Design, synthesis, and biological evaluation of novel bromo-pyrimidine analogues as tyrosine kinase inhibitors

Past, present, and future of Bcr-Abl inhibitors: from chemical development to clinical efficacy

(2018) Federico Rossari et al.   Journal of Hematology & Oncology

Part-1: Design, synthesis and biological evaluation of novel bromo-pyrimidine analogs as tyrosine kinase inhibitors

(2016) Chandrashekar Suradhenupura Munikrishnappa et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Improved Angiostatic Activity of Dasatinib by Modulation with Hydrophobic Chains

(2015) Emilia Păunescu et al.   ACS Medicinal Chemistry Letters

Biphenyl derivatives incorporating urea unit as novel VEGFR-2 inhibitors: Design, synthesis and biological evaluation

(2013) Chen Wang et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and biological evaluation of novel 4,5-dihydropyrazole derivatives as potent anticancer and antimicrobial agents

(2012) Y. Rajendra Prasad et al.   MEDICINAL CHEMISTRY RESEARCH

Exploration of (S)-3-aminopyrrolidine as a potentially interesting scaffold for discovery of novel Abl and PI3K dual inhibitors

(2011) Cunlong Zhang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design and synthesis of novel Gefitinib analogues with improved anti-tumor activity

(2010) Xiaoqing Wu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis of new 4-isopropylthiazole hydrazide analogs and some derived clubbed triazole, oxadiazole ring systems – A novel class of potential antibacterial, antifungal and antitubercular agents

(2009) B.P. Mallikarjuna et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Molecular biology of bcr-abl1-positive chronic myeloid leukemia

(2008) A. Quintas-Cardama et al.   BLOOD

Therapeutic Options Against BCR-ABL1 T315I-Positive Chronic Myelogenous Leukemia

(2008) A. Quintas-Cardama et al.   CLINICAL CANCER RESEARCH

Synthesis of some new 1,2,4-triazoles, their Mannich and Schiff bases and evaluation of their antimicrobial activities

(2008) Hacer Bayrak et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and antimicrobial studies of novel dichlorofluorophenyl containing aminotriazolothiadiazines

(2007) Mari Sithambaram Karthikeyan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Overcoming kinase resistance in chronic myeloid leukemia

(2007) Francis Lee et al.   INTERNATIONAL JOURNAL OF BIOCHEMISTRY & CELL BIOLOGY