Visible-Light 2,4-Dinitrophenol-Mediated Photoannulation of α-Azidochalcones into 2,5-Diaryloxazoles

Pd/Cu-Catalyzed C–H/C–H Cross Coupling of (Hetero)Arenes with Azoles through Arylsulfonium Intermediates

(2021) Ze-Yu Tian et al.   ORGANIC LETTERS

Recent Updates on Azido‐reductive Cyclization Approaches: Syntheses of aza ‐Heterocyclic Frameworks

(2021) Jay Prakash Soni et al.   Asian Journal of Organic Chemistry

Photoinduced Heterogeneous C−H Arylation by a Reusable Hybrid Copper Catalyst

(2020) Isaac Choi et al.   CHEMISTRY-A EUROPEAN JOURNAL

Photocatalyst‐Free Visible‐Light Enabled Synthesis of Substituted Pyrroles from α ‐Keto Vinyl Azides

(2020) Satheesh Borra et al.   ADVANCED SYNTHESIS & CATALYSIS

Visible-Light Photocatalysis as an Enabling Technology for Drug Discovery: A Paradigm Shift for Chemical Reactivity

(2020) Peijun Li et al.   ACS Medicinal Chemistry Letters

Organic Azides: Versatile Synthons in Transition Metal‐Catalyzed C( sp 2 )−H Amination/Annulation for N‐Heterocycle Synthesis

(2020) Zi‐Kui Liu et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis, anti-inflammatory and analgesic evaluation of thiazole/oxazole substituted benzothiazole derivatives

(2020) Gajendra Kumar et al.   BIOORGANIC CHEMISTRY

CO2/Photoredox Cocatalyzed Tandem Oxidative Cyclization of α-Bromo Ketones and Amines to Construct Substituted Oxazoles

(2019) Xiaowei Zhang et al.   JOURNAL OF ORGANIC CHEMISTRY

Divergent Conversion of N-Acyl-isoxazol-5(2H)-ones to Oxazoles and 1,3-Oxazin-6-ones Using Photoredox Catalysis

(2019) Mingjing Mei et al.   ORGANIC LETTERS

Reaction conditions for the regiodivergent direct arylations at C2‐ or C5‐positions of oxazoles using phosphine‐free palladium catalysts

(2019) Xinzhe Shi et al.   ADVANCED SYNTHESIS & CATALYSIS

Visible-Light Photocatalysis: Does It Make a Difference in Organic Synthesis?

(2018) Leyre Marzo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of 2,5-disubstituted oxazoles via cobalt(iii)-catalyzed cross-coupling of N-pivaloyloxyamides and alkynes

(2018) Xiaolong Yu et al.   CHEMICAL COMMUNICATIONS

Recent advance in oxazole-based medicinal chemistry

(2018) Hui-Zhen Zhang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Metal-free iodine(iii)-promoted synthesis of 2,5-diaryloxazoles

(2018) Xueying Yang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Access to 2,3-Fused Pyrroles via Visible Light Driven Coupling of α-Azidochalcones with 1/2-Naphthols, or 2-Hydroxy-1,4-Naphthoquinone

(2018) Satheesh Borra et al.   JOURNAL OF ORGANIC CHEMISTRY

Design, Synthesis and Biological Evaluation of 2 (((5-aryl-1,2,4-oxadiazol-3-yl)methyl)thio)benzo[d]oxazoles: New Antiinflammatory and Antioxidant Agents

(2018) Satyanarayana Yatam et al.   ChemistrySelect

Structure–Activity Relationships of New Natural Product-Based Diaryloxazoles with Selective Activity against Androgen Receptor-Positive Breast Cancer Cells

(2017) Andrew J. Robles et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Heterogeneous Gold(I)-Catalyzed [2 + 2 + 1] Annulation of Terminal Alkynes, Nitriles, and Oxygen Atoms Leading to 2,5-Disubstituted Oxazoles

(2017) Weisen Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Application of Vinyl Azides in Chemical Synthesis: A Recent Update

(2017) Hirohito Hayashi et al.   JOURNAL OF ORGANIC CHEMISTRY

Access to 1a,6b-Dihydro-1H-benzofuro[2,3-b]azirines and Benzofuran-2-amines via Visible Light Triggered Decomposition of α-Azidochalcones

(2017) Satheesh Borra et al.   ORGANIC LETTERS

Synthesis of Substituted Oxazoles by Visible-Light Photocatalysis

(2016) Tanmay Chatterjee et al.   JOURNAL OF ORGANIC CHEMISTRY

Visible Light Driven Photocascade Catalysis: Ru(bpy)3(PF6)2/TBHP-Mediated Synthesis of Fused β-Carbolines in Batch and Flow Microreactors

(2016) D. Chandrasekhar et al.   ORGANIC LETTERS

Visible Light Photocatalysis: Applications and New Disconnections in the Synthesis of Pharmaceutical Agents

(2016) James J. Douglas et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

A facile synthesis of 2,5-disubstituted oxazoles via a copper-catalyzed cascade reaction of alkenes with azides

