Synthesis and Evaluation of Anticancer Activity of Pyrazolone Appended Triarylmethanes (TRAMs)

Troger's Base Derived Butterfly Shaped Contorted AIEgens for Dead Bacterial Cell‐Imaging

(2021) Valmik P. Jejurkar et al.   ChemistrySelect

Design, Synthesis, Molecular Docking and Anticancer Evaluation of Pyrazole Linked Pyrazoline Derivatives with Carbothioamide tail as EGFR Kinase Inhibitors

(2020) Farah Nawaz et al.   Anti-Cancer Agents in Medicinal Chemistry

2D-QSAR Modeling and Molecular Docking Studies on 1H-Pyrazole-1-carbothioamide Derivatives as EGFR Kinase Inhibitors

(2020) Tawassl T. H. Hajalsiddig et al.   ACS Omega

Design and Development of Axially Chiral Bis(Naphthofuran) Luminogens as Fluorescent Probe for Cell‐imaging

(2020) Valmik P. Jejurkar et al.   CHEMISTRY-A EUROPEAN JOURNAL

Advances in The Catalytic Synthesis of Triarylmethanes (TRAMs)

(2019) Rajpratap Kshatriya et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Solvent-Free, Mechanochemically Scalable Synthesis of 2,3-Dihydroquinazolin-4(1H)-one Using Brønsted Acid Catalyst

(2019) Gauravi Yashwantrao et al.   ACS Sustainable Chemistry & Engineering

Brønsted Acid Catalyzed Domino Synthesis of Functionalized 4H‐Chromens and Their ADMET, Molecular Docking and Antibacterial Studies

(2019) Rajpratap Kshatriya et al.   ChemistrySelect

Squaramide-Catalyzed Enantioselective Michael Addition of Pyrazol-3-ones to ortho-Quinone Methides

(2019) Laura Carceller Ferrer et al.   LETTERS IN ORGANIC CHEMISTRY

Synthesis, Antimicrobial Screening and In Silico Appraisal of Iminocarbazole Derivatives

(2019) Valmik P. Jejurkar et al.   ChemistrySelect

Repurposing mosloflavone/5,6,7-trimethoxyflavone-resveratrol hybrids: Discovery of novel p38-α MAPK inhibitors as potent interceptors of macrophage-dependent production of proinflammatory mediators

(2019) Ahmed H.E. Hassan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Pyrazolone structural motif in medicinal chemistry: Retrospect and prospect

(2019) Zefeng Zhao et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Flavone-based arylamides as potential anticancers: Design, synthesis and in vitro cell-based/cell-free evaluations

(2019) Ahmed H.E. Hassan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Overview on the Recent Strategies for the Enantioselective Synthesis of 1, 1-Diarylalkanes, Triarylmethanes and Related Molecules Containing the Diarylmethine Stereocenter

(2018) Sankalan Mondal et al.   ChemCatChem

Synthesis of Chiral Pyrazolone and Spiropyrazolone Derivatives through Squaramide-Catalyzed Reaction of Pyrazolin-5-ones with o-Quinone Methides

(2018) Ji Zhou et al.   ORGANIC LETTERS

Design, synthesis and cytotoxicity of chimeric erlotinib-alkylphospholipid hybrids

(2018) Md. Maqusood Alam et al.   BIOORGANIC CHEMISTRY

2D, 3D, G-QSAR and Docking Studies of Thiazolyl-pyrazoline Analogues as Potent (Epidermal Growth Factor Receptor-tyrosine Kinase) EGFR-TK Inhibitors

(2017) Ghodgaonkar Sunayana et al.   Letters in Drug Design & Discovery

Environmentally Benign, Highly Efficient and Expeditious Solvent-Free Synthesis of Trisubstituted Methanes Catalyzed by Sulfated Polyborate

(2017) Valmik P. Jejurkar et al.   ChemistrySelect

SwissADME: a free web tool to evaluate pharmacokinetics, drug-likeness and medicinal chemistry friendliness of small molecules

(2017) Antoine Daina et al.   Scientific Reports

Design, synthesis and biological evaluation of pyrazolyl-nitroimidazole derivatives as potential EGFR/HER-2 kinase inhibitors

(2016) Xiang-Xiang Tao et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

The role of HER2, EGFR, and other receptor tyrosine kinases in breast cancer

(2016) Jennifer L. Hsu et al.   CANCER AND METASTASIS REVIEWS

Modern advances in heterocyclic chemistry in drug discovery

(2016) Alexandria P. Taylor et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

PLIP: fully automated protein–ligand interaction profiler

(2015) Sebastian Salentin et al.   NUCLEIC ACIDS RESEARCH

Directing Group Assisted Nucleophilic Substitution of Propargylic Alcohols via o-Quinone Methide Intermediates: Brønsted Acid Catalyzed, Highly Enantio- and Diastereoselective Synthesis of 7-Alkynyl-12a-acetamido-Substituted Benzoxanthenes

(2015) Satyajit Saha et al.   ORGANIC LETTERS

Recent Advances in the Synthesis of Triarylmethanes by Transition Metal Catalysis

(2015) Masakazu Nambo et al.   ACS Catalysis

Synthetic methodologies of achiral diarylmethanols, diaryl and triarylmethanes (TRAMs) and medicinal properties of diaryl and triarylmethanes-an overview

(2014) Sankalan Mondal et al.   RSC Advances

Synthesis, molecular docking and evaluation of thiazolyl-pyrazoline derivatives as EGFR TK inhibitors and potential anticancer agents

(2011) Peng-Cheng Lv et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and biological evaluation of pyrazole derivatives containing thiourea skeleton as anticancer agents

(2010) Peng-Cheng Lv et al.   BIOORGANIC & MEDICINAL CHEMISTRY

RNA helicase A is a DNA-binding partner for EGFR-mediated transcriptional activation in the nucleus

(2010) L. Huo et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Synthesis and applications of Rhodamine derivatives as fluorescent probes

(2009) Mariana Beija et al.   CHEMICAL SOCIETY REVIEWS

Triphenylmethylamides (TPMAs): Structure–activity relationship of compounds that induce apoptosis in melanoma cells

(2008) Rahul Palchaudhuri et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

The Complex Role of the Triphenylmethyl Motif in Anticancer Compounds

(2008) Rahul Palchaudhuri et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY