Synthetic glycoconjugates inhibitors of tumor-related galectin-3: an update

Cu-Catalyzed Click Reaction in Carbohydrate Chemistry

(2016) Vinod K. Tiwari et al.   CHEMICAL REVIEWS

Glyco-nano-oncology: Novel therapeutic opportunities by combining small and sweet

(2016) Pablo F. Hockl et al.   PHARMACOLOGICAL RESEARCH

Protein Glycosylation in Cancer

(2015) Sean R. Stowell et al.   Annual Review of Pathology-Mechanisms of Disease

Synthetic 1,2,3-triazole-linked glycoconjugates bind with high affinity to human galectin-3

(2015) Marcelo Fiori Marchiori et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Thio- and selenoglycosides as ligands for biomedically relevant lectins: Valency–activity correlations for benzene-based dithiogalactoside clusters and first assessment for (di)selenodigalactosides

(2015) Sabine André et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

G3-C12 Peptide Reverses Galectin-3 from Foe to Friend for Active Targeting Cancer Treatment

(2015) Wei Sun et al.   MOLECULAR PHARMACEUTICS

Cancer intelligence acquired (CIA): tumor glycosylation and sialylation codes dismantling antitumor defense

(2014) Kayluz Frias Boligan et al.   CELLULAR AND MOLECULAR LIFE SCIENCES

Antibodies against Mucin-Based Glycopeptides AffectTrypanosoma cruziCell Invasion and Tumor Cell Viability

(2014) Vanessa L. Campo et al.   CHEMBIOCHEM

Defining the Potential of Aglycone Modifications for Affinity/Selectivity Enhancement against Medically Relevant Lectins: Synthesis, Activity Screening, and HSQC-Based NMR Analysis

(2014) Subhash R. Rauthu et al.   CHEMBIOCHEM

Lactose-Functionalized Dendrimers Arbitrate the Interaction of Galectin-3/MUC1 Mediated Cancer Cellular Aggregation

(2014) Anna K. Michel et al.   CHEMBIOCHEM

Galectins: Major Signaling Modulators Inside and Outside the Cell

(2014) D. Compagno et al.   CURRENT MOLECULAR MEDICINE

Galectin-3 inhibitors: a patent review (2008–present)

(2014) Helen Blanchard et al.   EXPERT OPINION ON THERAPEUTIC PATENTS

Influencing factors on the synthesis of magnetically responsive lipases

(2014) Jing Li et al.   JOURNAL OF MOLECULAR CATALYSIS B-ENZYMATIC

Design and synthesis of glycoprotein-based multivalent glyco-ligands for influenza hemagglutinin and human galectin-3

(2013) Helen Wang et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Investigation into the Feasibility of Thioditaloside as a Novel Scaffold for Galectin-3-Specific Inhibitors

(2013) Khuchtumur Bum-Erdene et al.   CHEMBIOCHEM

Human Galectin-3 Selective and High Affinity Inhibitors. Present State and Future Perspectives

(2013) R. Tellez-Sanz et al.   CURRENT MEDICINAL CHEMISTRY

Tuning the Preference of Thiodigalactoside- and Lactosamine-Based Ligands to Galectin-3 over Galectin-1

(2013) Hilde van Hattum et al.   JOURNAL OF MEDICINAL CHEMISTRY

Combinatorial One-Pot Synthesis of Poly-N-acetyllactosamine Oligosaccharides with Leloir-Glycosyltransferases

(2011) Claudia Rech et al.   ADVANCED SYNTHESIS & CATALYSIS

Inhibitory potential of chemical substitutions at bioinspired sites of β-d-galactopyranose on neoglycoprotein/cell surface binding of two classes of medically relevant lectins

(2011) Denis Giguère et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Taloside Inhibitors of Galectin-1 and Galectin-3

(2011) Patrick M. Collins et al.   Chemical Biology & Drug Design

Inhibition of Galectins with Small Molecules

(2011) Christopher T. Öberg et al.   CHIMIA

Glycosylation, galectins and cellular signaling

(2011) Cecile Boscher et al.   CURRENT OPINION IN CELL BIOLOGY

Mechanisms of cancer-associated glycosylation changes

(2011) Fabio Dall'Olio   Frontiers in Bioscience-Landmark

Structural Basis for Distinct Binding Properties of the Human Galectins to Thomsen-Friedenreich Antigen

(2011) Cheng-Feng Bian et al.   PLoS One

Glycoclusters presenting lactose on calix[4]arene cores display trypanocidal activity

(2011) Eva Galante et al.   TETRAHEDRON

Synthesis of 3-amido-3-deoxy-β-d-talopyranosides: all-cis-substituted pyranosides as lectin inhibitors

(2011) Christopher T. Öberg et al.   TETRAHEDRON

Monovalent Interactions of Galectin-1

(2010) Emma Salomonsson et al.   BIOCHEMISTRY

1H-1,2,3-Triazol-1-yl thiodigalactoside derivatives as high affinity galectin-3 inhibitors

(2010) Bader A. Salameh et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Multimeric Lactoside “Click Clusters” as Tools to Investigate the Effect of Linker Length in Specific Interactions with Peanut Lectin, Galectin-1, and -3

(2010) Sébastien G. Gouin et al.   CHEMBIOCHEM

Interaction between circulating galectin-3 and cancer-associated MUC1 enhances tumour cell homotypic aggregation and prevents anoikis

(2010) Qicheng Zhao et al.   Molecular Cancer

Application of copper(I)-catalysed azide/alkyne cycloaddition (CuAAC) ‘click chemistry’ in carbohydrate drug and neoglycopolymer synthesis

(2010) Valquiria Aragão-Leoneti et al.   TETRAHEDRON

Synthesis and Evaluation of New Thiodigalactoside-Based Chemical Probes to Label Galectin-3

(2009) Monique van Scherpenzeel et al.   CHEMBIOCHEM

Fragment-based development of triazole-substituted O-galactosyl aldoximes with fragment-induced affinity and selectivity for galectin-3

(2009) Johan Tejler et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Biological Modulation by Lectins and Their Ligands in Tumor Progression and Metastasis

(2008) Avraham Raz et al.   Anti-Cancer Agents in Medicinal Chemistry

Galectin–glycan lattices regulate cell-surface glycoprotein organization and signalling: Table 1

(2008) Omai B. Garner et al.   BIOCHEMICAL SOCIETY TRANSACTIONS

Mammalian galectins: Structure, carbohydrate specificity, and functions

(2008) E. M. Rapoport et al.   BIOCHEMISTRY-MOSCOW

Synthesis of stable and selective inhibitors of human galectins-1 and -3

(2008) Denis Giguère et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Protein subtype-targeting through ligand epimerization: Talose-selectivity of galectin-4 and galectin-8

(2008) Christopher T. Öberg et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Double Affinity Amplification of Galectin–Ligand Interactions through Arginine–Arene Interactions: Synthetic, Thermodynamic, and Computational Studies with Aromatic Diamido Thiodigalactosides

(2008) Ian Cumpstey et al.   CHEMISTRY-A EUROPEAN JOURNAL

Galectins: structure, function and therapeutic potential

(2008) Ri-Yao Yang et al.   EXPERT REVIEWS IN MOLECULAR MEDICINE

Arginine Binding Motifs: Design and Synthesis of Galactose-Derived Arginine Tweezers as Galectin-3 Inhibitors

(2008) Christopher T. Öberg et al.   JOURNAL OF MEDICINAL CHEMISTRY