Styrylsulfonates and -Sulfonamides through Pd-Catalysed Matsuda-Heck Reactions of Vinylsulfonic Acid Derivatives and Arenediazonium Salts

Total Synthesis of K777: Successful Application of Transition-Metal-Catalyzed Alkyne Hydrothiolation toward the Modular Synthesis of a Potent Cysteine Protease Inhibitor

(2016) Erica R. Kiemele et al.   ORGANIC LETTERS

Stereoselective Synthesis of 3-Hydroxy-4-arylcyclopentanones and 4-Arylcyclopentenones through a Heck-Matsuda Desymmetrization ofmeso cis-4-Cyclopentene-1,3-diol

(2015) Rafaela C. Carmona et al.   ADVANCED SYNTHESIS & CATALYSIS

Highlytrans-Selective Arylation of Achmatowicz Rearrangement Products by Reductive γ-Deoxygenation and Heck-Matsuda Reaction: Asymmetric Total Synthesis of (−)-Musellarins A-C and Their Analogues

(2015) Zhilong Li et al.   CHEMISTRY-A EUROPEAN JOURNAL

Acetamidoarenediazonium Salts: Opportunities for Multiple Arene Functionali­zation

(2015) Bernd Schmidt et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Propofol depresses cerebellar Purkinje cell activity via activation of GABAA and glycine receptors in vivo in mice

(2015) Ri Jin et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

Dual Role of Acetanilides: Traceless Removal of a Directing Group through Deacetylation/Diazotation and Palladium-Catalyzed C–C-Coupling Reactions

(2015) Bernd Schmidt et al.   JOURNAL OF ORGANIC CHEMISTRY

Stereoselective Synthesis of Z-α,β-Unsaturated Sulfones Using Peterson Reagents

(2015) Kaori Ando et al.   ORGANIC LETTERS

An efficient one-pot, three-component synthesis of vinyl sulfones via iodide-catalyzed radical alkenylation

(2015) Weizheng Fan et al.   TETRAHEDRON

Synthesis and Evaluation of Oxyguanidine Analogues of the Cysteine Protease Inhibitor WRR-483 against Cruzain

(2015) Brian D. Jones et al.   ACS Medicinal Chemistry Letters

Heck-Matsuda Arylation of Olefins Through a Bicatalytic Approach: Improved Procedures and Rationalization

(2014) Nicolas Oger et al.   ADVANCED SYNTHESIS & CATALYSIS

The Evolving Role of Chemical Synthesis in Antibacterial Drug Discovery

(2014) Peter M. Wright et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Vinylsulfones Via Palladium-Catalyzed Decarboxylative Coupling of Cinnamic Acids with Aromatic Sulfinic Acid Sodium Salts

(2014) Ruqing Guo et al.   CATALYSIS LETTERS

An Easy Route to (Hetero)arylboronic Acids

(2014) William Erb et al.   CHEMISTRY-A EUROPEAN JOURNAL

Discovery of Vinyl Sulfones as a Novel Class of Neuroprotective Agents toward Parkinson’s Disease Therapy

(2014) Seo Yeon Woo et al.   JOURNAL OF MEDICINAL CHEMISTRY

Continuous-Flow Heck–Matsuda Reaction: Homogeneous versus Heterogeneous Palladium Catalysts

(2014) Nicolas Oger et al.   JOURNAL OF ORGANIC CHEMISTRY

Chemo-, Regio- and Stereoselective Heck Arylation of Allylated Malonates: Mechanistic Insights by ESI-MS and Synthetic Application toward 5-Arylmethyl-γ-lactones

(2014) Caio C. Oliveira et al.   ORGANIC LETTERS

Design and synthesis of 2-substituted benzoxazoles as novel PTP1B inhibitors

(2013) Arun P. Chandrasekharappa et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of pyrrolyl and pyrazolyl sulfonamides

(2013) V. Padmavathi et al.   Chemistry of Heterocyclic Compounds

Convenient Synthesis of Various Substituted Homotaurines from Alk-2-enamides

(2013) Youfeng Nai et al.   HELVETICA CHIMICA ACTA

Scope and limitations of the Heck–Matsuda-coupling of phenol diazonium salts and styrenes: a protecting-group economic synthesis of phenolic stilbenes

