Metal‐Free Synthesis of Anthranils by PhIO Mediated Heterocyclization of ortho ‐Carbonyl Anilines

Synthesis of 2,1-Benzoisoxazole-Containing 1,2,3-Triazoles through Copper-Catalyzed Three-Component Domino Reactions of o-Bromoacetophenones, Aldehydes, and Sodium Azide

(2020) Yuwei Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Rh-Catalyzed C–H Amination/Annulation of Acrylic Acids and Anthranils by Using −COOH as a Deciduous Directing Group: An Access to Diverse Quinolines

(2020) Yang Gao et al.   ORGANIC LETTERS

An overview on medicinal perspective of thiazolidine-2,4-dione: A remarkable scaffold in the treatment of type 2 diabetes

(2020) Garima Bansal et al.   Journal of Advanced Research

Copper-Catalyzed Electrophilic Amination of Arylboronic Acids with Anthranils: An Access to N-Aryl-2-aminophenones

(2020) Yang Gao et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal-Free, Visible-Light-Enabled Direct C3–H Arylation of Anthranils

(2020) Tapas Adak et al.   ORGANIC LETTERS

Quinoline-Fused Lactones via Tandem Oxidation Cyclization: Metal-Free sp3 C–H Functionalization

(2020) Alankrita Garia et al.   JOURNAL OF ORGANIC CHEMISTRY

Thermo-promoted Reactions of Anthranils with Carboxylic Acids, Amines, Phenols and Malononitrile under Catalyst-free Conditions

(2019) Jing Jiang et al.   JOURNAL OF ORGANIC CHEMISTRY

Transition-Metal-Free Synthesis of Fused Quinazolinones by Oxidative Cyclization of N-Pyridylindoles

(2019) Alankrita Garia et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 3-phenylbenzo[c]isoxazoles by thermocyclization of 2-azidobenzophenones

(2019) A. V. Odinokov et al.   RUSSIAN CHEMICAL BULLETIN

Rhodium-Catalyzed Reaction of Sulfoxonium Ylides and Anthranils toward Indoloindolones via a (4 + 1) Annulation

(2019) Xiaopeng Wu et al.   ORGANIC LETTERS

Base-Mediated [3 + 4]-Cycloaddition of Anthranils with Azaoxyallyl Cations: A New Approach to Multisubstituted Benzodiazepines

(2019) Juan Feng et al.   ORGANIC LETTERS

Practical Synthesis of Benzimidazo[1,2-a]quinolines via Rh(III)-Catalyzed C–H Activation Cascade Reaction from Imidamides and Anthranils

(2019) Yao Hu et al.   ORGANIC LETTERS

Dual Role of Anthranils as Amination and Transient Directing Group Sources: Synthesis of 2-Acyl Acridines

(2018) Saegun Kim et al.   ORGANIC LETTERS

Cobalt-Catalyzed Electrophilic Aminations with Anthranils: An Expedient Route to Condensed Quinolines

(2018) Jie Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rapid and High-Yield Electrosynthesis of Benzisoxazole and Some Derivatives

(2018) Seyyedamirhossein Hosseini et al.   ChemElectroChem

Recent Advances in Iodosobenzene-Mediated Construction of Heterocyclic Scaffolds: Transition-Metal-Free Approaches and Scope

(2017) Krishnanka Shekhar Gayen et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Diverting Reactive Intermediates Toward Unusual Chemistry: Unexpected Anthranil Products from Davis–Beirut Reaction

(2017) Jie S. Zhu et al.   JOURNAL OF ORGANIC CHEMISTRY

Benzisoxazole: a privileged scaffold for medicinal chemistry

(2017) K. P. Rakesh et al.   MedChemComm

Chemoselective Reductive Heterocyclization by Controlling the Binomial Architecture of Metal Particles and Acid–Base Properties of the Support

(2017) L. Marti et al.   ACS Catalysis

Sulfimine-Promoted Fast O Transfer: One-step Synthesis of Sulfoximine from Sulfide

