Enantioselective Cascade Michael/Hemiaminal Formation of α,β-Unsaturated Iminoindoles with Aldehydes Using a Chiral Aminomethylpyrrolidine Catalyst Bearing a SO2C6F5 Group as a Strongly Electron Withdrawing Arylsulfonyl Group

Construction of Enantioenriched 4,5,6,7‐Tetrahydrofuro[2,3‐ b ]pyridines through a Multicatalytic Sequence Merging Gold and Amine Catalysis

(2021) Manon Genet et al.   ADVANCED SYNTHESIS & CATALYSIS

Isothiourea-Catalyzed Enantioselective Synthesis of Tetrahydro-α-carbolinones

(2020) Honglei Liu et al.   ORGANIC LETTERS

Enantioselective Dearomative Cyclization of Homotryptamines with Allenamides into Indolo[2,3‐ b ]quinolines

(2020) Soumen Biswas et al.   ADVANCED SYNTHESIS & CATALYSIS

Bifunctional Brønsted Base Catalyzed [3 + 3] Annulations of Indolin-2-imines and α,β-Unsaturated Imides: An Enantioselective Approach to α-Carbolinones

(2020) Lin Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

Discovery and Total Synthesis of a Bis(cyclotryptamine) Alkaloid Bearing the Elusive Piperidinoindoline Scaffold

(2020) Jordan J. Dotson et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Hypoiodite-Catalyzed Chemoselective Tandem Oxidation of Homotryptamines to Peroxy- and Epoxytetrahydropyridoindolenines

(2020) Muhammet Uyanik et al.   ORGANIC LETTERS

Prevalence of Diarylprolinol Silyl Ethers as Catalysts in Total Synthesis and Patents

(2019) Gabriel J. Reyes-Rodríguez et al.   CHEMICAL REVIEWS

Profiling the Privileges of Pyrrolidine-Based Catalysts in Asymmetric Synthesis - from Polar to Light-Driven Radical Chemistry

(2019) Alberto Vega Penaloza et al.   ACS Catalysis

Total Synthesis and Anti-Cancer Activity of All Known Communesin Alkaloids and Related Derivatives

(2019) Matthew M. Pompeo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Iminium and enamine catalysis in enantioselective photochemical reactions

(2018) You-Quan Zou et al.   CHEMICAL SOCIETY REVIEWS

A catalytic N-deacylative alkylation approach to hexahydropyrrolo[2,3-b]indole alkaloids

(2018) Nivesh Kumar et al.   CHEMICAL COMMUNICATIONS

Construction of Azepino[2,3-b]indole Core via Sulfur Ylide Mediated Annulations

(2018) Jun-Long Li et al.   ORGANIC LETTERS

Highly Stereoselective Assembly of α-Carbolinone Skeletons via N-Heterocyclic Carbene-Catalyzed [4 + 2] Annulations

(2018) Kai-Chuan Yang et al.   ORGANIC LETTERS

Structurally Diverse Alkaloids from the Seeds of Peganum harmala

(2017) Kai-Bo Wang et al.   JOURNAL OF NATURAL PRODUCTS

Recent Advances in Asymmetric Organocatalyzed Conjugate Additions to Nitroalkenes

(2017) Diego Alonso et al.   MOLECULES

Synthesis of Dihydropyridinone-Fused Indoles and α-Carbolines via N-Heterocyclic Carbene-Catalyzed [3 + 3] Annulation of Indolin-2-imines and Bromoenals

(2017) Liang Yi et al.   ORGANIC LETTERS

Cyclohepta[b]indoles: A Privileged Structure Motif in Natural Products and Drug Design

(2016) Erik Stempel et al.   ACCOUNTS OF CHEMICAL RESEARCH

Chaetominine reduces MRP1-mediated drug resistance via inhibiting PI3K/Akt/Nrf2 signaling pathway in K562/Adr human leukemia cells

(2016) Jingyun Yao et al.   BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS

Assessment of the Cytotoxic and Apoptotic Eἀects of Chaetominine in a Human Leukemia Cell Line

(2016) Jingyun Yao et al.   Biomolecules & Therapeutics

Indoles — A promising scaffold for drug development

(2016) T.V. Sravanthi et al.   EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES

The Construction of 3-Methyl-4-arylpiperidinesviaatrans- Perhydroindolic Acid-Catalyzed Asymmetric Aza-Diels-Alder Reaction

(2015) Qianjin An et al.   ADVANCED SYNTHESIS & CATALYSIS

The Diarylprolinol Silyl Ethers: Ten Years After

(2015) Bjarke S. Donslund et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Concise Total Synthesis of Dehaloperophoramidine

(2015) Kirill Popov et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Indole Derivatives as Anticancer Agents for Breast Cancer Therapy: A Review

(2015) Jagpreet Singh Sidhu et al.   Anti-Cancer Agents in Medicinal Chemistry

Regioselective Csp2–H dual functionalization of indoles using hypervalent iodine(iii): bromo-amination via 1,3-migration of imides on indolyl(phenyl)iodonium imides

(2015) Katsuhiko Moriyama et al.   CHEMICAL COMMUNICATIONS

A review on recent developments of indole-containing antiviral agents

(2015) Ming-Zhi Zhang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Indole Alkaloids from Chaetomium globosum

(2015) Guo-Bo Xu et al.   JOURNAL OF NATURAL PRODUCTS

Marine Indole Alkaloids

(2015) Natalie Netz et al.   Marine Drugs

Simple indole alkaloids and those with a nonrearranged monoterpenoid unit

(2015) Minoru Ishikura et al.   NATURAL PRODUCT REPORTS

A facile and efficient synthesis of hexahydro-1H-pyrido[2,3-b]indol-2-one scaffolds via a sequential Michael addition/amidation/reductive cyclization process

