Design, synthesis and biological evaluation of pleuromutilin-Schiff base hybrids as potent anti-MRSA agents in vitro and in vivo
Published 2021 View Full Article
- Home
- Publications
- Publication Search
- Publication Details
Title
Design, synthesis and biological evaluation of pleuromutilin-Schiff base hybrids as potent anti-MRSA agents in vitro and in vivo
Authors
Keywords
Antibacterial activity, MRSA, Pleuromutilin, 1,2,4-Triazole, Schiff base
Journal
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Volume 223, Issue -, Pages 113624
Publisher
Elsevier BV
Online
2021-06-12
DOI
10.1016/j.ejmech.2021.113624
References
Ask authors/readers for more resources
Related references
Note: Only part of the references are listed.- Antibacterial Activity and Pharmacokinetic Profile of a Promising Antibacterial Agent: 22-(2-Amino-phenylsulfanyl)-22-Deoxypleuromutilin
- (2020) Xiangyi Zuo et al. MOLECULES
- Efficiency comparison of apigenin-7-O-glucoside and trolox in antioxidative stress and anti-inflammatory properties
- (2020) Wei Wang et al. JOURNAL OF PHARMACY AND PHARMACOLOGY
- Design, synthesis and biological evaluation of novel pleuromutilin derivatives containing piperazine and 1,2,3-triazole linker
- (2020) Guang-Yu Zhang et al. BIOORGANIC CHEMISTRY
- Leave it to Lefamulin: A Pleuromutilin Treatment Option in Community-Acquired Bacterial Pneumonia
- (2019) Young Ran Lee et al. DRUGS
- Design, synthesis and biological evaluation of novel pleuromutilin derivatives possessing acetamine phenyl linker
- (2019) Zhen Jin et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis and antibacterial activities of novel pleuromutilin derivatives bearing an aminothiophenol moiety
- (2018) Zhao-Sheng Zhang et al. Chemical Biology & Drug Design
- Design, synthesis and antibacterial evaluation of novel pleuromutilin derivatives possessing piperazine linker
- (2017) Mei-Ling Gao et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Novel Aldimine-Type Schiff Bases of 4-Amino-5-[(3,4,5-trimethoxyphenyl)methyl]-1,2,4-triazole-3-thione/thiol: Docking Study, Synthesis, Biological Evaluation, and Anti-Tubulin Activity
- (2016) Alieh Ameri et al. ARCHIV DER PHARMAZIE
- Design, synthesis, and structure-activity relationship studies of novel pleuromutilin derivatives having a piperazine ring
- (2016) Jian Luo et al. Chemical Biology & Drug Design
- Novel 3-Aminothiazolquinolones: Design, Synthesis, Bioactive Evaluation, SARs, and Preliminary Antibacterial Mechanism
- (2016) Sheng-Feng Cui et al. JOURNAL OF MEDICINAL CHEMISTRY
- New thiophene-1,2,4-triazole-5(3)-ones: Highly bioactive thiosemicarbazides, structures of Schiff bases and triazole–thiols
- (2014) Yasemin Ünver et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis and Biological Activities of Novel Pleuromutilin Derivatives with a Substituted Thiadiazole Moiety as Potent Drug-Resistant Bacteria Inhibitors
- (2014) Ruofeng Shang et al. JOURNAL OF MEDICINAL CHEMISTRY
- Risk factors for anti-MRSA drug resistance
- (2012) Yasuhisa Abe et al. INTERNATIONAL JOURNAL OF ANTIMICROBIAL AGENTS
- Meticillin-resistant Staphylococcus aureus (MRSA): global epidemiology and harmonisation of typing methods
- (2012) Stefania Stefani et al. INTERNATIONAL JOURNAL OF ANTIMICROBIAL AGENTS
- In vitro biofilm formation and bactericidal activities of methicillin-resistant Staphylococcus aureus clones prevalent in Korea
- (2011) Jeong-Ok Cha et al. DIAGNOSTIC MICROBIOLOGY AND INFECTIOUS DISEASE
- Pleuromutilin and its Derivatives-The Lead Compounds for Novel Antibiotics
- (2011) Y. -Z. Tang et al. MINI-REVIEWS IN MEDICINAL CHEMISTRY
- A Field Guide to Pandemic, Epidemic and Sporadic Clones of Methicillin-Resistant Staphylococcus aureus
- (2011) Stefan Monecke et al. PLoS One
- Synthesis and evaluation of some new benzothiazole derivatives as potential antimicrobial agents
- (2010) Balram Soni et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Pleuromutilin derivatives having a purine ring. Part 3: Synthesis and antibacterial activity of novel compounds possessing a piperazine ring spacer
- (2008) Yoshimi Hirokawa et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Methicillin-resistant Staphylococcus aureus and animals: zoonosis or humanosis?
- (2008) M. Morgan JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY
Discover Peeref hubs
Discuss science. Find collaborators. Network.
Join a conversationPublish scientific posters with Peeref
Peeref publishes scientific posters from all research disciplines. Our Diamond Open Access policy means free access to content and no publication fees for authors.
Learn More