Strain-Promoted Azide–Alkyne Cycloaddition-Based PSMA-Targeting Ligands for Multimodal Intraoperative Tumor Detection of Prostate Cancer

Global cancer statistics 2020: GLOBOCAN estimates of incidence and mortality worldwide for 36 cancers in 185 countries

(2021) Hyuna Sung et al.   CA-A CANCER JOURNAL FOR CLINICIANS

Synthesis, Preclinical Evaluation, and First-in-Human PET Study of Quinoline-Containing PSMA Tracers with Decreased Renal Excretion

(2021) Xiaojun Zhang et al.   JOURNAL OF MEDICINAL CHEMISTRY

An Overview of Recent Advances in Biomedical Applications of Click Chemistry

(2021) Jasleen Kaur et al.   BIOCONJUGATE CHEMISTRY

The importance of linkers in the structure of PSMA ligands

(2021) Anastasia A. Uspenskaya et al.   CURRENT MEDICINAL CHEMISTRY

Modular medical imaging agents based on azide‐alkyne Huisgen cycloadditions: Synthesis and pre‐clinical evaluation of 18F‐labeled PSMA‐tracers for prostate cancer imaging.

(2020) Verena I. Böhmer et al.   CHEMISTRY-A EUROPEAN JOURNAL

Novel 177Lu-labeled Albumin-binder-conjugated PSMA-targeting Agents with Extremely High Tumor Uptake and Enhanced Tumor-to-kidney Absorbed Dose Ratio

(2020) Hsiou-Ting Kuo et al.   JOURNAL OF NUCLEAR MEDICINE

Click Chemistry as a Tool for Cell Engineering and Drug Delivery

(2019) Yukiya Takayama et al.   MOLECULES

Chelators and metal complex stability for radiopharmaceutical applications

(2019) Nkemakonam C. Okoye et al.   RADIOCHIMICA ACTA

Click Chemistry in the Design and Production of Hybrid Tracers

(2019) Albertus W. Hensbergen et al.   ACS Omega

Hybrid Tracers Based on Cyanine Backbones Targeting Prostate-Specific Membrane Antigen – Tuning Pharmacokinetic Properties and Exploring Dye–Protein Interaction

(2019) Albertus Wijnand Hensbergen et al.   JOURNAL OF NUCLEAR MEDICINE

Recent Advances in Bioorthogonal Click Chemistry for Efficient Synthesis of Radiotracers and Radiopharmaceuticals

(2019) Mushtaq et al.   MOLECULES

Image-Guided Surgery: Are We Getting the Most Out of Small-Molecule Prostate-Specific-Membrane-Antigen-Targeted Tracers?

(2019) Albertus Wijnand Hensbergen et al.   BIOCONJUGATE CHEMISTRY

Targeting prostate cancer: Prostate-specific membrane antigen based diagnosis and therapy

(2018) Till Wüstemann et al.   MEDICINAL RESEARCH REVIEWS

Single Low-Dose Injection of Evans Blue Modified PSMA-617 Radioligand Therapy Eliminates Prostate-Specific Membrane Antigen Positive Tumors

(2018) Zhantong Wang et al.   BIOCONJUGATE CHEMISTRY

Synthesis and in vitro and in vivo evaluation of urea-based PSMA inhibitors with increased lipophilicity

(2018) Martina Wirtz et al.   EJNMMI Research

PSMA-11–Derived Dual-Labeled PSMA Inhibitors for Preoperative PET Imaging and Precise Fluorescence-Guided Surgery of Prostate Cancer

(2017) Ann-Christin Baranski et al.   JOURNAL OF NUCLEAR MEDICINE

Metal-Based PSMA Radioligands

(2017) Eleni Gourni et al.   MOLECULES

A Practical Guide on the Synthesis of Metal Chelates for Molecular Imaging and Therapy by Means of Click Chemistry

(2016) Johannes Notni et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis and pre-clinical evaluation of a new class of high-affinity 18F-labeled PSMA ligands for detection of prostate cancer by PET imaging

(2016) James Kelly et al.   EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING

Preclinical Evaluation of 18 F-PSMA-1007, a New Prostate-Specific Membrane Antigen Ligand for Prostate Cancer Imaging

