Design, synthesis, biological evaluations and in silico studies of sulfonate ester derivatives of 2-(2-benzylidenehydrazono)thiazolidin-4-one as potential α-glucosidase inhibitors

Synthesis and studies of thiazolidinedione–isatin hybrids as α-glucosidase inhibitors for management of diabetes

(2021) Ramandeep Kaur et al.   Future Medicinal Chemistry

Exploring efficacy of indole-based dual inhibitors for α-glucosidase and α-amylase enzymes: In silico, biochemical and kinetic studies

(2020) Abdel-Nasser Kawde et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

Synthesis, α-glucosidase inhibition, and molecular docking studies of novel N-substituted hydrazide derivatives of atranorin as antidiabetic agents

(2020) Thuc-Huy Duong et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, in vitro alpha-glucosidase inhibitory potential of benzimidazole bearing bis-Schiff bases and their molecular docking study

(2019) Fazal Rahim et al.   BIOORGANIC CHEMISTRY

Synthesis of new arylhydrazide bearing Schiff bases/thiazolidinone: α-Amylase, urease activities and their molecular docking studies

(2019) Fazal Rahim et al.   BIOORGANIC CHEMISTRY

Design, synthesis, in vitro, and in silico studies of novel diarylimidazole-1,2,3-triazole hybrids as potent α-glucosidase inhibitors

(2019) Mina Saeedi et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and molecular docking studies of imines as α-glucosidase and α-amylase inhibitors

(2019) Analy Aispuro-Pérez et al.   BIOORGANIC CHEMISTRY

Hybrids of Isatin‐Pyrazole as Potential α‐Glucosidase Inhibitors: Synthesis, Biological Evaluations and Molecular Docking Studies

(2019) Ramandeep Kaur et al.   ChemistrySelect

Synthesis, α- glucosidase inhibition and molecular docking study of coumarin based derivatives

(2018) Muhammad Taha et al.   BIOORGANIC CHEMISTRY

Synthesis of Bis -indolylmethane sulfonohydrazides derivatives as potent α -Glucosidase inhibitors

(2018) Mohammed Gollapalli et al.   BIOORGANIC CHEMISTRY

Diabesity and antidiabetic drugs

(2018) Joseph M. Pappachan et al.   MOLECULAR ASPECTS OF MEDICINE

Xanthenone-based hydrazones as potent α-glucosidase inhibitors: Synthesis, solid state self-assembly and in silico studies

(2018) Qamar-un-Nisa Tariq et al.   BIOORGANIC CHEMISTRY

Novel hybrids of benzothiazole-1,3,4-oxadiazole-4-thiazolidinone: Synthesis, in silico ADME study, molecular docking and in vivo anti-diabetic assessment

(2018) Rubina Bhutani et al.   BIOORGANIC CHEMISTRY

Hydrazinyl arylthiazole based pyridine scaffolds: Synthesis, structural characterization, in vitro α -glucosidase inhibitory activity, and in silico studies

(2017) Farman Ali et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Molecular docking studies and synthesis of novel bisbenzimidazole derivatives as inhibitors of α-glucosidase

(2016) Musa Özil et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Heterocyclic Compounds: Effective α-Amylase and α-Glucosidase Inhibitors

(2016) Mina Saeedi et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Influence of gallic acid on α-amylase and α-glucosidase inhibitory properties of acarbose

(2016) Ganiyu Oboh et al.   JOURNAL OF FOOD AND DRUG ANALYSIS

Synthesis of new oxadiazole derivatives as α-glucosidase inhibitors

(2015) Muhammad Taha et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Pyridine sulfonamide as a small key organic molecule for the potential treatment of type-II diabetes mellitus and Alzheimer’s disease: In vitro studies against yeast α-glucosidase, acetylcholinesterase and butyrylcholinesterase

(2015) Sadaf Riaz et al.   BIOORGANIC CHEMISTRY

Synthesis of 4-thiazolidinone analogs as potent in vitro anti-urease agents

(2015) Fazal Rahim et al.   BIOORGANIC CHEMISTRY

Synthesis of novel flavone hydrazones: In-vitro evaluation of α-glucosidase inhibition, QSAR analysis and docking studies

(2015) Syahrul Imran et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Copper catalyzed synthesis of unsymmetrical diaryl sulfones from an arenediazonium salt and sodium p-toluenesulfinate

(2015) Sitaram Haribhau Gund et al.   RSC Advances

A new series of N2-substituted-5-(p-toluenesulfonylamino)phthalimide analogues as α-glucosidase inhibitors

(2013) Xiaoli Bian et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Template-based protein structure modeling using the RaptorX web server

(2012) Morten Källberg et al.   Nature Protocols

Design, Synthesis, and Evaluation of Thiazolidinone Derivatives as Antimicrobial and Anti-viral Agents

(2011) Veerasamy Ravichandran et al.   Chemical Biology & Drug Design

IDF Diabetes Atlas: Global estimates of the prevalence of diabetes for 2011 and 2030

(2011) David R. Whiting et al.   DIABETES RESEARCH AND CLINICAL PRACTICE

Molecular Dynamics Simulation and Free Energy Calculation Studies of the Binding Mechanism of Allosteric Inhibitors with p38α MAP Kinase

(2011) Ying Yang et al.   Journal of Chemical Information and Modeling

Diagnosis and Classification of Diabetes Mellitus

(2009)   DIABETES CARE

Antioxidant Anti-Inflammatory Treatment in Type 2 Diabetes

(2009) A. Ceriello et al.   DIABETES CARE

Synthesis and evaluation of the α-glucosidase inhibitory activity of 3-[4-(phenylsulfonamido)benzoyl]-2H-1-benzopyran-2-one derivatives

(2009) Shaojie Wang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

4-Thiazolidinone – A biologically active scaffold

(2007) Amit Verma et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

QMEAN: A comprehensive scoring function for model quality assessment

(2007) Pascal Benkert et al.   PROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS