Design, synthesis and docking studies of new hydrazinyl-thiazole derivatives as anticancer and antimicrobial agents

Eco-friendly sequential one-pot synthesis, molecular docking, and anticancer evaluation of arylidene-hydrazinyl-thiazole derivatives as CDK2 inhibitors

(2021) Abeer M. El-Naggar et al.   BIOORGANIC CHEMISTRY

Thiazole–Chalcone Hybrids as Prospective Antitubercular and Antiproliferative Agents: Design, Synthesis, Biological, Molecular Docking Studies and In Silico ADME Evaluation

(2021) Ashok Babu Kasetti et al.   MOLECULES

Experimental and computational study of hydrolysis and photolysis of antibiotic ceftriaxone: Degradation kinetics, pathways, and toxicity

(2021) Biljana F. Abramović et al.   SCIENCE OF THE TOTAL ENVIRONMENT

New functionalized 6‐thienylpyrimidine‐5‐carbonitriles as antiproliferative agents against human breast cancer cells

(2021) Omaima M. AboulWafa et al.   ARCHIV DER PHARMAZIE

Design, multistep synthesis and in-vitro antimicrobial and antioxidant screening of coumarin clubbed chalcone hybrids through molecular hybridization approach

(2021) Sathish Kumar Konidala et al.   Arabian Journal of Chemistry

2-Anilinopyrimidine derivatives: Design, synthesis, in vitro anti-proliferative activity, EGFR and ARO inhibitory activity, cell cycle analysis and molecular docking study

(2020) Omaima M. AboulWafa et al.   BIOORGANIC CHEMISTRY

Ceftobiprole Compared With Vancomycin Plus Aztreonam in the Treatment of Acute Bacterial Skin and Skin Structure Infections: Results of a Phase 3, Randomized, Double-blind Trial (TARGET)

(2020) J Scott Overcash et al.   CLINICAL INFECTIOUS DISEASES

Design, synthesis and molecular modeling studies of 2-styrylquinazoline derivatives as EGFR inhibitors and apoptosis inducers

(2020) Noha H. Amin et al.   BIOORGANIC CHEMISTRY

Synthesis and Biological Evaluation of Some Novel Thiazole-Based Heterocycles as Potential Anticancer and Antimicrobial Agents

(2019) Sraa Abu-Melha et al.   MOLECULES

Bacterial Proteinaceous Compounds With Multiple Activities Toward Cancers and Microbial Infection

(2019) Gisele Rodrigues et al.   Frontiers in Microbiology

Role of sulphur-heterocycles in medicinal chemistry: An update

(2019) Shelly Pathania et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Heterocycles in Medicinal Chemistry

(2019) Josef Jampilek   MOLECULES

Burden of Liver Diseases in the World

(2018) Sumeet K. Asrani et al.   JOURNAL OF HEPATOLOGY

Synthesis, characterization, antimicrobial activity and theoretical studies of new thiophene-based tripodal ligands

(2017) Tarik Harit et al.   JOURNAL OF MOLECULAR STRUCTURE

Peptides with Dual Antimicrobial and Anticancer Activities

(2017) Mário R. Felício et al.   Frontiers in Chemistry

Sulfur Containing Scaffolds in Drugs: Synthesis and Application in Medicinal Chemistry

(2016) Minghao Feng et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Synthesis, biological evaluation and 3D-QSAR study of novel 4,5-dihydro-1H-pyrazole thiazole derivatives as BRAFV600E inhibitors

(2015) Meng-Yue Zhao et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Isavuconazole: A New Broad-Spectrum Triazole Antifungal Agent

(2015) Marisa H. Miceli et al.   CLINICAL INFECTIOUS DISEASES

Synthesis of novel thiazole-based 8,9-dihydro-7H-pyrimido[4,5-b][1,4]diazepines as potential antitumor and antifungal agents

(2015) Juan Ramírez et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Antimicrobial peptide FF/CAP18 induces apoptotic cell death in HCT116 colon cancer cells via changes in the metabolic profile

(2015) KENGO KURODA et al.   INTERNATIONAL JOURNAL OF ONCOLOGY

AROS Is a Significant Biomarker for Tumor Aggressiveness in Non-cirrhotic Hepatocellular Carcinoma

(2015) Jung-Hee Kwon et al.   JOURNAL OF KOREAN MEDICAL SCIENCE

Synthesis and biological evaluation of novel series of thieno[2,3-d]pyrimidine derivatives as anticancer and antimicrobial agents

(2012) Nargues S. Habib et al.   MEDICINAL CHEMISTRY RESEARCH

Overview of the Chemistry of 2-Thiazolines

(2009) Annie-Claude Gaumont et al.   CHEMICAL REVIEWS

Characterization of Dasatinib and Its Structural Analogs as CYP3A4 Mechanism-Based Inactivators and the Proposed Bioactivation Pathways

(2009) X. Li et al.   DRUG METABOLISM AND DISPOSITION

Synthesis and anticancer activity of N-bis(trifluoromethyl)alkyl-N′-thiazolyl and N-bis(trifluoromethyl)alkyl-N′-benzothiazolyl ureas

(2009) Elena L. Luzina et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and antibacterial activity of isothiazolyl oxazolidinones and analogous 3(2H)-isothiazolones

(2009) Neda Adibpour et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Modes of Action of the New Arylguanidine Abafungin beyond Interference with Ergosterol Biosynthesis and in vitro Activity against Medically Important Fungi

(2008) C. Borelli et al.   CHEMOTHERAPY