Direct C(sp 2 )−H Amination to Synthesize Primary 3-aminoquinoxalin-2(1H )-ones under Simple and Mild Conditions

Metal- and Base-Free Room-Temperature Amination of Organoboronic Acids with N -Alkyl Hydroxylamines

(2018) Hong-Bao Sun et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-catalyzed Direct C-3 Benzylation of Quinoxalin-2(1H)-ones with Methylarenes under Microwave Irradiation

(2018) Leqian Hu et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of dibenzothiazines from sulfides by one-pot N,O-transfer and intramolecular C–H amination

(2018) Yan-Na Ma et al.   GREEN CHEMISTRY

Cobalt(II)-Catalyzed Electrooxidative C–H Amination of Arenes with Alkylamines

(2018) Xinlong Gao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Quinoxalinone as a Privileged Platform in Drug Development

(2018) Leilei Shi et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Metal-free oxidative coupling of quinoxalin-2(1H)-ones with arylaldehydes leading to 3-acylated quinoxalin-2(1H)-ones

(2018) Jin-Wei Yuan et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Persulfate-promoted oxidative C–N bond coupling of quinoxalinones and NH-sulfoximines

(2018) Ladawan Sumunnee et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Catalyst-Directed Chemoselective Double Amination of Bromo-chloro(hetero)arenes: A Synthetic Route toward Advanced Amino-aniline Intermediates

(2018) Alexandre A. Mikhailine et al.   ORGANIC LETTERS

Manganese-Catalyzed ortho-C-H Amidation of Weakly Coordinating Aromatic Ketones

(2018) Xianqiang Kong et al.   ORGANIC LETTERS

Direct C–H Cyanoalkylation of Quinoxalin-2(1H)-ones via Radical C–C Bond Cleavage

(2018) Lin Yang et al.   ORGANIC LETTERS

Visible light photoredox-catalyzed phosphorylation of quinoxalin-2(1 H )-ones

(2018) Yubin Kim et al.   TETRAHEDRON LETTERS

Mn(OAc) 3 *2H 2 O promoted addition of arylboronic acids to quinoxalin-2-ones

(2018) Boora Ramesh et al.   TETRAHEDRON LETTERS

Copper mediated C–H amination with oximes: en route to primary anilines

(2018) Lin-Lin Xu et al.   Chemical Science

Bisphosphines: A Prominent Ancillary Ligand Class for Application in Nickel-Catalyzed C–N Cross-Coupling

(2018) Christopher M. Lavoie et al.   ACS Catalysis

Metal-free aerobic oxidative direct C–H amination of electron-deficient alkenes via photoredox catalysis

(2018) Jing-Rui Xin et al.   Organic Chemistry Frontiers

Metal-free direct oxidative C–C bond coupling of pyrazolones and quinoxalinones

(2018) Saowanee Toonchue et al.   Organic Chemistry Frontiers

Photocatalyst-free Photoredox Arylation of Quinoxalin-2(1H )-Ones with Aryldiazo Sulfones

(2018) Hye Im Jung et al.   BULLETIN OF THE KOREAN CHEMICAL SOCIETY

Direct Synthesis of Primary Anilines via Nickel-mediated C(sp 2 )-H Aminations

(2018) Lin Yu et al.   ADVANCED SYNTHESIS & CATALYSIS

Direct C−H Trifluoromethylation of Quinoxalin-2(1H )-ones under Transition-Metal-Free Conditions

(2018) Liping Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

Manganese-Catalyzed C−H Amidation of Heteroarenes in Water

(2018) Xianqiang Kong et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of β-Trifluoromethylated Alkyl Azides via a Manganese-Catalyzed Trifluoromethylazidation of Alkenes with CF3 SO2 Na and TMSN3

(2018) Yuecheng Zhang et al.   ADVANCED SYNTHESIS & CATALYSIS

Transition-Metal-Free Decarboxylation of 3,3,3-Trifluoro-2,2-dimethylpropanoic Acid for the Preparation of C(CF3)Me2-Containing Heteroarenes

(2018) Shuai Liu et al.   ORGANIC LETTERS

A renaissance of ligand-to-metal charge transfer by cerium photocatalysis

(2018) Rong Zhao et al.   Organic Chemistry Frontiers

Transition-metal-free direct C-3 alkylation of quinoxalin-2(1H)-ones with ethers

(2018) Jinwei Yuan et al.   Organic Chemistry Frontiers

[3+2] Cyclization of Azidotrimethylsilane with Quinoxalin-2(1H )-Ones to Synthesize Tetrazolo[1,5-a ]quinoxalin-4(5H )-Ones

(2018) Qiming Yang et al.   ADVANCED SYNTHESIS & CATALYSIS

Metal-Free C(sp2)–H/N–H Cross-Dehydrogenative Coupling of Quinoxalinones with Aliphatic Amines under Visible-Light Photoredox Catalysis

(2018) Wei Wei et al.   ORGANIC LETTERS

Iodine-Catalyzed C–N Bond Formation: Synthesis of 3-Aminoquinoxalinones under Ambient Conditions

(2017) Abhishek Gupta et al.   JOURNAL OF ORGANIC CHEMISTRY

Organocatalytic Direct N-Acylation of Amides with Aldehydes under Oxidative Conditions

(2017) Chenguang Zheng et al.   JOURNAL OF ORGANIC CHEMISTRY

Silver-catalyzed decarboxylative acylation of quinoxalin-2(1H)-ones with α-oxo-carboxylic acids

(2017) Xiaobao Zeng et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper(II)-Catalyzed Oxidative Coupling of Anilines, Methyl Arenes, and TMSN3 via C(sp3/sp2)–H Functionalization and C–N Bond Formation

(2017) Devulapally Mahesh et al.   ORGANIC LETTERS

Radical Enamination of Vinyl Azides: Direct Synthesis of N-Unprotected Enamines

(2017) Yongquan Ning et al.   ORGANIC LETTERS

Nickel-Catalyzed Synthesis of Primary Aryl and Heteroaryl Amines via C–O Bond Cleavage

(2017) Huifeng Yue et al.   ORGANIC LETTERS

Copper-Assisted Direct Nitration of Cyclic Ketones with Ceric Ammonium Nitrate for the Synthesis of Tertiary α-Nitro-α-substituted Scaffolds

(2017) Zhi-Qiang Zhang et al.   ORGANIC LETTERS

Transition-Metal-Free Direct C–H Arylation of Quinoxalin-2(1H)-ones with Diaryliodonium Salts at Room Temperature

(2017) Kun Yin et al.   ORGANIC LETTERS

Diastereoselective Radical Oxidative C–H Aminations toward Chiral Atropoisomeric (P, N) Ligand Precursors

(2017) Yan-Na Ma et al.   ORGANIC LETTERS

Transition-Metal-Catalyzed Monoarylation of Ammonia

(2017) Johannes Schranck et al.   ACS Catalysis

Copper-mediated C(sp3)–H azidation with Me3SiN3: synthesis of imidazoles from ketones and aldehydes

(2016) Zeqiang Xie et al.   CHEMICAL COMMUNICATIONS

Direct phosphonation of quinoxalin-2(1H)-ones under transition-metal-free conditions

(2016) Ming Gao et al.   CHEMICAL COMMUNICATIONS

Applications of Palladium-Catalyzed C–N Cross-Coupling Reactions

(2016) Paula Ruiz-Castillo et al.   CHEMICAL REVIEWS

Fe-Catalyzed Amination of (Hetero)Arenes with a Redox-Active Aminating Reagent under Mild Conditions

(2016) Jianzhong Liu et al.   CHEMISTRY-A EUROPEAN JOURNAL

A Metal and Base-Free Chemoselective Primary Amination of Boronic Acids Using Cyanamidyl/Arylcyanamidyl Radical as Aminating Species: Synthesis and Mechanistic Studies by Density Functional Theory

(2016) Nachiketa Chatterjee et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal-Free Radical Oxidative Cyclization of o-Azidoaryl Acetylenic Ketones with Sulfinic Acids To Access Sulfone-Containing 4-Quinolones

(2016) Nengneng Zhou et al.   JOURNAL OF ORGANIC CHEMISTRY

Photocatalytic Hydrogen-Evolution Cross-Couplings: Benzene C–H Amination and Hydroxylation

(2016) Yi-Wen Zheng et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-catalysed oxidative amination of quinoxalin-2(1H)-ones with aliphatic amines

(2016) Yi Li et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Direct and Practical Synthesis of Primary Anilines through Iron-Catalyzed C–H Bond Amination

(2016) Luca Legnani et al.   ACS Catalysis

Copper-mediated C(sp3)–H amination in a multiple C–N bond-forming strategy for the synthesis of N-heterocycles

(2016) Zeqiang Xie et al.   Organic Chemistry Frontiers

Nickel-Catalyzed Monoarylation of Ammonia

(2015) Andrey Borzenko et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Nickel-Catalyzed Amination of Aryl Chlorides with Ammonia or Ammonium Salts

(2015) Rebecca A. Green et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rhodium-Catalyzed Regioselective Direct C-H Amidation of 2,4-Diarylquinazoline with Sulfonyl Azides: An Example of Steric Hindrance Regulated Mono- and Diamidation Selectivity

(2015) Chunyan Zhang et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Direct Transformation of Secondary Allylic and Benzylic Alcohols into Azides and Amides: An Efficient Utility of Azide as a Nitrogen Source

(2015) Balaji V. Rokade et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Amination–Oxidation Strategy for the Copper-Catalyzed Synthesis of Monoarylamines

(2015) Christopher Thomas et al.   JOURNAL OF ORGANIC CHEMISTRY

Transition-Metal-Free Access to Primary Anilines from Boronic Acids and a Common +NH2 Equivalent.

(2015) Samantha Voth et al.   JOURNAL OF ORGANIC CHEMISTRY

Assembly of Primary (Hetero)Arylamines via CuI/Oxalic Diamide-Catalyzed Coupling of Aryl Chlorides and Ammonia

(2015) Mengyang Fan et al.   ORGANIC LETTERS

Synthesis of 4-Ynamides and Cyclization by the Vilsmeier Reagent to Dihydrofuran-2(3H)-ones

(2015) Zhaocheng Zhang et al.   ORGANIC LETTERS

Site-selective arene C-H amination via photoredox catalysis

(2015) N. A. Romero et al.   SCIENCE

Ceric Ammonium Nitrate (CAN)–Catalyzed Multicomponent Reactions: An Efficient Catalyst for Green Organic Synthesis

(2015) Neelam P. Prajapati et al.   SYNTHETIC COMMUNICATIONS

Catalytic Methods for Aromatic C–H Amination: An Ideal Strategy for Nitrogen-Based Functional Molecules

(2015) Jiao Jiao et al.   ACS Catalysis

Assisted Tandem Palladium(II)/Palladium(0)-Catalyzed C- and N-Arylations of Quinoxalin-2(1 H)-ones in Water

(2014) Amandine Carrër et al.   ADVANCED SYNTHESIS & CATALYSIS

Ruthenium-Catalyzed C7 Amidation of Indoline CH Bonds with Sulfonyl Azides

(2014) Changduo Pan et al.   CHEMISTRY-A EUROPEAN JOURNAL

Iridium-Catalyzed Phosphoramidation of Arene C–H Bonds with Phosphoryl Azide

(2014) Changduo Pan et al.   JOURNAL OF ORGANIC CHEMISTRY

Advances in the Chemistry of Quinoxalinone Derivatives

(2014) Leilei Shi et al.   MINI-REVIEWS IN ORGANIC CHEMISTRY

Ceric Ammonium Nitrate (CAN) Catalyzed Modification of Ketones via Two C–C Bond Cleavages with the Retention of the Oxo-Group

(2014) Peng Feng et al.   ORGANIC LETTERS

Copper-Catalyzed C(sp2)–H Amidation with Azides as Amino Sources

(2014) Jiangling Peng et al.   ORGANIC LETTERS

(NH4)2Ce(NO3)6 as an inexpensive, eco-friendly, efficient catalyst for the synthesis of 5-substituted 1-H tetrazoles from nitriles

(2014) Satyanand Kumar et al.   TETRAHEDRON LETTERS

Copper-mediated C(sp2)–H amination using TMSN3 as a nitrogen source: redox-neutral access to primary anilines

(2014) Jiangling Peng et al.   Organic Chemistry Frontiers

Electrochemical C–H Amination: Synthesis of Aromatic Primary Amines via N-Arylpyridinium Ions

(2013) Tatsuya Morofuji et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A palladium-catalyzed coupling of 3-chloroquinoxalinones with various nitrogen-containing nucleophiles

(2013) Etienne Brachet et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Palladium(II)-Catalyzed Oxidative Arylation of Quinoxalin-2(1H)-ones with Arylboronic Acids

(2013) Amandine Carrër et al.   ORGANIC LETTERS

Functionalizations of Aryl CH Bonds in 2-Arylpyridines via Sequential Borylation and Copper Catalysis

(2012) Liting Niu et al.   ADVANCED SYNTHESIS & CATALYSIS

An Efficient Synthesis of Quinoxalinone Derivatives as Potent Inhibitors of Aldose Reductase

(2012) Yanchun Yang et al.   ChemMedChem

Copper-Catalyzed C–H Azidation of Anilines under Mild Conditions

(2012) Conghui Tang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis and applications of Fe3O4-diisopropylaminoacetamide as a versatile and reusable magnetic nanoparticle supported N,N-diisopropylethylamine equivalent

(2012) Parintip Rattanaburi et al.   TETRAHEDRON LETTERS

CuI-Nanoparticles-Catalyzed Selective Synthesis of Phenols, Anilines, and Thiophenols from Aryl Halides in Aqueous Solution

(2011) Hua-Jian Xu et al.   JOURNAL OF ORGANIC CHEMISTRY

Cerium(IV) Ammonium Nitrate as a Catalyst in Organic Synthesis

(2010) Vellaisamy Sridharan et al.   CHEMICAL REVIEWS

Copper-Mediated Reductive Amination of Aryl Halides with Trimethylsilyl Azide

(2010) Yasunari Monguchi et al.   CHEMISTRY-A EUROPEAN JOURNAL

Part I: Synthesis, cancer chemopreventive activity and molecular docking study of novel quinoxaline derivatives

(2010) Shadia A. Galal et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

An Efficient Copper-Catalyzed Amination of Aryl Halides by Aqueous Ammonia

(2009) Deping Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

Room-Temperature Copper-Catalyzed Carbon-Nitrogen Coupling of Aryl Iodides and Bromides Promoted by Organic Ionic Bases

(2009) Chu-Ting Yang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Easy Copper-Catalyzed Synthesis of Primary Aromatic Amines by Couplings Aromatic Boronic Acids with Aqueous Ammonia at Room Temperature

(2009) Honghua Rao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A General Palladium-Catalyzed Amination of Aryl Halides with Ammonia

(2009) Thomas Schulz et al.   CHEMISTRY-A EUROPEAN JOURNAL

A Very Simple Copper-Catalyzed Synthesis of Anilines by Employing Aqueous Ammonia

(2008) Ning Xia et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Ammonium salts as an inexpensive and convenient nitrogen source in the Cu-catalyzed amination of aryl halides at room temperature

(2008) Jinho Kim et al.   CHEMICAL COMMUNICATIONS

Fragment Based Design of New H4Receptor−Ligands with Anti-inflammatory Properties in Vivo

(2008) Rogier A. Smits et al.   JOURNAL OF MEDICINAL CHEMISTRY

Copper-Catalyzed Synthesis of Primary Arylamines via Cascade Reactions of Aryl Halides with Amidine Hydrochlorides

(2008) Xiaoting Gao et al.   JOURNAL OF ORGANIC CHEMISTRY

Oxidative alkylamination of azinones as a direct route to aminoazinones: study of some condensed diazinones

(2007) Anna V. Gulevskaya et al.   TETRAHEDRON