(2013) Bernd Schmidt et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

“Dba-free” palladium intermediates of the Heck–Matsuda reaction

(2013) Angelo H. L. Machado et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Palladium-Catalyzed Asymmetric Addition of Diarylphosphines to α,β-Unsaturated Sulfonic Esters for the Synthesis of Chiral Phosphine Sulfonate Compounds

(2013) Junzhu Lu et al.   ORGANIC LETTERS

A simple catalytic system based on PdCl2(CH3CN)2 in water for cross-coupling reactions using diazonium salts

(2013) Ouissam El Bakouri et al.   TETRAHEDRON

Fluorous mixture synthesis of fluorous-Fmoc reagents using a one-pot double tagging strategy

(2013) Yuya Sugiyama et al.   TETRAHEDRON LETTERS

Dual Catalysis: Vinyl Sulfones through Tandem Iron-Catalyzed Allylic Sulfonation Amine-Catalyzed Isomerization

(2012) Markus Jegelka et al.   ChemCatChem

Selective arene functionalization through sequential oxidative and non-oxidative Heck reactions

(2012) Bernd Schmidt et al.   CHEMICAL COMMUNICATIONS

Sustainable Heck-Matsuda Reaction with Catalytic Amounts of Diazonium Salts: An Experimental and Theoretical Study

(2012) Nicolas Susperregui et al.   CHEMISTRY-A EUROPEAN JOURNAL

Heck-Matsuda Arylation as a Strategy to Access Kavalactones Isolated from Polygala sabulosa, Piper methysticum, and Analogues

(2012) Cristian Soldi et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Stereoselective Arylation of Substituted Cyclopentenes by Substrate-Directable Heck–Matsuda Reactions: A Concise Total Synthesis of the Sphingosine 1-Phosphate Receptor (S1P1) Agonist VPC01091

(2012) Caio C. Oliveira et al.   JOURNAL OF ORGANIC CHEMISTRY

Effect of Chiral Diene Ligands in Rhodium-Catalyzed Asymmetric Addition of Arylboronic Acids to α,β-Unsaturated Sulfonyl Compounds

(2012) Takahiro Nishimura et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Coumarins from Free ortho-Hydroxy Cinnamates by Heck-Matsuda Arylations: A Scalable Total Synthesis of (R)-Tolterodine

(2012) Daniela A. Barancelli et al.   ORGANIC LETTERS

Palladium-Nanoparticle-Catalyzed Matsuda–Heck Reaction in Water

(2012) Dattaprasad Pore et al.   SYNLETT

Synthesis of an Isoindoline-Annulated, Tricyclic Sultam Library via Microwave-Assisted, Continuous-Flow Organic Synthesis (MACOS)

(2012) Paul Hanson et al.   SYNTHESIS-STUTTGART

The first examples of the enantioselective Heck–Matsuda reaction: arylation of unactivated cyclic olefins using chiral bisoxazolines

(2012) Carlos Roque D. Correia et al.   TETRAHEDRON LETTERS

Synthesis of a Unique Isoindoline/Tetrahydroisoquinoline-based Tricyclic Sultam Library Utilizing a Heck-aza-Michael Strategy

(2012) Qin Zang et al.   ACS Combinatorial Science

Functionalization of the 3-Position of Thiophene and Benzo[b]thiophene Moieties by Palladium-Catalyzed CC Bond Forming Reactions using Diazonium Salts

(2011) Mónica Raduán et al.   ADVANCED SYNTHESIS & CATALYSIS

Aryl Diazonium versus Iodonium Salts: Preparation, Applications and Mechanisms for the Suzuki-Miyaura Cross-Coupling Reaction

(2011) Hélène Bonin et al.   ADVANCED SYNTHESIS & CATALYSIS

Evolution and Synthetic Applications of the Heck-Matsuda Reaction: The Return of Arenediazonium Salts to Prominence

(2011) Jason G. Taylor et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Pd-Catalyzed Arylation Reactions with Phenol Diazonium Salts: Application in the Synthesis of Diarylheptanoids

