Synthesis of Aminoboronic Acid Derivatives from Amines and Amphoteric Boryl Carbonyl Compounds

A Qualitative Analysis of a “Bora-Brook Rearrangement”: The Ambident Reactivity of Boryl-Substituted Alkoxide Including the Carbon-to-Oxygen Migration of a Boryl Group

(2016) Haruki Kisu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Boron-selective reactions as powerful tools for modular synthesis of diverse complex molecules

(2015) Liang Xu et al.   CHEMICAL SOCIETY REVIEWS

Synthesis of Boron- and Silicon-Containing Amino Acids through Copper-Catalysed Conjugate Additions to Dehydroalanine Derivatives

(2015) Francesca Bartoccini et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A General Method for Interconversion of Boronic Acid Protecting Groups: Trifluoroborates as Common Intermediates

(2015) Quentin I. Churches et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Chemically and Configurationally Stable Monofluoro Acylboronates: Effect of Ligand Structure on their Formation, Properties, and Reactivities

(2015) Hidetoshi Noda et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Asymmetric Synthesis of α-Aminoboronic Acid Derivatives by Copper-Catalyzed Enantioselective Hydroamination

(2015) Daiki Nishikawa et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

N–B dative bond-induced [3.3.0] bicyclic boronate-tethered exo-selective intramolecular Diels–Alder reaction

(2015) Chao Feng et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Condensation-Driven Assembly of Boron-Containing Bis(Heteroaryl) Motifs Using a Linchpin Approach

(2015) Shinya Adachi et al.   ORGANIC LETTERS

Synthesis of many different types of organic small molecules using one automated process

(2015) J. Li et al.   SCIENCE

Air- and Moisture-Stable Amphoteric Molecules: Enabling Reagents in Synthesis

(2014) Zhi He et al.   ACCOUNTS OF CHEMICAL RESEARCH

An Organotrifluoroborate for Broadly Applicable One-Step18F-Labeling

(2014) Zhibo Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Site-Differentiated Polyboron Arenes Prepared by Direct CH Borylation and Their Highly Selective Suzuki-Miyaura Cross-Coupling Reactions

(2014) Liang Xu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Reagent for the One-Step Preparation of Potassium Acyltrifluoroborates (KATs) from Aryl- and Heteroarylhalides

(2014) Gábor Erős et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

n-Alkylboronic Acid Inhibitors Reveal Determinants of Ligand Specificity in the Quorum-Quenching and Siderophore Biosynthetic Enzyme PvdQ

(2014) Kenneth D. Clevenger et al.   BIOCHEMISTRY

Boron-Containing Enamine and Enamide Linchpins in the Synthesis of Nitrogen Heterocycles

(2014) Jeffrey D. St. Denis et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A high-throughput, multiplexed assay for superfamily-wide profiling of enzyme activity

(2014) Daniel A Bachovchin et al.   Nature Chemical Biology

Development of the Direct Suzuki–Miyaura Cross-Coupling of Primary B-Alkyl MIDA-boronates and Aryl Bromides

(2014) Jeffrey D. St. Denis et al.   ORGANIC LETTERS

Synthesis and chemoselective ligations of MIDA acylboronates with O-Me hydroxylamines

(2014) Hidetoshi Noda et al.   Chemical Science

Boronic Esters in Asymmetric Synthesis

(2013) Donald S. Matteson   JOURNAL OF ORGANIC CHEMISTRY

Syntheses and anti-tubercular activity ofβ-substituted andα,β-disubstituted peptidylβ-aminoboronates and boronic acids

(2013) Alexey S. Gorovoy et al.   JOURNAL OF PEPTIDE SCIENCE

Catalytic Enantioselective One-pot Aminoborylation of Aldehydes: A Strategy for Construction of Nonracemic α-Amino Boronates

(2013) Kai Hong et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

End-to-end conformational communication through a synthetic purinergic receptor by ligand-induced helicity switching

(2013) Robert A. Brown et al.   Nature Chemistry

A β-Boronopeptide Bundle of Known Structure As a Vehicle for Polyol Recognition

(2013) Michael S. Melicher et al.   ORGANIC LETTERS

[3,3]-Sigmatropic Rearrangement of Boronated Allylcyanates: A New Route to α-Aminoboronate Derivatives and Trisubstituted Tetrahydrofurans