(2016) Jens Cardinale et al.   JOURNAL OF NUCLEAR MEDICINE

„PSMA-radioguided surgery“ beim lokal begrenzten Prostatakarzinomrezidiv

(2016) I. Rauscher et al.   UROLOGE

„PSMA-radioguided surgery“ beim lokal begrenzten Prostatakarzinomrezidiv

(2016) I. Rauscher et al.   UROLOGE

Towards Personalized Treatment of Prostate Cancer: PSMA I&T, a Promising Prostate-Specific Membrane Antigen-Targeted Theranostic Agent

(2016) Kristell L.S. Chatalic et al.   Theranostics

Preclinical Evaluation of a Tailor-Made DOTA-Conjugated PSMA Inhibitor with Optimized Linker Moiety for Imaging and Endoradiotherapy of Prostate Cancer

(2015) M. Bene ova et al.   JOURNAL OF NUCLEAR MEDICINE

68Ga- and 177Lu-Labeled PSMA I&T: Optimization of a PSMA-Targeted Theranostic Concept and First Proof-of-Concept Human Studies

(2015) M. Weineisen et al.   JOURNAL OF NUCLEAR MEDICINE

[111In]PSMA-I&T: expanding the spectrum of PSMA-I&T applications towards SPECT and radioguided surgery

(2015) Margret Schottelius et al.   EJNMMI Research

(R)-NODAGA-PSMA: A Versatile Precursor for Radiometal Labeling and Nuclear Imaging of PSMA-Positive Tumors

(2015) Eleni Gourni et al.   PLoS One

Targeting human prostate cancer with111In-labeled D2B IgG, F(ab′)2and Fab fragments in nude mice with PSMA-expressing xenografts

(2014) Susanne Lütje et al.   Contrast Media & Molecular Imaging

Pretargeted imaging using bioorthogonal chemistry in mice

(2014) Raffaella Rossin et al.   CURRENT OPINION IN CHEMICAL BIOLOGY

Dual-Modality Image-Guided Surgery of Prostate Cancer with a Radiolabeled Fluorescent Anti-PSMA Monoclonal Antibody

(2014) S. Lutje et al.   JOURNAL OF NUCLEAR MEDICINE

Development of Targeted Near-Infrared Imaging Agents for Prostate Cancer

(2014) X. Wang et al.   MOLECULAR CANCER THERAPEUTICS

Targeted Radionuclide and Fluorescence Dual-modality Imaging of Cancer: Preclinical Advances and Clinical Translation

(2014) S. Lütje et al.   MOLECULAR IMAGING AND BIOLOGY

Improving the biodistribution of PSMA-targeting tracers with a highly negatively charged linker

(2014) Steve S. Huang et al.   PROSTATE

Positive Surgical Margins After Radical Prostatectomy: A Systematic Review and Contemporary Update

(2013) Ofer Yossepowitch et al.   EUROPEAN UROLOGY

Improved labelling of DTPA- and DOTA-conjugated peptides and antibodies with 111In in HEPES and MES buffer

(2012) Maarten Brom et al.   EJNMMI Research

Sequential SPECT and Optical Imaging of Experimental Models of Prostate Cancer with a Dual Modality Inhibitor of the Prostate-Specific Membrane Antigen

(2011) Sangeeta Ray Banerjee et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Growing Applications of “Click Chemistry” for Bioconjugation in Contemporary Biomedical Research

(2009) Kido Nwe et al.   CANCER BIOTHERAPY AND RADIOPHARMACEUTICALS

U-SPECT-II: An Ultra-High-Resolution Device for Molecular Small-Animal Imaging

(2009) F. van der Have et al.   JOURNAL OF NUCLEAR MEDICINE

Synthesis and Evaluation of Technetium-99m- and Rhenium-Labeled Inhibitors of the Prostate-Specific Membrane Antigen (PSMA)

(2008) Sangeeta R. Banerjee et al.   JOURNAL OF MEDICINAL CHEMISTRY

Interactions between Human Glutamate Carboxypeptidase II and Urea-Based Inhibitors: Structural Characterization†

(2008) Cyril Barinka et al.   JOURNAL OF MEDICINAL CHEMISTRY