Rh(III)-Catalyzed [5 + 1] Annulation of Indole-enaminones with Diazo Compounds To Form Highly Functionalized Carbazoles

Synthesis of Highly Fused Pyrano[2,3-b]pyridines via Rh(III)-Catalyzed C–H Activation and Intramolecular Cascade Annulation under Room Temperature

(2020) Xu Han et al.   JOURNAL OF ORGANIC CHEMISTRY

Rhodium(III)-Catalyzed Redox-Neutral [3+3] Annulation of N-nitrosoanilines with Cyclopropenones: A Traceless Approach to Quinolin-4(1H)-One Scaffolds

(2020) Lingjun Liu et al.   MOLECULES

Rhodium(III)-Catalyzed C–H Alkenylation: Access to Maleimide-Decorated Tryptophan and Tryptophan-Containing Peptides

(2020) Jingjing Peng et al.   ORGANIC LETTERS

Sulfoximines-Assisted Rh(III)-Catalyzed C–H Activation and Intramolecular Annulation for the Synthesis of Fused Isochromeno-1,2-Benzothiazines Scaffolds under Room Temperature

(2020) Bao Wang et al.   MOLECULES

Rh(III)-Catalyzed Dual C–H Functionalization/Cyclization Cascade by a Removable Directing Group: A Method for Synthesis of Polycyclic Fused Pyrano[de]Isochromenes

(2020) Zhihao Shu et al.   JOURNAL OF ORGANIC CHEMISTRY

Rhodium-catalyzed C H activation/cyclization of enaminones with sulfoxonium ylides toward polysubstituted naphthalenes

(2019) Zhenlian Wang et al.   TETRAHEDRON LETTERS

Rh(III)-Catalyzed Annulation of Boc-Protected Benzamides with Diazo Compounds: Approach to Isocoumarins

(2019) Guangyu Dong et al.   MOLECULES

Cp*Rh(III)-Catalyzed C–H Bond Difluorovinylation of Indoles with α,α-Difluorovinyl Tosylate

(2019) Lisheng Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Rh(III)-Catalyzed Hydroarylation of Alkyne MIDA Boronates via C–H Activation of Indole Derivatives

(2019) Xiao Fei et al.   JOURNAL OF ORGANIC CHEMISTRY

Rhodium(III)-Catalyzed [4+2] Annulation via C-H Activation: Synthesis of Multi-Substituted Naphthalenone Sulfoxonium Ylides

(2019) Xiaohan Song et al.   MOLECULES

A General Carbazole Synthesis via Stitching of Indole–Ynones with Nitromethanes: Application to Total Synthesis of Carbazomycin A, Calothrixin B, and Staurosporinone

(2019) Shweta Singh et al.   ORGANIC LETTERS

C3‐Functionalized Chromones Synthesis by Tandem C−H Elaboration and Chromone Annulation of Enaminones

(2019) Leiqing Fu et al.   Asian Journal of Organic Chemistry

Enaminone, Enaminoesters, and Related Compounds in the Metal-Free Synthesis of Pyridines and Fused Pyridines

(2019) Branko Stanovnik   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 2-Amino-5-acylthiazoles by a Tertiary Amine-Promoted One-Pot Three-Component Cascade Cyclization Using Elemental Sulfur as a Sulfur Source

(2019) Rong-Geng Fu et al.   JOURNAL OF ORGANIC CHEMISTRY

Rh(III)-Catalyzed C–H Bond Activation for the Construction of Heterocycles with sp3-Carbon Centers

(2019) Run Wang et al.   Catalysts

One-Pot Synthesis of 5-Acyl-1,2,3-Thiadiazoles from Enaminones, Tosylhydrazine, and Elemental Sulfur under Transition-Metal-Free Conditions

(2019) Zan Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Regioselective Cyclization of (Indol-3-yl)pentyn-3-ols as an Approach to (Tetrahydro)carbazoles

(2018) Prabhakararao Tharra et al.   ORGANIC LETTERS

Rh(III)-Catalyzed C–H Activation of Benzoylacetonitriles and Tandem Cyclization with Diazo Compounds to Substituted Benzo[de]chromenes

(2018) Feifei Fang et al.   ORGANIC LETTERS

Regioselective Formal [4 + 2] Cycloadditions of Enaminones with Diazocarbonyls through RhIII-Catalyzed C–H Bond Functionalization