(2015) Xiong-Li Liu et al.   TETRAHEDRON

A catalytic asymmetric total synthesis of (−)-perophoramidine

(2015) B. M. Trost et al.   Chemical Science

Aminocatalysis: Beyond Steric Shielding and Hydrogen-Bonding

(2014) Bruno Matos Paz et al.   CHEMISTRY-A EUROPEAN JOURNAL

Vascular L-Type Ca2+ Channel Blocking Activity of Sulfur-Containing Indole Alkaloids from Glycosmis petelotii

(2014) Nguyen Manh Cuong et al.   JOURNAL OF NATURAL PRODUCTS

Ir-Catalyzed Reverse Prenylation of 3-Substituted Indoles: Total Synthesis of (+)-Aszonalenin and (−)-Brevicompanine B

(2014) Jonathan Ruchti et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Studies Toward Communesin F: A Diels–Alder Approach

(2014) Jakob Danielsson et al.   ORGANIC LETTERS

Visible Light-Induced Aerobic Oxyamidation of Indoles: A Photocatalytic Strategy for the Preparation of Tetrahydro-5H-indolo[2,3-b]quinolinols

(2013) Jing An et al.   ADVANCED SYNTHESIS & CATALYSIS

The four-step total synthesis of (−)-chaetominine

(2013) Qi-Long Peng et al.   CHEMICAL COMMUNICATIONS

Hydrogen-Bonding in Aminocatalysis: From Proline and Beyond

(2013) Łukasz Albrecht et al.   CHEMISTRY-A EUROPEAN JOURNAL

Asymmetric Total Synthesis of Neoxaline

(2013) Tetsuya Ideguchi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The Synthesis of Indoline and Benzofuran Scaffolds Using a Suzuki–Miyaura Coupling/Oxidative Cyclization Strategy

(2013) Somnath Jana et al.   ORGANIC LETTERS

Double Annulative Cascade of Tryptophan-Containing Peptides Triggered by Selectfluor

(2013) Bret Tréguier et al.   ORGANIC LETTERS

Asymmetric aza-Diels-Alder and Cation-olefin Cyclization Sequence: a Concise Way to Fused Chiral Cyclopenta[b]piperidines

(2012) Qing-Zhu Li et al.   ChemCatChem

Synthesis of some new indolo[2,3-c]isoquinolinyl pyrazoles, -1,3,4-oxadiazoles and their biological activities

(2012) Anand R. Saundane et al.   MEDICINAL CHEMISTRY RESEARCH

(S)-Proline-catalyzed nitro-Michael reactions: towards a better understanding of the catalytic mechanism and enantioselectivity

(2012) Hui Yang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Enantioselective Total Syntheses of Communesins A and B

(2011) Zhiwei Zuo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Quantum Mechanical Investigations of Organocatalysis: Mechanisms, Reactivities, and Selectivities

(2011) Paul Ha-Yeon Cheong et al.   CHEMICAL REVIEWS

NCIPLOT: A Program for Plotting Noncovalent Interaction Regions

(2011) Julia Contreras-García et al.   Journal of Chemical Theory and Computation

Direct annulation and alkylation of indoles with 2-aminobenzyl alcohols catalyzed by TFA

(2011) Forest J. Robertson et al.   TETRAHEDRON

Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety

(2010) Anna J. Kochanowska-Karamyan et al.   CHEMICAL REVIEWS

Alkaloids from a deep ocean sediment-derived fungus Penicillium sp. and their antitumor activities

(2010) Lin Du et al.   JOURNAL OF ANTIBIOTICS

Scalable Total Syntheses ofN-Linked Tryptamine Dimers by Direct Indole−Aniline Coupling: Psychotrimine and Kapakahines B and F

(2010) Timothy Newhouse et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Synthesis of (+)-Perophoramidine and Determination of the Absolute Configuration

(2010) Haoxing Wu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Revealing Noncovalent Interactions

(2010) Erin R. Johnson et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Simple indole alkaloids and those with a nonrearranged monoterpenoid unit

(2010) Minoru Ishikura et al.   NATURAL PRODUCT REPORTS

Total Synthesis of Kapakahine E and F

(2010) Vinson R. Espejo et al.   ORGANIC LETTERS

Organocatalytic Regio- and Stereoselective Inverse-Electron-Demand Aza-Diels-Alder Reaction of α,β-Unsaturated Aldehydes andN-Tosyl-1-aza-1,3-butadienes

(2009) Bo Han et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Light in Aminocatalysis: The Asymmetric Intermolecular α-Alkylation of Aldehydes

(2009) Paolo Melchiorre   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Amide-based bifunctional organocatalysts in asymmetric reactions

(2009) Xiaohua Liu et al.   CHEMICAL COMMUNICATIONS

Organocatalysis—after the gold rush

(2009) Søren Bertelsen et al.   CHEMICAL SOCIETY REVIEWS

Asymmetric Aminocatalysis-Gold Rush in Organic Chemistry

(2008) Paolo Melchiorre et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalytic Asymmetric Inverse-Electron-Demand Aza-Diels-Alder Reaction ofN-Sulfonyl-1-aza-1,3-butadienes and Aldehydes

(2008) Bo Han et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The Role of Noninnocent Solvent Molecules in Organocatalyzed Asymmetric Michael Addition Reactions

(2008) Mahendra P. Patil et al.   CHEMISTRY-A EUROPEAN JOURNAL

The advent and development of organocatalysis

(2008) David W. C. MacMillan   NATURE

Total Synthesis of Chaetominine

(2008) Mathieu Toumi et al.   ORGANIC LETTERS