylenedioxypyrovalerone (MDPV), a Principal Constituent of Psychoactive ‘Bath Salts’ Products

(2012) Michael H Baumann et al.   NEUROPSYCHOPHARMACOLOGY

Halonium-Initiated C–O Bond Formation via Umpolung of α-Carbon to the Carbonyl: Efficient Access to 5-Amino-3(2H)-furanones

(2012) Ying Wei et al.   ORGANIC LETTERS

One-Pot Cascade Leading to Direct α-Imidation of Ketones by a Combination of N-Bromosuccinimide and 1,8-Diazabicyclo[5.4.1]undec-7-ene

(2012) Ying Wei et al.   ORGANIC LETTERS

Synthesis of α-Amino Ketones from Terminal Alkynes via Rhodium-Catalyzed Denitrogenative Hydration of N-Sulfonyl-1,2,3-triazoles

(2011) Tomoya Miura et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

N-Bromosuccinimide Promoted One-Pot Synthesis of Guanidine: Scope and Mechanism

(2011) Ling Zhou et al.   ORGANIC LETTERS

One-Pot Multicomponent Synthesis of Diversely Substituted 2-Aminopyrroles. A Short General Synthesis of Rigidins A, B, C, and D

(2011) Liliya V. Frolova et al.   ORGANIC LETTERS

Scope and Mechanistic Studies of Electrophilic Alkoxyetherification

(2011) Jie Chen et al.   ORGANIC LETTERS

Catalytic Asymmetric Bromoamination of Chalcones: Highly Efficient Synthesis of Chiral α-Bromo-β-Amino Ketone Derivatives

(2010) Yunfei Cai et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Bromolactonization Using Amino-thiocarbamate Catalyst

(2010) Ling Zhou et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-catalyzed amination of (bromophenyl)ethanolamine for a concise synthesis of aniline-containing analogues of NMDA NR2B antagonist ifenprodil

(2010) Cédric Bouteiller et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis and Biological Evaluation of Bupropion Analogues as Potential Pharmacotherapies for Cocaine Addiction

(2009) F. Ivy Carroll et al.   JOURNAL OF MEDICINAL CHEMISTRY

Environmentally benign electrophilic and radical bromination ‘on water’: H2O2–HBr system versus N-bromosuccinimide

(2009) Ajda Podgoršek et al.   TETRAHEDRON

Asymmetric Hydrogenation of Aromatic Ketones Catalyzed by the TolBINAP/DMAPEN−Ruthenium(II) Complex: A Significant Effect ofN-Substituents of Chiral 1,2-Diamine Ligands on Enantioselectivity

(2008) Hirohito Ooka et al.   JOURNAL OF ORGANIC CHEMISTRY