(2018) Shuguang Zhou et al.   ORGANIC LETTERS

Rh(III)-Catalyzed Enaminone-Directed Alkenyl C–H Activation for the Synthesis of Salicylaldehydes

(2018) Bing Qi et al.   ORGANIC LETTERS

Rh(III)-Catalyzed Enaminone-Directed C–H Coupling with α-Diazo-α-phosphonoacetate for Reactivity Discovery: Fluoride-Mediated Dephosphonation for C–C Coupling Reactions

(2018) Chao Song et al.   ORGANIC LETTERS

Bismuth(III) Triflate Catalyzed Three-Component Reactions of Indoles, Ketones, and α-Bromoacetaldehyde Acetals Enable Indole-to-Carbazole Transformation

(2018) Yanlong Gu et al.   ORGANIC LETTERS

Overview on the synthetic routes to nicotine nitriles

(2018) M. A. Salem et al.   SYNTHETIC COMMUNICATIONS

Cytotoxic indolocarbazoles alkaloids from the streptomyces sp. A65

(2018) Biao Zhou et al.   TETRAHEDRON

Rhodium(III)-Catalyzed C-H Activation of Benzoylacetonitriles and Cyclization with Sulfoxonium Ylides to Naphthols

(2018) Chaofan Zhou et al.   ADVANCED SYNTHESIS & CATALYSIS

Rhodium(III)-Catalyzed C–H Activation of α-Iminonitriles or α-Imino Esters and Cyclization with Acrylates to 2H-Isoindoles

(2018) Yazhou Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Synergistic Indium and Silver Dual Catalysis: A Regioselective [2 + 2 + 1]-Oxidative N-Annulation Approach for the Diverse and Polyfunctionalized N-Arylpyrazoles

(2018) Raju S. Thombal et al.   ORGANIC LETTERS

Reactivity of Morita–Baylis–Hillman Adducts in C–H Functionalization of (Hetero)aryl Nitrones: Access to Bridged Cycles and Carbazoles

(2018) Ashok Kumar Pandey et al.   ORGANIC LETTERS

Rh(iii)-Catalyzed regioselective C–H [4 + 2] C-annulation of vinyl enaminones with alkynes to form polysubstituted salicylaldehydes

(2018) Yinsong Zhao et al.   Organic Chemistry Frontiers

Carbene-Catalyzed Construction of Carbazoles from Enals and 2-Methyl-3-oxoacetate Indoles

(2018) Dehai Liu et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Polyaromatic Rings: Rh(III)-Catalyzed [5 + 1] Annulation of Enaminones with Vinyl Esters through C–H Bond Functionalization

(2018) Gaohui Liang et al.   ORGANIC LETTERS

Direct Synthesis of 3-Acylindoles through Rhodium(III)-Catalyzed Annulation of N-Phenylamidines with α-Cl Ketones

(2018) Jianhui Zhou et al.   ORGANIC LETTERS

Brønsted Acid Catalyzed One-Pot Benzannulation of 2-Alkenylindoles under Aerial Oxidation: A Route to Carbazoles and Indolo[2,3-a]carbazole Alkaloids

(2018) Shuvendu Saha et al.   ORGANIC LETTERS

Rh(III)-Catalyzed C–H Cyclization of Arylnitrones with Diazo Compounds: Access to 3-Carboxylate Substituted N-Hydroxyindoles

(2017) Yazhou Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Modular Synthesis of Carbazole-Based Conjugated Molecules through a One-Pot Annulation/Dehydrogenation Sequence

(2017) Shanping Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis, in vitro antiproliferative activity, antioxidant activity and molecular modeling studies of new carbazole Mannich bases

(2017) Pedavenkatagari Narayana Reddy et al.   MEDICINAL CHEMISTRY RESEARCH

Propargyl Alcohols as One-Carbon Synthons: Redox-Neutral Rhodium(III)-Catalyzed C–H Bond Activation for the Synthesis of Isoindolinones Bearing a Quaternary Carbon

(2017) Xiaowei Wu et al.   ORGANIC LETTERS

N-Bromosuccinimide (NBS)-Catalyzed C–H Bond Functionalization: An Annulation of Alkynes with Electron Withdrawing Group (EWG)-Substituted Acetyl Indoles for the Synthesis of Carbazoles

(2017) Han Wang et al.   ORGANIC LETTERS

Cobalt(III)- and Rhodium(III)-Catalyzed C–H Amidation and Synthesis of 4-Quinolones: C–H Activation Assisted by Weakly Coordinating and Functionalizable Enaminone

