Design, synthesis, molecular modeling, and biological evaluation of novel kojic acid derivatives containing bioactive heterocycle moiety as inhibitors of tyrosinase and antibrowning agents

The natural-based optimization of kojic acid conjugated to different thio-quinazolinones as potential anti-melanogenesis agents with tyrosinase inhibitory activity

(2021) Nima Sepehri et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, antioxidant and anti-tyrosinase activity of 1,2,4-triazole hydrazones as antibrowning agents

(2020) Zhiyun Peng et al.   FOOD CHEMISTRY

A comprehensive review on tyrosinase inhibitors

(2019) Samaneh Zolghadri et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Antityrosinase and antioxidant activities of guanidine compounds and effect of guanylthiourea on melanogenesis

(2019) Yu-Xia Wang et al.   PROCESS BIOCHEMISTRY

Antibrowning Compounds for Minimally Processed Potatoes: A Review

(2019) Gloria Bobo-García et al.   FOOD REVIEWS INTERNATIONAL

Benzo[b]thiophene-thiazoles as potent anti-Toxoplasma gondii agents: Design, synthesis, tyrosinase/tyrosine hydroxylase inhibitors, molecular docking study, and antioxidant activity

(2019) Beata Rosada et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Hydroxyphenyl thiosemicarbazones as inhibitors of mushroom tyrosinase and antibrowning agents

(2019) M. Carcelli et al.   FOOD CHEMISTRY

Advances in the tyrosinase inhibitors from plant source

(2018) Marco Bonesi et al.   CURRENT MEDICINAL CHEMISTRY

Novel hydroxypyridinone derivatives containing an oxime ether moiety: Synthesis, inhibition on mushroom tyrosinase and application in anti-browning of fresh-cut apples

(2018) Le-Le Shao et al.   FOOD CHEMISTRY

Swertiajaponin as an anti-browning and antioxidant flavonoid

(2018) Kyoung Mi Moon et al.   FOOD CHEMISTRY

Interactions of hemin with bovine serum albumin and human hemoglobin: A fluorescence quenching study

(2018) Magdalena Makarska-Bialokoz   SPECTROCHIMICA ACTA PART A-MOLECULAR AND BIOMOLECULAR SPECTROSCOPY

Recent advances in controlling polyphenol oxidase activity of fruit and vegetable products

(2018) Federica Tinello et al.   Innovative Food Science & Emerging Technologies

1,2,3-Triazole-based kojic acid analogs as potent tyrosinase inhibitors: Design, synthesis and biological evaluation

(2018) Morteza Ashooriha et al.   BIOORGANIC CHEMISTRY

Synthesis of N-Aryl-2-aminobenzoxazoles from Substituted Benzoxazole-2-thiol and 2-Chloro-N-arylacetamides in KOH-DMF System

(2017) Guang-cheng Wang et al.   HETEROCYCLES

Rifampicin as a novel tyrosinase inhibitor: Inhibitory activity and mechanism

(2017) Wei-Ming Chai et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

An insight of binding interaction between Tryptophan, Tyrosine and Phenylalanine separately with green gold nanoparticles by fluorescence quenching method

(2017) Swarup Roy   OPTIK

Pre-storage kojic acid application delays pericarp browning and maintains antioxidant activities of litchi fruit

(2017) Hafiz Muhammad Shoaib Shah et al.   POSTHARVEST BIOLOGY AND TECHNOLOGY

Synthesis, biological evaluation and molecular docking study of N -arylbenzo[ d ]oxazol-2-amines as potential α-glucosidase inhibitors

(2016) Guangcheng Wang et al.   BIOORGANIC & MEDICINAL CHEMISTRY

4-Hydroxy cinnamic acid as mushroom preservation: Anti-tyrosinase activity kinetics and application

(2016) Yong-Hua Hu et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

Synthesis and Biological Evaluation of Kojic Acid Derivatives Containing 1,2,4-triazole as Potent Tyrosinase Inhibitors

(2015) Wenlin Xie et al.   Chemical Biology & Drug Design

Effects of Curing Treatment on the Browning of Fresh-cut Potatoes

(2014) Zhiqiang Hou et al.   AMERICAN JOURNAL OF POTATO RESEARCH

Synthesis, structure–activity relationship analysis and kinetics study of reductive derivatives of flavonoids as Helicobacter pylori urease inhibitors

(2013) Zhu-Ping Xiao et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis, characterization and biological evaluation of paeonol thiosemicarbazone analogues as mushroom tyrosinase inhibitors

(2013) Tian-Hua Zhu et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

Optimization of O3-Acyl Kojic Acid Derivatives as Potent and Selective Human Neutrophil Elastase Inhibitors

(2013) Susana D. Lucas et al.   JOURNAL OF MEDICINAL CHEMISTRY

Discovery of 4-oxo-6-((pyrimidin-2-ylthio)methyl)-4H-pyran-3-yl 4-nitrobenzoate (ML221) as a functional antagonist of the apelin (APJ) receptor

(2012) Patrick R. Maloney et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Heterocycles in drugs and drug discovery

(2012) A. Gomtsyan   Chemistry of Heterocyclic Compounds

Natural and Synthetic Tyrosinase Inhibitors as Antibrowning Agents: An Update

(2012) M. R. Loizzo et al.   COMPREHENSIVE REVIEWS IN FOOD SCIENCE AND FOOD SAFETY

Stability, solubility, mechanical and barrier properties of cassava starch – Carnauba wax edible coatings to preserve fresh-cut apples

(2011) Marcela Chiumarelli et al.   FOOD HYDROCOLLOIDS

Synthesis and Biological Evaluation of Kojyl Thioether Derivatives as Tyrosinase Inhibitors

(2010) Ho-Sik Rho et al.   BULLETIN OF THE KOREAN CHEMICAL SOCIETY

Tryptophan Fluorescence Quenching by Enzyme Inhibitors As a Tool for Enzyme Active Site Structure Investigation: Epoxide Hydrolase

(2009) Evgenia Matveeva et al.   CURRENT PHARMACEUTICAL BIOTECHNOLOGY