Straightforward access to N-trifluoromethyl amides, carbamates, thiocarbamates and ureas

Optimization of the Synthesis of Flavone–Amino Acid and Flavone–Dipeptide Hybrids via Buchwald–Hartwig Reaction

(2017) Dávid Pajtás et al.   JOURNAL OF ORGANIC CHEMISTRY

N-Trifluoromethylation of Nitrosoarenes with Sodium Triflinate

(2017) Angela van der Werf et al.   ORGANIC LETTERS

Efficient Synthesis of Trifluoromethyl Amines through a Formal Umpolung Strategy from the Bench-Stable Precursor (Me4 N)SCF3

(2016) Thomas Scattolin et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Big Data from Pharmaceutical Patents: A Computational Analysis of Medicinal Chemists’ Bread and Butter

(2016) Nadine Schneider et al.   JOURNAL OF MEDICINAL CHEMISTRY

Analysis of Past and Present Synthetic Methodologies on Medicinal Chemistry: Where Have All the New Reactions Gone?

(2015) Dean G. Brown et al.   JOURNAL OF MEDICINAL CHEMISTRY

Rethinking amide bond synthesis

(2011) Vijaya R. Pattabiraman et al.   NATURE

Facile Formation ofN-Acyl-oxazolidinone Derivatives Using Acid Fluorides

(2010) Corinna S. Schindler et al.   ORGANIC LETTERS

Toward the Synthesis of the RareN-(Trifluoromethyl)amides and theN-(Difluoromethylene)-N-(trifluoromethyl)amines [RN(CF3)CF2R′] Using BrF3

(2009) Youlia Hagooly et al.   JOURNAL OF ORGANIC CHEMISTRY

N-Methylation of Peptides: A New Perspective in Medicinal Chemistry

(2008) Jayanta Chatterjee et al.   ACCOUNTS OF CHEMICAL RESEARCH

Amide bond formation: beyond the myth of coupling reagents

(2008) Eric Valeur et al.   CHEMICAL SOCIETY REVIEWS

Peptidomimetics, a synthetic tool of drug discovery

(2008) Josef Vagner et al.   CURRENT OPINION IN CHEMICAL BIOLOGY

Fluorine in medicinal chemistry

(2007) Sophie Purser et al.   CHEMICAL SOCIETY REVIEWS