Design and synthesis of new imidazo[1,2-b]pyrazole derivatives, in vitro α-glucosidase inhibition, kinetic and docking studies

Evaluation of α -glucosidase inhibiting potentials with docking calculations of synthesized arylidene-pyrazolones

(2018) Faryal Chaudhry et al.   BIOORGANIC CHEMISTRY

Design, synthesis and in vitro α-glucosidase inhibition of novel dihydropyrano[3,2-c]quinoline derivatives as potential anti-diabetic agents

(2018) Hamideh Nikookar et al.   BIOORGANIC CHEMISTRY

Design, synthesis, docking study, α-glucosidase inhibition, and cytotoxic activities of acridine linked to thioacetamides as novel agents in treatment of type 2 diabetes

(2018) Maryam Mohammadi-Khanaposhtani et al.   BIOORGANIC CHEMISTRY

New 6-amino-pyrido[2,3- d ]pyrimidine-2,4-diones as novel agents to treat type 2 diabetes: A simple and efficient synthesis, α -glucosidase inhibition, molecular modeling and kinetic study

(2018) Mehdi Adib et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Pyrano[3,2-c]quinoline derivatives as new class of α-glucosidase inhibitors to treat type 2 diabetes: synthesis, in vitro biological evaluation and kinetic study

(2018) Zahra Heydari et al.   Medicinal Chemistry

A review on tacrine-based scaffolds as multi-target drugs (MTDLs) for Alzheimer's disease

(2017) Bilqees Sameem et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

The therapeutic voyage of pyrazole and its analogs: A review

(2016) Mohemmed Faraz Khan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of Novel Tacrine Analogs as Acetylcholinesterase Inhibitors

(2016) Mohammad Mahdavi et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Efficient three-step synthesis of benzo[e]imidazo[1,2-c][1,2,3]triazines

(2016) Hedieh Pilali et al.   SYNTHETIC COMMUNICATIONS

Synthesis and biological evaluation of 1,3,4,5-tetrasubstituted pyrazole derivatives

(2016) Hoda Yahyavi et al.   ZEITSCHRIFT FUR NATURFORSCHUNG SECTION B-A JOURNAL OF CHEMICAL SCIENCES

Organocatalyzed solvent free an efficient novel synthesis of 2,4,5-trisubstituted imidazoles for α-glucosidase inhibition to treat diabetes

(2015) Muhammad Yar et al.   BIOORGANIC CHEMISTRY

Design, synthesis, in vitro cytotoxic activity evaluation, and apoptosis-induction study of new 9(10H)-acridinone-1,2,3-triazoles

(2015) Maryam Mohammadi-Khanaposhtani et al.   MOLECULAR DIVERSITY

Synthesis of new benzo[f]imidazo[1,2-d][1,4]oxazepines: AgNO3-mediated intramolecular hydroamination

(2015) Mohammad Mahdavi et al.   TETRAHEDRON LETTERS

Sulfamic acid-functionalized hydroxyapatite-encapsulated γ-Fe2O3 nanoparticles as a magnetically recoverable catalyst for synthesis of N-fused imidazole-quinoline conjugates under solvent-free conditions

(2015) Arash Mouradzadegun et al.   RSC Advances

Facile, novel and efficient synthesis of new pyrazolo[3,4-b]pyridine products from condensation of pyrazole-5-amine derivatives and activated carbonyl groups

(2015) A. Ghaedi et al.   RSC Advances

Imidazo[2,1-b]thiazole derivatives as new inhibitors of 15-lipoxygenase

(2014) Maliheh Barazandeh Tehrani et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

New imidazo[1,2-b]pyrazoles as anticancer agents: Synthesis, biological evaluation and structure activity relationship analysis

(2014) Sandrine Grosse et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and anticancer activity of acyl thioureas bearing pyrazole moiety

(2013) İrfan Koca et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Design, synthesis and biological evaluation of novel hybrid compounds of imidazole scaffold-based 2-benzylbenzofuran as potent anticancer agents

(2013) Xue-Quan Wang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Antinociceptive, anti-inflammatory and antipyretic effects of 1.5-diphenyl-1H-Pyrazole-3-carbohydrazide, a new heterocyclic pyrazole derivative

(2013) David do Carmo Malvar et al.   LIFE SCIENCES

Comprehensive Review in Current Developments of Imidazole-Based Medicinal Chemistry

(2013) Ling Zhang et al.   MEDICINAL RESEARCH REVIEWS

Hydroxycoumarin Derivatives: Novel and Potent α-Glucosidase Inhibitors

(2010) Qiong Shen et al.   JOURNAL OF MEDICINAL CHEMISTRY

New di- and triorganotin(IV) complexes of tripodal Schiff base ligand containing three imidazole arms: Synthesis, structural characterization, anti-inflammatory activity and thermal studies

(2010) Mala Nath et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

Synthesis and antitubercular screening of imidazole derivatives☆

(2009) Jyoti Pandey et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

One-pot synthesis and antibacterial activities of pyrazolo[4′,3′:5,6]pyrido[2,3-d]pyrimidine-dione derivatives

(2008) Ayoob Bazgir et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, antimicrobial and antiviral evaluation of substituted imidazole derivatives

(2008) Deepika Sharma et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design of Annulated Pyrazoles as Inhibitors of HIV-1 Reverse Transcriptase∥

(2008) Zachary K. Sweeney et al.   JOURNAL OF MEDICINAL CHEMISTRY

Discovery of novel α-glucosidase inhibitors based on the virtual screening with the homology-modeled protein structure

(2007) Hwangseo Park et al.   BIOORGANIC & MEDICINAL CHEMISTRY