Manufacturing Process Development for Belzutifan, Part 6: Ensuring Scalability for a Deoxyfluorination Reaction

Manufacturing Process Development for Belzutifan, Part 5: A Streamlined Fluorination–Dynamic Kinetic Resolution Process

(2021) Tao Wang et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Manufacturing Process Development for Belzutifan, Part 3: Completing a Streamlined Through-Process with a Safe and Scalable Oxidation

(2021) Zhiwei Chen et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Manufacturing Process Development for Belzutifan, Part 4: Nitrogen Flow Criticality for Transfer Hydrogenation Control

(2021) Nastaran Salehi Marzijarani et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Manufacturing Process Development for Belzutifan, Part 2: A Continuous Flow Visible-Light-Induced Benzylic Bromination

(2021) Cecilia Bottecchia et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Manufacturing Process Development for Belzutifan, Part 1: A Concise Synthesis of the Indanone Starting Material

(2021) Feng Peng et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Deoxyfluorination using CuF2 enabled by a Lewis base activating group strategy

(2020) Deepali Eilidh Sood et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rapid Deoxyfluorination of Alcohols with N ‐Tosyl‐4‐chlorobenzenesulfonimidoyl Fluoride (SulfoxFluor) at Room Temperature

(2019) Junkai Guo et al.   CHEMISTRY-A EUROPEAN JOURNAL

3-[(1S,2S,3R)-2,3-Difluoro-1-hydroxy-7-methylsulfonylindan-4-yl]oxy-5-fluorobenzonitrile (PT2977), a Hypoxia-Inducible Factor 2α (HIF-2α) Inhibitor for the Treatment of Clear Cell Renal Cell Carcinoma

(2019) Rui Xu et al.   JOURNAL OF MEDICINAL CHEMISTRY

XtalFluor-E: A useful and versatile reagent in organic transformations

(2019) Leyla Mohammadkhani et al.   JOURNAL OF FLUORINE CHEMISTRY

Deoxyfluorination with Sulfonyl Fluorides: Navigating Reaction Space with Machine Learning

(2018) Matthew K. Nielsen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Recent Developments in the Deoxyfluorination of Alcohols and Phenols: New Reagents, Mechanistic Insights, and Applications

(2017) Xiang-Guo Hu et al.   SYNTHESIS-STUTTGART

AlkylFluor: Deoxyfluorination of Alcohols

(2016) Nathaniel W. Goldberg et al.   ORGANIC LETTERS

PyFluor: A Low-Cost, Stable, and Selective Deoxyfluorination Reagent

(2015) Matthew K. Nielsen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Good Partnership between Sulfur and Fluorine: Sulfur-Based Fluorination and Fluoroalkylation Reagents for Organic Synthesis

(2014) Chuanfa Ni et al.   CHEMICAL REVIEWS

Deoxofluorination Reactions Using N,N-Disubstituted Aminodifluorosulfinium Tetrafluoroborate Salts

(2013) Olivier Mahé et al.   JOURNAL OF FLUORINE CHEMISTRY

Late-Stage Deoxyfluorination of Alcohols with PhenoFluor

(2013) Filippo Sladojevich et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Discovery of 4-tert-Butyl-2,6-dimethylphenylsulfur Trifluoride as a Deoxofluorinating Agent with High Thermal Stability as Well as Unusual Resistance to Aqueous Hydrolysis, and Its Diverse Fluorination Capabilities Including Deoxofluoro-Arylsulfinylation with High Stereoselectivity

(2010) Teruo Umemoto et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Highly Efficient Conversion of Primary or Secondary Alcohols into Fluorides with n-Perfluorobutanesulfonyl Fluoride-Tetrabutylammonium Triphenyldifluorosilicate

(2009) Xueqing Zhao et al.   SYNLETT