Propylphosphonic Anhydride (T3P®) as Coupling Reagent for Solid‐Phase Peptide Synthesis

OxymaPure Coupling Reagents: Beyond Solid-Phase Peptide Synthesis

(2020) Ayman El-Faham et al.   SYNTHESIS-STUTTGART

Sustainability Challenges in Peptide Synthesis and Purification: From R&D to Production

(2019) Albert Isidro-Llobet et al.   JOURNAL OF ORGANIC CHEMISTRY

γ-Valerolactone (GVL): An eco-friendly anchoring solvent for solid-phase peptide synthesis

(2019) Othman Al Musaimi et al.   TETRAHEDRON LETTERS

Rapid Development of a Commercial Process for Linrodostat, an Indoleamine 2,3-Dioxygenase (IDO) Inhibitor

(2019) Kenneth J. Fraunhoffer et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Anaphylaxis Induced by Peptide Coupling Agents: Lessons Learned from Repeated Exposure to HATU, HBTU, and HCTU

(2019) Kate J. McKnelly et al.   JOURNAL OF ORGANIC CHEMISTRY

Choosing the Right Coupling Reagent for Peptides: A Twenty-Five-Year Journey

(2018) Fernando Albericio et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Regeneration of aged DMF for use in solid-phase peptide synthesis

(2018) Jordan Kevin Magtaan et al.   JOURNAL OF PEPTIDE SCIENCE

Cyclization of Linear Tetrapeptides Containing N -Methylated Amino Acids by using 1-Propanephosphonic Acid Anhydride

(2016) Shengping Zhang et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

An optimized and scalable synthesis of propylphosphonic anhydride for general use

(2015) Hana Pizova et al.   TETRAHEDRON LETTERS

An Efficient and Epimerization Free Synthesis of C-Terminal Arylamides Derived from α-Amino Acids and Peptide Acids via T3P Activation

(2014) Chilakapati Madhu et al.   International Journal of Peptide Research and Therapeutics

K-Oxyma: a Strong Acylation-Promoting, 2-CTC Resin-Friendly Coupling Additive

(2013) Prabhakar Cherkupally et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Propanephosphonic Acid Anhydride (T3P®) - A Benign Reagent for Diverse Applications Inclusive of Large-Scale Synthesis

(2013) Vommina Sureshbabu et al.   SYNTHESIS-STUTTGART

Evaluation of alternative solvents in common amide coupling reactions: replacement of dichloromethane and N,N-dimethylformamide

(2012) Donna S. MacMillan et al.   GREEN CHEMISTRY

Peptide Coupling Reagents, More than a Letter Soup

(2011) Ayman El-Faham et al.   CHEMICAL REVIEWS

General and Scalable Amide Bond Formation with Epimerization-Prone Substrates Using T3P and Pyridine

(2011) Joshua R. Dunetz et al.   ORGANIC LETTERS

A Novel Family of Onium Salts Based Upon Isonitroso Meldrum's Acid Proves Useful as Peptide Coupling Reagents

(2010) Ayman El-Faham et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

PyOxP and PyOxB: the Oxyma-based novel family of phosphonium salts

(2010) Ramon Subirós-Funosas et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

COMU: A Safer and More Effective Replacement for Benzotriazole-Based Uronium Coupling Reagents

(2009) Ayman El-Faham et al.   CHEMISTRY-A EUROPEAN JOURNAL

Oxyma: An Efficient Additive for Peptide Synthesis to Replace the Benzotriazole-Based HOBt and HOAt with a Lower Risk of Explosion[1]

(2009) Ramon Subirós-Funosas et al.   CHEMISTRY-A EUROPEAN JOURNAL

COMU: A third generation of uronium-type coupling reagents

(2009) Ayman El-Faham et al.   JOURNAL OF PEPTIDE SCIENCE

Propylphosphonic Anhydride (T3P®): A Remarkably Efficient Reagent for the One-Pot Transformation of Aromatic, Heteroaromatic, and Aliphatic Aldehydes to Nitriles

(2009) John Augustine et al.   SYNLETT