(2013) Sabrina Touchet et al.   ORGANIC LETTERS

Oxidative Geminal Functionalization of Organoboron Compounds

(2012) Zhi He et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Boron Containing Compounds as Protease Inhibitors

(2012) Reem Smoum et al.   CHEMICAL REVIEWS

Boronate-Mediated Biologic Delivery

(2012) Gregory A. Ellis et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Versatile Scaffold for Site-Specific Modification of Cyclic Tetrapeptides

(2012) Christopher J. White et al.   ORGANIC LETTERS

Potassium Boc-Protected Secondary Aminomethyltrifluoroborates: Synthesis and Suzuki–Miyaura Cross-Coupling Reactions

(2012) Gary A. Molander et al.   ORGANIC LETTERS

Synthesis of Acyltrifluoroborates

(2012) Aaron M. Dumas et al.   ORGANIC LETTERS

Preparation and Properties of (Hydroxymethyl)boronic Acid and its Pinanediol Ester

(2011) Donald S. Matteson   AUSTRALIAN JOURNAL OF CHEMISTRY

N-Methyliminodiacetate (MIDA): A Useful Protecting Group for the Generation of Complex Organoboron Compounds

(2011) Quentin I. Churches   AUSTRALIAN JOURNAL OF CHEMISTRY

Aminoboronic acids and esters: from synthetic challenges to the discovery of unique classes of enzyme inhibitors

(2011) Sabrina Touchet et al.   CHEMICAL SOCIETY REVIEWS

One-Pot Reductive Amination and Suzuki–Miyaura Cross-Coupling of Formyl Aryl and Heteroaryl MIDA Boronates in Array Format

(2011) Jonathan E. Grob et al.   JOURNAL OF ORGANIC CHEMISTRY

Amphoteric α-Boryl Aldehydes

(2011) Zhi He et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Pinene-Derived Iminodiacetic Acid (PIDA): A Powerful Ligand for Stereoselective Synthesis and Iterative Cross-Coupling of C(sp3) Boronate Building Blocks

(2011) Junqi Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Mechanistic Insights into Direct Amide Bond Formation Catalyzed by Boronic Acids: Halogens as Lewis Bases

(2010) Tommaso Marcelli   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Novel macrocyclic HCV NS3 protease inhibitors derived from α-amino cyclic boronates

(2010) Xianfeng Li et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of an Acyltrifluoroborate and Its Fusion with Azides To Form Amides

(2010) Gary A. Molander et al.   JOURNAL OF ORGANIC CHEMISTRY

Macrocyclization of Linear Peptides Enabled by Amphoteric Molecules

(2010) Ryan Hili et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of Amidomethyltrifluoroborates and Their Use in Cross-Coupling Reactions

(2010) Gary A. Molander et al.   ORGANIC LETTERS

Synthesis of Aminoboronic Acids and Their Applications in Bifunctional Catalysis

(2009) Irene Georgiou et al.   ACCOUNTS OF CHEMICAL RESEARCH

Chemoselectivity and the Curious Reactivity Preferences of Functional Groups

(2009) Nicholas A. Afagh et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and NMR properties of novel 5,6-dihydroborauracil derivatives

(2009) Tomasz Ruman et al.   BIOORGANIC CHEMISTRY

A General Solution for Unstable Boronic Acids: Slow-Release Cross-Coupling from Air-Stable MIDA Boronates

(2009) David M. Knapp et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Suzuki–Miyaura Cross-Coupling Reactions of Alkylboronic Acid Derivatives or Alkyltrifluoroborates with Aryl, Alkenyl or Alkyl Halides and Triflates

(2008) Henri Doucet   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Functionalization of Organotrifluoroborates: Reductive Amination

(2008) Gary A. Molander et al.   JOURNAL OF ORGANIC CHEMISTRY

Multistep Synthesis of Complex Boronic Acids from Simple MIDA Boronates

(2008) Eric P. Gillis et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Asymmetric Copper-Catalyzed Synthesis of α-Amino Boronate Esters fromN-tert-Butanesulfinyl Aldimines

(2008) Melissa A. Beenen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY