Discovery and Structure-Based Optimization of Potent and Selective WD Repeat Domain 5 (WDR5) Inhibitors Containing a Dihydroisoquinolinone Bicyclic Core

Title
Discovery and Structure-Based Optimization of Potent and Selective WD Repeat Domain 5 (WDR5) Inhibitors Containing a Dihydroisoquinolinone Bicyclic Core
Authors
Keywords
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Journal
JOURNAL OF MEDICINAL CHEMISTRY
Volume 63, Issue 2, Pages 656-675
Publisher
American Chemical Society (ACS)
Online
2019-12-20
DOI
10.1021/acs.jmedchem.9b01608

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