Does the circulating ketoconazole metabolite N-deacetyl ketoconazole contribute to the drug-drug interaction potential of the parent compound?

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Characterization of chemical-induced sterile inflammation in vitro: application of the model compound ketoconazole in a human hepatic co-culture system

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Human arylacetamide deacetylase hydrolyzes ketoconazole to trigger hepatocellular toxicity

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No Increased Risk of Ketoconazole Toxicity in Drug-Drug Interaction Studies

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The Treatment of Cushing's Disease

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Influence of sildenafil and tadalafil on the enzyme- and transporter-inducing effects of bosentan and ambrisentan in LS180 cells

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