A practical protocol for large‐scale copper‐mediated radioiodination of organoboronic precursors: Radiosynthesis of [123I]KX‐1 for Auger radiotherapy

Preclinical Efficacy of a PARP-1 Targeted Auger-Emitting Radionuclide in Prostate Cancer

(2023) Sreeja Sreekumar et al.   INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES

Effect of Water on Direct Radioiodination of Small Molecules/Peptides Using Copper-Mediated Iododeboronation in Water–Alcohol Solvent

(2023) Yuto Kondo et al.   ACS Omega

Copper-mediated radioiodination and radiobromination via aryl boronic precursor and its application to 125I/77Br–labeled prostate-specific membrane antigen imaging probes

(2022) Yuto Kondo et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Copper‐mediated radioiodination reaction through aryl boronic acid or ester precursor and its application to direct radiolabeling of a cyclic peptide

(2021) Yuto Kondo et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

PARP Theranostic Auger Emitters Are Cytotoxic in BRCA Mutant Ovarian Cancer and Viable Tumors from Ovarian Cancer Patients Enable Ex-Vivo Screening of Tumor Response

(2020) Aladdin Riad et al.   MOLECULES

Rapid Cu-Catalyzed [211At]Astatination and [125I]Iodination of Boronic Esters at Room Temperature

(2018) Sean W. Reilly et al.   ORGANIC LETTERS

Radiosynthesis of SPECT tracers via a copper mediated 123I iodination of (hetero)aryl boron reagents

(2016) Thomas C. Wilson et al.   CHEMICAL COMMUNICATIONS

A Highly Efficient Copper-Mediated Radioiodination Approach Using Aryl Boronic Acids

(2016) Pu Zhang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Copper-Mediated Aromatic Radiofluorination Revisited: Efficient Production of PET Tracers on a Preparative Scale

(2015) Boris D. Zlatopolskiy et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of [18F]Arenes via the Copper-Mediated [18F]Fluorination of Boronic Acids

(2015) Andrew V. Mossine et al.   ORGANIC LETTERS