(2017) Yongtao Xie et al.   ChemistrySelect

Transfer of Electrophilic NH Using Convenient Sources of Ammonia: Direct Synthesis of NH Sulfoximines from Sulfoxides

(2016) Marina Zenzola et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of 2,1-benzisoxazole-3(1H)-ones by base-mediated photochemical N–O bond-forming cyclization of 2-azidobenzoic acids

(2016) Daria Yu Dzhons et al.   Beilstein Journal of Organic Chemistry

Silver- versus gold-catalyzed sequential oxidative cyclization of unprotected 2-alkynylanilines with oxone

(2016) A. Arcadi et al.   CHEMICAL COMMUNICATIONS

Advances in Synthetic Applications of Hypervalent Iodine Compounds

(2016) Akira Yoshimura et al.   CHEMICAL REVIEWS

Cooperative Co(III)/Cu(II)-Catalyzed C–N/N–N Coupling of Imidates with Anthranils: Access to 1H-Indazoles via C–H Activation

(2016) Lei Li et al.   ORGANIC LETTERS

Synthesis of 3-Substituted 2,1-Benzisoxazoles by the Oxidative Cyclization of 2-Aminoacylbenzenes with Oxone

(2016) Antonio Arcadi et al.   SYNTHESIS-STUTTGART

Synthesis and pharmacological characterization of 2-aminobenzaldehyde oxime analogs as dual inhibitors of neutrophil elastase and proteinase 3

(2015) Tsong-Long Hwang et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Copper-Catalyzed Direct Synthesis of 1,2,4-Oxadiazoles from Amides and Organic Nitriles by Oxidative N-O Bond Formation

(2015) Malleswara Rao Kuram et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Utility of Nitrogen Extrusion of Azido Complexes for the Synthesis of Nitriles, Benzoxazoles, and Benzisoxazoles

(2015) Phongprapan Nimnual et al.   JOURNAL OF ORGANIC CHEMISTRY

Substrate Controlled Synthesis of Benzisoxazole and Benzisothiazole Derivatives via PhI(OAc)2-Mediated Oxidation Followed by Intramolecular Oxidative O–N/S–N Bond Formation

(2015) Devireddy Anand et al.   JOURNAL OF ORGANIC CHEMISTRY

General synthesis of 2,1-benzisoxazoles (anthranils) from nitroarenes and benzylic C–H acids in aprotic media promoted by combination of strong bases and silylating agents

(2015) Michał Wiȩcław et al.   MOLECULAR DIVERSITY

One-pot synthesis of 2,1-benzisoxazoles (anthranils) by a stannous chloride-mediated tandem reduction–heterocyclization of 2-nitroacylbenzenes under neutral conditions

(2012) Jay Chauhan et al.   TETRAHEDRON LETTERS

Identification of Novel Antitubulin Agents by Using a Virtual Screening Approach Based on a 7-Point Pharmacophore Model of the Tubulin Colchi-Site

(2011) Alberto Massarotti et al.   Chemical Biology & Drug Design

Chameleonic Reactivity of Vicinal Diazonium Salt of Acetylenyl-9,10-anthraquinones: Synthetic Application toward Two Heterocyclic Targets

(2011) A. A. Stepanov et al.   JOURNAL OF ORGANIC CHEMISTRY

Intramolecular Fe(II)-Catalyzed N−O or N−N Bond Formation from Aryl Azides

(2010) Benjamin J. Stokes et al.   ORGANIC LETTERS

Metal-Free Intramolecular Aziridination of Alkenes Using Hypervalent Iodine Based Sulfonyliminoiodanes

(2009) Robert M. Moriarty et al.   ORGANIC LETTERS

Docking Study Yields Four Novel Inhibitors of the Protooncogene Pim-1 Kinase†

(2008) Albert C. Pierce et al.   JOURNAL OF MEDICINAL CHEMISTRY