(2011) Bernd Schmidt et al.   JOURNAL OF ORGANIC CHEMISTRY

A Domino Approach (Hydrolysis/Dehydrohalogenation/Heck Coupling) for the Synthesis of Styrene Sulfonate Salts

(2011) G. K. Surya Prakash et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Unprecedented Substoichiometric Use of Hazardous Aryl Diazonium Salts in the Heck-Matsuda Reaction via a Double Catalytic Cycle

(2011) François Le Callonnec et al.   ORGANIC LETTERS

Fluorous aryl compounds by Matsuda–Heck reaction

(2011) Jordi Salabert et al.   TETRAHEDRON

Recent advances in the Heck–Matsuda reaction in heterocyclic chemistry

(2011) François-Xavier Felpin et al.   TETRAHEDRON

Mizoroki-Heck Reactions with 4-Phenoldiazonium Salts

(2010) Bernd Schmidt et al.   ADVANCED SYNTHESIS & CATALYSIS

A Selective and Benign Synthesis of Functionalized Benzalacetones via Mizoroki-Heck Reaction Using Aryldiazonium Salts

(2010) Therese Stern et al.   ADVANCED SYNTHESIS & CATALYSIS

Asymmetric Organocatalysis with Sulfones

(2010) Martin Nielsen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Discovery of novel N-acylsulfonamide analogs as potent and selective EP3 receptor antagonists

(2010) Masaki Asada et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

PhI(OAc)2/KI-Mediated Reaction of Aryl Sulfinates with Alkenes, Alkynes, and α,β-Unsaturated Carbonyl Compounds: Synthesis of Vinyl Sulfones and β-Iodovinyl Sulfones

(2010) Praewpan Katrun et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A sulfonamidoquinoline-derived Zn2+ fluorescent sensor with 1:1 Zn2+ binding stoichiometry

(2010) Changli Zhang et al.   INORGANIC CHEMISTRY COMMUNICATIONS

Nicotine self-administration differentially modulates glutamate and GABA transmission in hypothalamic paraventricular nucleus to enhance the hypothalamic-pituitary-adrenal response to stress

(2010) Guoliang Yu et al.   JOURNAL OF NEUROCHEMISTRY

Functionalized alkoxy arene diazonium salts from paracetamol

(2010) Bernd Schmidt et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Tandem Ir-Catalyzed Allylic Substitution Reaction of Allyl Sulfinates and Isomerization

(2010) Qing-Long Xu et al.   ORGANIC LETTERS

6,7-Dihydro-5H-pyrrolo[1,2-a] imidazoles as potent and selective α1A adrenoceptor partial agonists

(2009) Lee R. Roberts et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Deprotection of Arenediazonium Tetrafluoroborate Ethers with BBr3

(2009) Ngoc Hoa Nguyen et al.   JOURNAL OF ORGANIC CHEMISTRY

Dihydroxylation of Vinyl Sulfones: Stereoselective Synthesis of (+)- and (−)-Febrifugine and Halofuginone

(2009) Noel P. McLaughlin et al.   JOURNAL OF ORGANIC CHEMISTRY

Pd-catalyzed Heck reaction for the synthesis of isomeric metallo tetravinylsulfo phthalocyanines and their photosensitizing properties

(2009) Hasrat Ali et al.   PHOTOCHEMICAL & PHOTOBIOLOGICAL SCIENCES

Analogues of 2-phenyl-ethenesulfonic acid phenyl ester have dual functions of inhibiting expression of inducible nitric oxide synthase and activating peroxisome proliferator-activated receptor γ

(2008) Yue-Zhi Lee et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

A versatile synthesis of 2,4-substituted oxazoles

(2008) Vijay Chudasama et al.   CHEMICAL COMMUNICATIONS

Catalytic Asymmetric Conjugate Addition of Grignard Reagents to α,β-Unsaturated Sulfones

(2008) Pieter H. Bos et al.   ORGANIC LETTERS

“Click, Click, Cyclize”: A DOS Approach to Sultams Utilizing Vinyl Sulfonamide Linchpins

(2008) Aihua Zhou et al.   ORGANIC LETTERS