Comparison of three novel radiotracers for GluN2B-containing NMDA receptors in non-human primates: (R)-[11C]NR2B-Me, (R)-[18F]of-Me-NB1, and (S)-[18F]of-NB1
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Title
Comparison of three novel radiotracers for GluN2B-containing NMDA receptors in non-human primates: (R)-[11C]NR2B-Me, (R)-[18F]of-Me-NB1, and (S)-[18F]of-NB1
Authors
Keywords
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Journal
JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM
Volume -, Issue -, Pages 0271678X2210844
Publisher
SAGE Publications
Online
2022-02-25
DOI
10.1177/0271678x221084416
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- An anatomically comprehensive atlas of the adult human brain transcriptome
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