(2017) Fen Wang et al.   ORGANIC LETTERS

One-pot synthesis of carbazoles from indoles via a metal free benzannulation

(2017) Sambasivarao Kotha et al.   TETRAHEDRON LETTERS

Recent developments in chemical reactivity of N,N-dimethylenamino ketones as synthons for various heterocycles

(2017) Hatem M. Gaber et al.   RSC Advances

Enaminones as Synthons for a Directed C−H Functionalization: RhIII -Catalyzed Synthesis of Naphthalenes

(2016) Shuguang Zhou et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Visible light-photocatalysed carbazole synthesis via a formal (4+2) cycloaddition of indole-derived bromides and alkynes

(2016) Zhi-Guang Yuan et al.   CHEMICAL COMMUNICATIONS

Synthesis of Benzo[a]carbazoles and an Indolo[2,3-a]carbazole from 3-Aryltetramic Acids

(2016) Nathanyal J. Truax et al.   JOURNAL OF ORGANIC CHEMISTRY

KIO3-Catalyzed Aerobic Cross-Coupling Reactions of Enaminones and Thiophenols: Synthesis of Polyfunctionalized Alkenes by Metal-Free C–H Sulfenylation

(2016) Jie-Ping Wan et al.   ORGANIC LETTERS

Indole-to-Carbazole Strategy for the Synthesis of Substituted Carbazoles under Metal-Free Conditions

(2016) Shanping Chen et al.   ORGANIC LETTERS

Biological potential of carbazole derivatives

(2015) Agata Głuszyńska   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Silver(I)-Catalyzed Dearomatization of Alkyne-Tethered Indoles: Divergent Synthesis of Spirocyclic Indolenines and Carbazoles

(2015) Michael J. James et al.   ORGANIC LETTERS

Facile Synthesis of Carbazoles via a Tandem Iodocyclization with 1,2-Alkyl Migration and Aromatization

(2015) Jia Wang et al.   ORGANIC LETTERS

Palladium-Catalyzed Triple Successive C–H Functionalization: Direct Synthesis of Functionalized Carbazoles from Indoles

(2015) Akhilesh K. Verma et al.   ORGANIC LETTERS

Rh(I)-catalyzed decarbonylation synthesis of carbazoles via C–N cleavage

(2015) Weizheng Fan et al.   TETRAHEDRON

From Indoles to Carbazoles: Tandem Cp*Rh(III)-Catalyzed C–H Activation/Brønsted Acid-Catalyzed Cyclization Reactions

(2015) Jia-Qiang Wu et al.   ACS Catalysis

A General Diversified Synthesis of Carbazoles and the First Synthesis of Karapinchamine A

(2014) Youai Qiu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis, biological evaluation and molecular modeling study of novel tacrine–carbazole hybrids as potential multifunctional agents for the treatment of Alzheimer's disease

(2014) Supatra Thiratmatrakul et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Benzannulation of Indoles to Carbazoles and Its Applications for Syntheses of Carbazole Alkaloids

(2014) Xiaojian Zheng et al.   ORGANIC LETTERS

Synthesis and evaluation of cytotoxic activities of new guanidines derived from carbazoles

(2013) Anna Caruso et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Occurrence, Biogenesis, and Synthesis of Biologically Active Carbazole Alkaloids

(2012) Arndt W. Schmidt et al.   CHEMICAL REVIEWS

Oridamycins A and B, Anti-Saprolegnia parasiticaIndolosesquiterpenes Isolated fromStreptomycessp. KS84

(2010) Kentaro Takada et al.   JOURNAL OF NATURAL PRODUCTS

An efficient synthesis of carbazoles from PtCl2-catalyzed cyclization of 1-(indol-2-yl)-2,3-allenols

(2009) Wangqing Kong et al.   CHEMICAL COMMUNICATIONS

γ-Lactone Carbazoles fromClausena anisata

(2009) Chihiro Ito et al.   JOURNAL OF NATURAL PRODUCTS

Synthesis of Carbazoles and 1,2-Dihydrocarbazoles by Domino ‘Twofold Heck-6π-Electrocyclization’ Reactions of Di- and Tribromo-N-methylindoles

(2009) Peter Langer et al.   SYNLETT

Intramolecular Pd(II)-Catalyzed Oxidative Biaryl Synthesis Under Air: Reaction Development and Scope

(2008) Benoît Liégault et al.   JOURNAL OF ORGANIC CHEMISTRY