Discovery of a Potent and Selective STAT5 PROTAC Degrader with Strong Antitumor Activity In Vivo in Acute Myeloid Leukemia
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Title
Discovery of a Potent and Selective STAT5 PROTAC Degrader with Strong Antitumor Activity In Vivo in Acute Myeloid Leukemia
Authors
Keywords
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Journal
Journal of Medicinal Chemistry
Volume -, Issue -, Pages -
Publisher
American Chemical Society (ACS)
Online
2023-02-04
DOI
10.1021/acs.jmedchem.2c01665
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Note: Only part of the references are listed.- A selective small-molecule STAT5 PROTAC degrader capable of achieving tumor regression in vivo
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