Phosphinic Dehydrodipeptides: Diversification of the P1′ Residue with the Morita–Baylis–Hillman Acetates and Inhibition of Alanyl Aminopeptidases

The Rational Design of Therapeutic Peptides for Aminopeptidase N using a Substrate-Based Approach

(2017) Shilvi Joshi et al.   Scientific Reports

Probing the Mechanism of Allylic Substitution of Morita-Baylis-Hillman Acetates (MBHAs) by using the Silyl Phosphonite Paradigm: Scope and Applications of a Versatile Transformation

(2015) Maria Kalyva et al.   CHEMISTRY-A EUROPEAN JOURNAL

Structure-Guided, Single-Point Modifications in the Phosphinic Dipeptide Structure Yield Highly Potent and Selective Inhibitors of Neutral Aminopeptidases

(2014) Stamatia Vassiliou et al.   JOURNAL OF MEDICINAL CHEMISTRY

The X-ray Crystal Structure of Human Aminopeptidase N Reveals a Novel Dimer and the Basis for Peptide Processing

(2012) Alan H. M. Wong et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Synthesis and Modifications of Phosphinic Dipeptide Analogues

(2012) Artur Mucha   MOLECULES

Remarkable Potential of the α-Aminophosphonate/Phosphinate Structural Motif in Medicinal Chemistry

(2011) Artur Mucha et al.   JOURNAL OF MEDICINAL CHEMISTRY

Diastereoselective Synthesis of the Leu-Pro Type Phosphinyl Dipeptide Isostere

(2011) Takehiro Yamagishi et al.   JOURNAL OF ORGANIC CHEMISTRY

Plasmodium falciparum neutral aminopeptidases: new targets for anti-malarials

(2009) Tina S. Skinner-Adams et al.   TRENDS IN BIOCHEMICAL SCIENCES