Multiple Roles of the Pyrimidyl Group in the Rhodium-Catalyzed Regioselective Synthesis and Functionalization of Indole-3-carboxylic Acid Esters

Substrate Activation Strategies in Rhodium(III)-Catalyzed Selective Functionalization of Arenes

(2015) Guoyong Song et al.   ACCOUNTS OF CHEMICAL RESEARCH

Direct and Site-Selective Palladium-Catalyzed C-7 Acylation of Indolines with Aldehydes

(2015) Youngmi Shin et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of Heterocycle-fused PyridineN-Oxides from Oximes and Diazo CompoundsviaRhIII-Catalyzed CH Activation and Annulation

(2015) Peng Sun et al.   ADVANCED SYNTHESIS & CATALYSIS

Cobalt(III)-Catalyzed Directed CH Coupling with Diazo Compounds: Straightforward Access towards Extended π-Systems

(2015) Dongbing Zhao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rh(iii)-catalyzed C–H activation/cyclization of benzamides and diazo compounds to form isocoumarins and α-pyrones

(2015) Xing Guang Li et al.   CHEMICAL COMMUNICATIONS

Neoechinulin B and its analogues as potential entry inhibitors of influenza viruses, targeting viral hemagglutinin

(2015) Xueqing Chen et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Rh(III)-Catalyzed C–H Amidation of Indoles with Isocyanates

(2015) Taejoo Jeong et al.   JOURNAL OF ORGANIC CHEMISTRY

Rhodium Catalyzed C2-Selective Cyanation of Indoles and Pyrroles

(2015) Manthena Chaitanya et al.   JOURNAL OF ORGANIC CHEMISTRY

Rhodium-Catalyzed C–H Activation of Phenacyl Ammonium Salts Assisted by an Oxidizing C–N Bond: A Combination of Experimental and Theoretical Studies

(2015) Songjie Yu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of Cinnolin-3(2H)-one Derivatives from Rh-Catalyzed Reaction of Azobenzenes with Diazotized Meldrum’s Acid

(2015) Jeong-Yu Son et al.   ORGANIC LETTERS

Realized C–H Functionalization of Aryldiazo Compounds via Rhodium Relay Catalysis

(2015) Lin Qiu et al.   ORGANIC LETTERS

Mild and Efficient One-Pot Synthesis of 2-(Perfluoroalkyl)indoles by Means of Sequential Michael-Type Addition and Pd(II)-Catalyzed Cross-Dehydrogenative Coupling (CDC) Reaction

(2015) Dandan Shen et al.   ORGANIC LETTERS

Rhodium(iii)-catalyzed C2-selective carbenoid functionalization and subsequent C7-alkenylation of indoles

(2014) Jingjing Shi et al.   CHEMICAL COMMUNICATIONS

Rh(iii)-catalyzed synthesis of 1-aminoindole derivatives from 2-acetyl-1-arylhydrazines and diazo compounds in water

(2014) Yujie Liang et al.   CHEMICAL COMMUNICATIONS

Arene C–H functionalisation using a removable/modifiable or a traceless directing group strategy

(2014) Fengzhi Zhang et al.   CHEMICAL SOCIETY REVIEWS

Regioselective Introduction of Heteroatoms at the C-8 Position of Quinoline N-Oxides: Remote C–H Activation Using N-Oxide as a Stepping Stone

(2014) Heejun Hwang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Formal Carbene Insertion into C–C Bond: Rh(I)-Catalyzed Reaction of Benzocyclobutenols with Diazoesters

(2014) Ying Xia et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rhodium(iii)-catalyzed formal oxidative [4 + 1] cycloaddition of benzohydroxamic acids and α-diazoesters. A facile synthesis of functionalized benzolactams

(2014) Hon-Wah Lam et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Rhodium(III)-Catalyzed C–C Bond Formation of Quinoline N-Oxides at the C-8 Position under Mild Conditions

(2014) Jisu Jeong et al.   ORGANIC LETTERS

Solvent-Controlled Switchable C–H Alkenylation of 4-Aryl-1H-pyrrole-3-carboxylates: Application to the Total Synthesis of (±)-Rhazinilam

(2014) Youla Su et al.   ORGANIC LETTERS

Rhodium(III)-Catalyzed C–C Coupling of Arenes with 2-Vinyloxiranes: Synthesis of Allylic Alcohols

(2014) Songjie Yu et al.   ORGANIC LETTERS

A General, Practical Palladium-Catalyzed Cyanation of (Hetero)Aryl Chlorides and Bromides

(2013) Todd D. Senecal et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Functionalization of C(sp2)H and C(sp3)H Bonds by Using Bidentate Directing Groups

(2013) Guy Rouquet et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rh(III)-Catalyzed Synthesis of Multisubstituted Isoquinoline and Pyridine N-Oxides from Oximes and Diazo Compounds

(2013) Zhuangzhi Shi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Coupling of Benzamides and Donor/Acceptor Diazo Compounds To Form γ-Lactams via Rh(III)-Catalyzed C–H Activation

(2013) Todd K. Hyster et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rhodium-Catalyzed Intermolecular Oxidative Cross-Coupling of (Hetero)Arenes with Chalcogenophenes

(2013) Vutukuri Prakash Reddy et al.   ORGANIC LETTERS

Rhodium Catalyzed Cyanation of Chelation Assisted C–H Bonds

(2013) Manthena Chaitanya et al.   ORGANIC LETTERS

Rh(iii)-catalyzed C–H activation/[4 + 3] cycloaddition of benzamides and vinylcarbenoids: facile synthesis of azepinones

(2013) Sunliang Cui et al.   Chemical Science

Diazo Compounds and N-Tosylhydrazones: Novel Cross-Coupling Partners in Transition-Metal-Catalyzed Reactions

(2012) Qing Xiao et al.   ACCOUNTS OF CHEMICAL RESEARCH

The Combined C–H Functionalization/Cope Rearrangement: Discovery and Applications in Organic Synthesis

(2012) Huw M. L. Davies et al.   ACCOUNTS OF CHEMICAL RESEARCH

Controlling Site Selectivity in Palladium-Catalyzed C–H Bond Functionalization

(2012) Sharon R. Neufeldt et al.   ACCOUNTS OF CHEMICAL RESEARCH

Transition-Metal-Catalyzed Enantioselective Heteroatom–Hydrogen Bond Insertion Reactions

(2012) Shou-Fei Zhu et al.   ACCOUNTS OF CHEMICAL RESEARCH

Pd(ii)-catalyzed direct C5-arylation of azole-4-carboxylates through double C–H bond cleavage

(2012) Ziyuan Li et al.   CHEMICAL COMMUNICATIONS

A General Synthesis of Indole-3-carboxylic Esters by Palladium-Catalyzed Direct Oxidative Carbonylation of 2-Alkynylaniline Derivatives

(2012) Bartolo Gabriele et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Pd(0)-Catalyzed Decarboxylative Coupling and Tandem C–H Arylation/Decarboxylation for the Synthesis of Heteroaromatic Biaryls

(2012) Debkumar Nandi et al.   JOURNAL OF ORGANIC CHEMISTRY

Rh-Catalyzed Intermolecular Carbenoid Functionalization of Aromatic C–H Bonds by α-Diazomalonates

(2012) Wai-Wing Chan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthetic Studies toward Lapidilectine-Type Kopsia Alkaloids

(2012) Erica E. Schultz et al.   ORGANIC LETTERS

Synthesis of 3-Carboxylated Indoles through a Tandem Process Involving Cyclization of 2-Ethynylanilines Followed by CO2 Fixation in the Absence of Transition Metal Catalysts

(2012) Kiyofumi Inamoto et al.   ORGANIC LETTERS

Efficient Construction of Fused Indolines with a 2-Quaternary Center via an Intramolecular Heck Reaction with a Low Catalyst Loading

(2012) Lei Zhao et al.   ORGANIC LETTERS

Versatile Synthesis of Isocoumarins and α-Pyrones by Ruthenium-Catalyzed Oxidative C–H/O–H Bond Cleavages

(2012) Lutz Ackermann et al.   ORGANIC LETTERS

Cationic Ruthenium(II) Catalysts for Oxidative C–H/N–H Bond Functionalizations of Anilines with Removable Directing Group: Synthesis of Indoles in Water

(2012) Lutz Ackermann et al.   ORGANIC LETTERS

Rhodium Catalyzed Chelation-Assisted C–H Bond Functionalization Reactions

(2011) Denise A. Colby et al.   ACCOUNTS OF CHEMICAL RESEARCH

Weak Coordination as a Powerful Means for Developing Broadly Useful C–H Functionalization Reactions

