The application of anisole in greener solid-phase peptide synthesis protocols – Compatibility with green bases in Fmoc removal and new green binary mixture for coupling

Transition-Metal-Free and Site-Selective Selenylation of Heterocyclic N-Oxides in Anisole as a Green Solvent

(2020) Suk Hun Lee et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Assessing the correlation of microscopy‐based and volumetry‐based measurements for resin swelling in a range of potential greener solvents for SPPS

(2020) Jordan Kevin Magtaan et al.   JOURNAL OF PEPTIDE SCIENCE

Fast Heck–Cassar–Sonogashira (HCS) Reactions in Green Solvents

(2020) L. Ferrazzano et al.   ORGANIC LETTERS

Investigation of Parameters that Affect Resin Swelling in Green Solvents

(2020) Chidi Amadi‐Kamalu et al.   ChemistryOpen

N‐Butylpyrrolidinone (NBP) for Solid‐Phase Peptide Synthesis, Environmentally Friendlier and Synthetically Better than DMF

(2020) Fernando Albericio et al.   ChemSusChem

Environmentally Friendly SPPS II: Scope of Green Fmoc Removal Protocol Using NaOH and Its Application for Synthesis of Commercial Drug Triptorelin

(2020) Adam Přibylka et al.   JOURNAL OF ORGANIC CHEMISTRY

Greening Solid-Phase Organic Synthesis: Environmentally Conscious Synthesis of Pharmaceutically Relevant Privileged Structures 5,6-Dihydropyridin-2(1H)-ones and Quinolin-2(1H)-ones

(2020) Eva Schütznerová et al.   JOURNAL OF ORGANIC CHEMISTRY

Green Solvent Selection for Suzuki–Miyaura Coupling of Amides

(2020) Peng Lei et al.   ACS Sustainable Chemistry & Engineering

The Green Transformation of Solid-Phase Peptide Synthesis

(2019) Yahya E Jad et al.   ACS Sustainable Chemistry & Engineering

Sustainability Challenges in Peptide Synthesis and Purification: From R&D to Production

(2019) Albert Isidro-Llobet et al.   JOURNAL OF ORGANIC CHEMISTRY

Making Solid-Phase Peptide Synthesis Greener: A Review of the Literature

(2019) Kyriakos G. Varnava et al.   Chemistry-An Asian Journal

A Green Approach for Organic Transformations Using Microwave Reactor

(2019) Subrata Das et al.   CURRENT ORGANIC SYNTHESIS

Green Solvent Mixtures for Solid-Phase Peptide Synthesis: A Dimethylformamide-Free Highly Efficient Synthesis of Pharmaceutical-Grade Peptides

(2019) Lucia Ferrazzano et al.   ACS Sustainable Chemistry & Engineering

Therapeutic peptides: Historical perspectives, current development trends, and future directions

(2018) Jolene L. Lau et al.   BIOORGANIC & MEDICINAL CHEMISTRY

N-Butylpyrrolidinone as Alternative Solvent for Solid-Phase Peptide Synthesis

(2018) John Lopez et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Greener solvents for solid-phase organic synthesis

(2018) Stefan B. Lawrenson   PURE AND APPLIED CHEMISTRY

Greener solvents for solid-phase synthesis

(2017) Stefan Lawrenson et al.   GREEN CHEMISTRY

The greening of peptide synthesis

(2017) Stefan B. Lawrenson et al.   GREEN CHEMISTRY

The Current State of Peptide Drug Discovery: Back to the Future?

(2017) Antoine Henninot et al.   JOURNAL OF MEDICINAL CHEMISTRY

Green Solid-Phase Peptide Synthesis (GSPPS) 3. Green Solvents for Fmoc Removal in Peptide Chemistry

(2017) Yahya E. Jad et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Green solid-phase peptide synthesis 4. γ-Valerolactone and N -formylmorpholine as green solvents for solid phase peptide synthesis

(2017) Ashish Kumar et al.   TETRAHEDRON LETTERS

Updating and further expanding GSK's solvent sustainability guide

(2016) Catherine M. Alder et al.   GREEN CHEMISTRY

CHEM21 selection guide of classical- and less classical-solvents

(2016) Denis Prat et al.   GREEN CHEMISTRY

Advances in Fmoc solid-phase peptide synthesis

(2016) Raymond Behrendt et al.   JOURNAL OF PEPTIDE SCIENCE

Deprotection Reagents in Fmoc Solid Phase Peptide Synthesis: Moving Away from Piperidine?

(2016) Omar Luna et al.   MOLECULES

Green Solid-Phase Peptide Synthesis 2. 2-Methyltetrahydrofuran and Ethyl Acetate for Solid-Phase Peptide Synthesis under Green Conditions

(2016) Yahya E. Jad et al.   ACS Sustainable Chemistry & Engineering

2-Methyltetrahydrofuran and cyclopentyl methyl ether for green solid-phase peptide synthesis

(2015) Yahya E. Jad et al.   AMINO ACIDS

Green Solvents in Carbohydrate Chemistry: From Raw Materials to Fine Chemicals

(2015) Angeles Farrán et al.   CHEMICAL REVIEWS

Development of GSK's acid and base selection guides

(2015) Richard K. Henderson et al.   GREEN CHEMISTRY

Peptide synthesis beyond DMF: THF and ACN as excellent and friendlier alternatives

(2015) Yahya E. Jad et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Polymer-Supported Stereoselective Synthesis of (1S,5S)-6-Oxa-3,8-diazabicyclo[3.2.1]octanes

(2013) Eva Schütznerová et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Development of GSK's reagent guides – embedding sustainability into reagent selection

(2013) Joseph P. Adams et al.   GREEN CHEMISTRY

2-Methyltetrahydrofuran (2-MeTHF): A Biomass-Derived Solvent with Broad Application in Organic Chemistry

(2012) Vittorio Pace et al.   ChemSusChem

Peptide Coupling Reagents, More than a Letter Soup

(2011) Ayman El-Faham et al.   CHEMICAL REVIEWS

Aspartimide formation in peptide chemistry: occurrence, prevention strategies and the role of N-hydroxylamines

(2011) Ramon Subirós-Funosas et al.   TETRAHEDRON

COMU: A Safer and More Effective Replacement for Benzotriazole-Based Uronium Coupling Reagents

(2009) Ayman El-Faham et al.   CHEMISTRY-A EUROPEAN JOURNAL

Oxyma: An Efficient Additive for Peptide Synthesis to Replace the Benzotriazole-Based HOBt and HOAt with a Lower Risk of Explosion[1]

(2009) Ramon Subirós-Funosas et al.   CHEMISTRY-A EUROPEAN JOURNAL

Solid-phase peptide synthesis using acetonitrile as a solvent in combination with PEG-based resins

(2009) Gerardo A. Acosta et al.   JOURNAL OF PEPTIDE SCIENCE

Peptidomimetics, a synthetic tool of drug discovery

(2008) Josef Vagner et al.   CURRENT OPINION IN CHEMICAL BIOLOGY