(2015) Jiu-ling Li et al.   CHEMICAL COMMUNICATIONS

The rapid synthesis of oxazolines and their heterogeneous oxidation to oxazoles under flow conditions

(2015) Steffen Glöckner et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Reactivities of vinyl azides and their recent applications in nitrogen heterocycle synthesis

(2015) Bao Hu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

N-Bromosuccinimide as a Brominating Agent for the Transformation of N-H (or N-Benzyl) Ketoaziridines into Oxazoles

(2015) Heshmat Samimi et al.   SYNTHESIS-STUTTGART

Iodine catalysed intramolecular C(sp3)–H functionalization: synthesis of 2,5-disubstituted oxazoles from N-arylethylamides

(2015) Supravat Samanta et al.   RSC Advances

One-Pot Conversion of Amino Acids into 2,5-Disubstituted Oxazoles: No Metals Needed

(2014) Ivan Romero-Estudillo et al.   ADVANCED SYNTHESIS & CATALYSIS

Reaction of Alkynes and Azides: Not Triazoles Through Copper-Acetylides but Oxazoles Through Copper-Nitrene Intermediates

(2014) Estela Haldón et al.   CHEMISTRY-A EUROPEAN JOURNAL

Direct C–H Bond Arylation of (Benzo)oxazoles with Aryl Chlorides Catalyzed by N-Heterocyclic Carbene–Palladium(II)–1-Methylimidazole Complex

(2014) Xiao-Bao Shen et al.   ORGANIC LETTERS

Visible Light Photoredox Catalysis with Transition Metal Complexes: Applications in Organic Synthesis

(2013) Christopher K. Prier et al.   CHEMICAL REVIEWS

Practical oxazole synthesis mediated by iodine from α-bromoketones and benzylamine derivatives

(2013) Wen-Chao Gao et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Iodine(III)-Promoted Synthesis of Oxazoles through Oxidative Cyclization of N-Styrylbenzamides

(2013) Boris Nachtsheim et al.   SYNLETT

Practical Synthesis of Polysubstituted ImidazolesviaIodine- Catalyzed Aerobic Oxidative Cyclization of Aryl Ketones and Benzylamines

(2012) Huawen Huang et al.   ADVANCED SYNTHESIS & CATALYSIS

Pd(ii)-catalyzed direct C5-arylation of azole-4-carboxylates through double C–H bond cleavage

(2012) Ziyuan Li et al.   CHEMICAL COMMUNICATIONS

Room Temperature Copper(II)-Catalyzed Oxidative Cyclization of Enamides to 2,5-Disubstituted Oxazoles via Vinylic C–H Functionalization

(2012) Chi Wai Cheung et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper(ii)-mediated oxidative cyclization of enamides to oxazoles

(2012) Alison E. Wendlandt et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

A New Approach to Ring Expansion of Keto Aziridines to 2,5-Diaryloxazoles

(2012) Heshmat Samimi et al.   SYNLETT

Nickel-Catalyzed CH Arylation of Azoles with Haloarenes: Scope, Mechanism, and Applications to the Synthesis of Bioactive Molecules

(2011) Takuya Yamamoto et al.   CHEMISTRY-A EUROPEAN JOURNAL

Copper-Catalyzed Oxidative Arylation of Heteroarenes under Mild Conditions Using Dioxygen as the Sole Oxidant

(2011) Fanzhi Yang et al.   CHEMISTRY-A EUROPEAN JOURNAL

An Efficient [2 + 2 + 1] Synthesis of 2,5-Disubstituted Oxazoles via Gold-Catalyzed Intermolecular Alkyne Oxidation

(2011) Weimin He et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Nickel-Catalyzed Direct CH Arylation and Alkenylation of Heteroarenes with Organosilicon Reagents

(2010) Hitoshi Hachiya et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Palladium/Copper Bimetallic Catalytic System: Dramatic Improvement for Suzuki-Miyaura-Type Direct CH Arylation of Azoles with Arylboronic Acids

(2010) Bo Liu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Regioselective Formation of 2,5-Disubstituted Oxazoles Via Copper(I)-Catalyzed Cycloaddition of Acyl Azides and 1-Alkynes

(2010) Israel Cano et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Visible light photocatalysis as a greener approach to photochemical synthesis

(2010) Tehshik P. Yoon et al.   Nature Chemistry

TBHP/I2-Mediated Domino Oxidative Cyclization for One-Pot Synthesis of Polysubstituted Oxazoles

(2010) Huanfeng Jiang et al.   ORGANIC LETTERS

Direct arylations on water: synthesis of 2,5-disubstituted oxazoles balsoxin and texaline

(2008) Stephan A. Ohnmacht et al.   CHEMICAL COMMUNICATIONS

Ligandless Microwave-Assisted Pd/Cu-Catalyzed Direct Arylation of Oxazoles

(2008) François Besselièvre et al.   JOURNAL OF ORGANIC CHEMISTRY