(2011) Keary M. Engle et al.   ACCOUNTS OF CHEMICAL RESEARCH

Grandilodines A−C, Biologically Active Indole Alkaloids fromKopsia grandifolia

(2011) Wai-Sum Yap et al.   JOURNAL OF NATURAL PRODUCTS

Rapid, robust, clean, catalyst-free synthesis of 2-halo-3-carboxyindoles

(2011) Aaron R. Kunzer et al.   TETRAHEDRON LETTERS

Multicomponent Cascade Reactions: A Novel and Expedient Approach to Functionalized Indoles by an Unprecedented Nucleophilic Addition-Heterocyclization-Oxidative Alkoxycarbonylation Sequence

(2010) Bartolo Gabriele et al.   ADVANCED SYNTHESIS & CATALYSIS

Arylation of α-Chiral Ketones by Palladium-Catalyzed Cross-Coupling Reactions of Tosylhydrazones with Aryl Halides

(2010) José Barluenga et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Substituted Indole from 2-Aminobenzaldehyde through [1,2]-Aryl Shift

(2010) Patrick Levesque et al.   JOURNAL OF ORGANIC CHEMISTRY

Iridium-Catalyzed, Silyl-Directed Borylation of Nitrogen-Containing Heterocycles

(2010) Daniel W. Robbins et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Insertion of α-Diazoesters into Vinyl Halides To Generate α,β-Unsaturated γ-Amino Esters

(2009) Romas Kudirka et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Indoles from Simple Anilines and Alkynes: Palladium-Catalyzed CH Activation Using Dioxygen as the Oxidant

(2009) Zhuangzhi Shi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Carbene Insertion into C−H Bonds

(2009) Michael P. Doyle et al.   CHEMICAL REVIEWS

Structural Optimization and Biological Evaluation of 2-Substituted 5-Hydroxyindole-3-carboxylates as Potent Inhibitors of Human 5-Lipoxygenase

(2009) Eva-Maria Karg et al.   JOURNAL OF MEDICINAL CHEMISTRY

One-pot synthesis of N-methylindoles from N-methylanilines and of benzofurans from phenols using transition-metal carbene X–H insertion reactions

(2009) Mark A. Honey et al.   TETRAHEDRON

Palladium-Catalyzed Oxidative Cyclization ofN-Aryl Enamines: From Anilines to Indoles

(2008) Sebastian Würtz et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Characteristics of arbidol-resistant mutants of influenza virus: Implications for the mechanism of anti-influenza action of arbidol

(2008) Irina A. Leneva et al.   ANTIVIRAL RESEARCH

Arbidol: A Broad-Spectrum Antiviral Compound that Blocks Viral Fusion

(2008) Y. Boriskin et al.   CURRENT MEDICINAL CHEMISTRY

Synthesis of 1-Amino-1H-indole-3-carboxylates by Copper(I)-Catalyzed Intramolecular Amination of Aryl Bromides

(2008) Ferdinand Melkonyan et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of N-Substituted Indole-3-carboxylic Acid Derivatives via Cu(I)-Catalyzed Intramolecular Amination of Aryl Bromides

(2008) Ferdinand S. Melkonyan et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Indole-3-carboxylic Acid Derivatives by Pd(0)-Catalyzed Intramolecular α-Arylation of β-(2-Iodoanilino) Esters

(2008) Daniel Solé et al.   JOURNAL OF ORGANIC CHEMISTRY

Catalytic C–H functionalization by metal carbenoid and nitrenoid insertion

(2008) Huw M. L. Davies et al.   NATURE

Regioselective C−H Functionalization Directed by a Removable Carboxyl Group:  Palladium-Catalyzed Vinylation at the Unusual Position of Indole and Related Heteroaromatic Rings

(2008) Atsushi Maehara et al.   ORGANIC LETTERS

Palladium-Catalyzed Synthesis of 3-Indolecarboxylic Acid Derivatives

(2008) Björn Söderberg et al.   SYNTHESIS-STUTTGART

Recent studies on the reactions of α-diazocarbonyl compounds

(2008) Zhenhua Zhang et al.   TETRAHEDRON