Deciphering structure-activity relationships in a series of Tat/TAR inhibitors

The Design of RNA Binders: Targeting the HIV Replication Cycle as a Case Study

(2014) Aurélie Blond et al.   ChemMedChem

Entropy-Enthalpy Compensation: Role and Ramifications in Biomolecular Ligand Recognition and Design

(2013) John D. Chodera et al.   Annual Review of Biophysics

Effect of different arginine methylations on the thermodynamics of Tat peptide binding to HIV-1 TAR RNA

(2013) Santosh Kumar et al.   BIOCHIMIE

Blocking HIV-1 Replication by Targeting the Tat-Hijacked Transcriptional Machinery

(2013) Serena Massari et al.   CURRENT PHARMACEUTICAL DESIGN

Thermodynamic studies of a series of homologous HIV-1 TAR RNA ligands reveal that loose binders are stronger Tat competitors than tight ones

(2013) Lise Pascale et al.   NUCLEIC ACIDS RESEARCH

Methods to enable the design of bioactive small molecules targeting RNA

(2013) Matthew D. Disney et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Recent Advances in Developing Small Molecules Targeting RNA

(2011) Lirui Guan et al.   ACS Chemical Biology

Dynamic Ensemble View of the Conformational Landscape of HIV-1 TAR RNA and Allosteric Recognition

(2011) Jia Lu et al.   BIOCHEMISTRY

Polyamide Amino Acids trimers as TAR RNA ligands and anti-HIV agents

(2010) Vanessa Bonnard et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Thermodynamics of Peptide−RNA Recognition: The Binding of a Tat Peptide to TAR RNA

(2010) Hemant Suryawanshi et al.   JOURNAL OF PHYSICAL CHEMISTRY B

Essential structural requirements for specific recognition of HIV TAR RNA by peptide mimetics of Tat protein

(2010) Amy Davidson et al.   NUCLEIC ACIDS RESEARCH

How binding of small molecule and peptide ligands to HIV-1 TAR alters the RNA motional landscape

(2009) Michael F. Bardaro et al.   NUCLEIC ACIDS RESEARCH

Simultaneous recognition of HIV-1 TAR RNA bulge and loop sequences by cyclic peptide mimics of Tat protein

(2009) A. Davidson et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

RNA targeting through binding of small molecules: Studies on t-RNA binding by the cytotoxic protoberberine alkaloidcoralyne

(2008) Md. Maidul Islam et al.   Molecular BioSystems