Journal
ORGANIC LETTERS
Volume 17, Issue 23, Pages 5780-5783Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.5b02875
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Funding
- NIH [GM073836, T32-EB005172]
- US DOE [DE-SC0012484]
- Alzheimer's Association [NIRP-14-305669]
- Merck
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A copper-mediated radiofluorination of aryl- and vinylboronic acids with (KF)-F-18 is described. This method exhibits high functional group tolerance and is effective for the radiofluorination of a range of electron-deficient, -neutral, and -rich aryl-, heteroaryl-, and vinylboronic acids. This method has been applied to the synthesis of [F-18]FPEB, a PET radiotracer for quantifying metabotropic glutamate 5 receptors.
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