Discovery of Benzo[cd]indol-2(1H)-ones and Pyrrolo[4,3,2-de]quinolin-2(1H)-ones as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain with Potential High Efficiency against Acute Gouty Arthritis

Title
Discovery of Benzo[cd]indol-2(1H)-ones and Pyrrolo[4,3,2-de]quinolin-2(1H)-ones as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain with Potential High Efficiency against Acute Gouty Arthritis
Authors
Keywords
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Journal
JOURNAL OF MEDICINAL CHEMISTRY
Volume 62, Issue 24, Pages 11080-11107
Publisher
American Chemical Society (ACS)
Online
2019-12-02
DOI
10.1021/acs.jmedchem.9b01010

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