Design, synthesis, biological evaluation and molecular docking study based on novel fused pyrazolothiazole scaffold

Design, synthesis, in vitro antimicrobial evaluation and molecular docking studies of indol-2-one tagged with morpholinosulfonyl moiety as DNA gyrase inhibitors

(2020) Mohamed A. Salem et al.   BIOORGANIC CHEMISTRY

Design, synthesis, molecular docking and biological activity evaluation of some novel indole derivatives as potent anticancer active agents and apoptosis inducers

(2019) Ahmed M. Sh. El-Sharief et al.   BIOORGANIC CHEMISTRY

An Eco-friendly Synthesis and Biological Screening of Fused Heterocyclic Compounds Containing a Thiophene Moiety via Gewald Reaction

(2019) Mohamed A. El-Borai et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

One-pot synthesis and molecular docking of some new spiropyranindol-2-one derivatives as immunomodulatory agents and in vitro antimicrobial potential with DNA gyrase inhibitor

(2019) Mohamed A. Salem et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design, synthesis, antiproliferative activity, molecular docking and cell cycle analysis of some novel (morpholinosulfonyl) isatins with potential EGFR inhibitory activity

(2018) Yousry A. Ammar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Microwave Assisted Synthesis of Fused Thiazoles in Multicomponent System and Theirin vitroAntitumor, Antioxidant, and Antimicrobial Activities

(2016) Mohamed A. El-Borai et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Synthesis and antimicrobial activity of novel 2-substituted benzimidazole, benzoxazole and benzothiazole derivatives

(2016) Vikas S. Padalkar et al.   Arabian Journal of Chemistry

Synthesis and biological evaluation of compounds which contain pyrazole, thiazole and naphthalene ring as antitumor agents

(2014) Ji-Wen Yuan et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Microwave-assisted synthesis of some new pyrazolopyridines and their antioxidant, antitumor and antimicrobial activities

(2013) Mohamed A. El-Borai et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of some new pyrazole-based 1,3-thiazoles and 1,3,4-thiadiazoles as anticancer agents

(2013) Kamal M. Dawood et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Muscarine, imidaozle, oxazole and thiazole alkaloids

(2013) Zhong Jin   NATURAL PRODUCT REPORTS

Synthesis and Antimicrobial Evaluation of Pyrazo-thiazoles

(2012) Harun Patel et al.   Letters in Drug Design & Discovery

Co(II), Cd(II), Hg(II) and U(VI)O2 complexes of o-hydroxyacetophenone[N-(3-hydroxy-2-naphthoyl)] hydrazone: Physicochemical study, thermal studies and antimicrobial activity

(2012) R.R. Zaky et al.   SPECTROCHIMICA ACTA PART A-MOLECULAR AND BIOMOLECULAR SPECTROSCOPY

Synthesis of pyrazolo[3,4-b]pyridines under microwave irradiation in multi-component reactions and their antitumor and antimicrobial activities – Part 1

(2011) M.A. El-borai et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Discovery of pyrazolthiazoles as novel and potent inhibitors of bacterial gyrase

(2010) Steven M. Ronkin et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Reevaluating Cathepsin D as a biomarker for breast cancer: Serum activity levels versus histopathology

(2010) Daniel E Abbott et al.   CANCER BIOLOGY & THERAPY

Synthesis and antimicrobial activity of some new thiazole, thiophene and pyrazole derivatives containing benzothiazole moiety

(2010) Samir Bondock et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Regiocontrolled Synthesis of Ring-Fused Thieno[2,3-c]pyrazoles through 1,3-Dipolar Cycloaddition of Nitrile Imines with Sulfur-Based Acetylenes

(2010) Jay Zumbar Chandanshive et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis, antitumor evaluation, molecular modeling and quantitative structure–activity relationship (QSAR) of some novel arylazopyrazolodiazine and triazine analogs

(2009) Ahmed El-Shafei et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Antiproliferative and Proapoptotic Activities of a New Class of Pyrazole Derivatives in HL-60 Cells

(2009) Maria Anzaldi et al.   CHEMISTRY & BIODIVERSITY

Synthesis and antiviral activity of new pyrazole and thiazole derivatives

(2009) Osama I. El-Sabbagh et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and antimicrobial activities of novel 1,5-diaryl pyrazoles

(2009) R. Venkat Ragavan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and preliminary evaluation of some substituted coumarins as anticonvulsant agents

(2008) Kamelia M. Amin et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Cathepsin D—Many functions of one aspartic protease

(2008) Petr Benes et al.   CRITICAL REVIEWS IN ONCOLOGY HEMATOLOGY

Synthesis of some novel 2,4-disubstituted thiazoles as possible antimicrobial agents

(2007) Prakash Karegoudar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and antifungal activity of some new 3-hydroxy-2-(1-phenyl-3-aryl-4-pyrazolyl) chromones

(2007) Om Prakash et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY