Antibacterial Activity of Enrofloxacin and Ciprofloxacin Derivatives ofβ-Octaarginine

Fluoroquinolone-Gyrase-DNA Complexes

(2014) Arkady Mustaev et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Correction: Structural Basis of Gate-DNA Breakage and Resealing by Type II Topoisomerases

(2014) Ivan Laponogov et al.   PLoS One

Curb challenges of the “Trojan Horse” approach: Smart strategies in achieving effective yet safe cell-penetrating peptide-based drug delivery

(2013) Yongzhuo Huang et al.   ADVANCED DRUG DELIVERY REVIEWS

Improved Efficacy of Fosmidomycin against Plasmodium and Mycobacterium Species by Combination with the Cell-Penetrating Peptide Octaarginine

(2013) Christof Sparr et al.   ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

Trihydroxamate Siderophore–Fluoroquinolone Conjugates Are Selective Sideromycin Antibiotics that Target Staphylococcus aureus

(2013) Timothy A. Wencewicz et al.   BIOCONJUGATE CHEMISTRY

Permeation through Phospholipid Bilayers, Skin-Cell Penetration, Plasma Stability, and CD Spectra ofα- andβ-Oligoproline Derivatives

(2013) Beata Kolesinska et al.   CHEMISTRY & BIODIVERSITY

Enantiomeric and Diastereoisomeric (Mixed)L/ D-Octaarginine Derivatives - A Simple Way of Modulating the Properties of Cell-Penetrating Peptides

(2013) Nirupam Purkayastha et al.   CHEMISTRY & BIODIVERSITY

Is there a future for cell-penetrating peptides in oligonucleotide delivery?

(2013) Soo Hyeon Lee et al.   EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS

Cell-penetrating peptides: 20 years later, where do we stand?

(2013) Chérine Bechara et al.   FEBS LETTERS

Inhibitory effect of short cationic homopeptides against Gram-positive bacteria

(2013) Fanny Guzmán et al.   JOURNAL OF PEPTIDE SCIENCE

Ratiometric Activatable Cell-Penetrating Peptides Provide Rapid In Vivo Readout of Thrombin Activation

(2012) Michael Whitney et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

MBX-500, a Hybrid Antibiotic withIn VitroandIn VivoEfficacy against Toxigenic Clostridium difficile

(2012) Michelle M. Butler et al.   ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

Zwitterionic Guanidine-Based Oligomers Mimicking Cell-Penetrating Peptides as a Nontoxic Alternative to Cationic Polymers to Enhance the Cellular Uptake of Micelles

(2012) Yoseop Kim et al.   BIOMACROMOLECULES

Synthesis and antibacterial activity of conjugates between norfloxacin and analogues of the siderophore vanchrobactin

(2012) Alba Souto et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Cell-penetrating Peptides as a Novel Transdermal Drug Delivery System

(2012) Saman A. Nasrollahi et al.   Chemical Biology & Drug Design

Cell-penetrating peptides: classes, origin, and current landscape

(2012) Francesca Milletti   DRUG DISCOVERY TODAY

Cell entry of cell penetrating peptides: tales of tails wagging dogs

(2012) Arwyn T. Jones et al.   JOURNAL OF CONTROLLED RELEASE

Direct cytosolic delivery of cargoes in vivo by a chimera consisting of D- and L-arginine residues

(2012) Yan Ma et al.   JOURNAL OF CONTROLLED RELEASE

Cell-penetrating Peptides as Versatile Vehicles for Oligonucleotide Delivery

(2012) Helerin Margus et al.   MOLECULAR THERAPY

Cell-penetrating peptides: breaking through to the other side

(2012) Erez Koren et al.   TRENDS IN MOLECULAR MEDICINE

Exploiting bacterial DNA gyrase as a drug target: current state and perspectives

(2011) Frédéric Collin et al.   APPLIED MICROBIOLOGY AND BIOTECHNOLOGY

On the Mechanism of Eukaryotic Cell Penetration by α- and β-Oligoarginines - Targeting Infected Erythro­cytes

(2011) Faustin Kamena et al.   CHEMISTRY & BIODIVERSITY

Conceptually New Entries into Cells

(2011) Javier Montenegro et al.   CHIMIA

Transduction of peptides and proteins into live cells by cell penetrating peptides

(2011) Franziska Mussbach et al.   JOURNAL OF CELLULAR BIOCHEMISTRY

Type IIA topoisomerase inhibition by a new class of antibacterial agents

(2010) Benjamin D. Bax et al.   NATURE

Structural basis of quinolone inhibition of type IIA topoisomerases and target-mediated resistance

(2010) Alexandre Wohlkonig et al.   NATURE STRUCTURAL & MOLECULAR BIOLOGY

A Unique 45-Amino-Acid Region in the Toprim Domain ofPlasmodium falciparumGyrase B Is Essential for Its Activity

(2009) Ashraf Dar et al.   EUKARYOTIC CELL

Structural insight into the quinolone–DNA cleavage complex of type IIA topoisomerases

(2009) Ivan Laponogov et al.   NATURE STRUCTURAL & MOLECULAR BIOLOGY

β-Peptidic Peptidomimetics

(2008) Dieter Seebach et al.   ACCOUNTS OF CHEMICAL RESEARCH

Inhibition of Herpes Simplex Virus Type 1 Infection by Cationic  -Peptides

(2008) R. Akkarawongsa et al.   ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

Physicochemical Properties of Antibacterial Compounds: Implications for Drug Discovery

(2008) Rosemarie O’Shea et al.   JOURNAL OF MEDICINAL CHEMISTRY

Dual Mechanism of Bacterial Lethality for a Cationic Sequence-Random Copolymer that Mimics Host-Defense Antimicrobial Peptides

(2008) Raquel F. Epand et al.   JOURNAL OF MOLECULAR BIOLOGY

Single-Molecule Motions of Oligoarginine Transporter Conjugates on the Plasma Membrane of Chinese Hamster Ovary Cells

(2008) H.-L. Lee et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Overcoming multidrug resistance of small-molecule therapeutics through conjugation with releasable octaarginine transporters

(2008) E. A. Dubikovskaya et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Function-Oriented Synthesis, Step Economy, and Drug Design

(2007) Paul A. Wender et al.   ACCOUNTS OF CHEMICAL RESEARCH

The design of guanidinium-rich transporters and their internalization mechanisms

(2007) Paul A. Wender et al.   ADVANCED DRUG DELIVERY REVIEWS

Live-cell analysis of cell penetration ability and toxicity of oligo-arginines

(2007) Gisela Tünnemann et al.   JOURNAL OF PEPTIDE SCIENCE