Polymeric Precipitation Inhibitor–Based Solid Supersaturable SMEDD Formulation of Canagliflozin: Improved Bioavailability and Anti-diabetic Activity
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Title
Polymeric Precipitation Inhibitor–Based Solid Supersaturable SMEDD Formulation of Canagliflozin: Improved Bioavailability and Anti-diabetic Activity
Authors
Keywords
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Journal
Journal of Pharmaceutical Innovation
Volume -, Issue -, Pages -
Publisher
Springer Science and Business Media LLC
Online
2020-05-19
DOI
10.1007/s12247-020-09445-1
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- (2016) Atsuo Tahara et al. JOURNAL OF PHARMACOLOGICAL SCIENCES
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